Zobrazeno 1 - 10 of 215 pro vyhledávání: '"Cellupica, E."'
1
Akademický článek
Mechanistic and Structural Insights on Difluoromethyl-1,3,4-oxadiazole Inhibitors of HDAC6.
Autor: Cellupica E; Research and Development, Italfarmaco Group, 20092 Milan, Italy., Gaiassi A; Research and Development, Italfarmaco Group, 20092 Milan, Italy., Rocchio I; Research and Development, Italfarmaco Group, 20092 Milan, Italy., Rovelli G; Research and Development, Italfarmaco Group, 20092 Milan, Italy., Pomarico R; Research and Development, Italfarmaco Group, 20092 Milan, Italy., Sandrone G; Research and Development, Italfarmaco Group, 20092 Milan, Italy., Caprini G; Research and Development, Italfarmaco Group, 20092 Milan, Italy., Cordella P; Research and Development, Italfarmaco Group, 20092 Milan, Italy., Cukier C; Department of Biochemistry, Selvita S.A., 30-394 Kraków, Poland., Fossati G; Research and Development, Italfarmaco Group, 20092 Milan, Italy., Marchini M; Research and Development, Italfarmaco Group, 20092 Milan, Italy., Bebel A; Department of Biochemistry, Selvita S.A., 30-394 Kraków, Poland., Airoldi C; Department of Biotechnology and Biosciences, University of Milano-Bicocca, 20126 Milan, Italy., Palmioli A; Department of Biotechnology and Biosciences, University of Milano-Bicocca, 20126 Milan, Italy., Stevenazzi A; Research and Development, Italfarmaco Group, 20092 Milan, Italy., Steinkühler C; Research and Development, Italfarmaco Group, 20092 Milan, Italy., Vergani B; Research and Development, Italfarmaco Group, 20092 Milan, Italy.
Publikováno v: International journal of molecular sciences [Int J Mol Sci] 2024 May 28; Vol. 25 (11). Date of Electronic Publication: 2024 May 28.
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2
Akademický článek
The Importance of the "Time Factor" for the Evaluation of Inhibition Mechanisms: The Case of Selected HDAC6 Inhibitors.
Autor: Cellupica E; Research and Development, Italfarmaco Group, Via dei Lavoratori 54, 20092 Cinisello Balsamo, Italy., Caprini G; Research and Development, Italfarmaco Group, Via dei Lavoratori 54, 20092 Cinisello Balsamo, Italy., Fossati G; Research and Development, Italfarmaco Group, Via dei Lavoratori 54, 20092 Cinisello Balsamo, Italy., Mirdita D; Department of Biosciences, University of Milan, Via Celoria 26, 20133 Milano, Italy., Cordella P; Research and Development, Italfarmaco Group, Via dei Lavoratori 54, 20092 Cinisello Balsamo, Italy., Marchini M; Research and Development, Italfarmaco Group, Via dei Lavoratori 54, 20092 Cinisello Balsamo, Italy., Rocchio I; Research and Development, Italfarmaco Group, Via dei Lavoratori 54, 20092 Cinisello Balsamo, Italy., Sandrone G; Research and Development, Italfarmaco Group, Via dei Lavoratori 54, 20092 Cinisello Balsamo, Italy., Stevenazzi A; Research and Development, Italfarmaco Group, Via dei Lavoratori 54, 20092 Cinisello Balsamo, Italy., Vergani B; Research and Development, Italfarmaco Group, Via dei Lavoratori 54, 20092 Cinisello Balsamo, Italy., Steinkühler C; Research and Development, Italfarmaco Group, Via dei Lavoratori 54, 20092 Cinisello Balsamo, Italy., Vanoni MA; Department of Biosciences, University of Milan, Via Celoria 26, 20133 Milano, Italy.
Publikováno v: Biology [Biology (Basel)] 2023 Jul 26; Vol. 12 (8). Date of Electronic Publication: 2023 Jul 26.
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3
Akademický článek
Difluoromethyl-1,3,4-oxadiazoles are slow-binding substrate analog inhibitors of histone deacetylase 6 with unprecedented isotype selectivity.
Autor: Cellupica E; Research and Development, Italfarmaco Group, Cinisello Balsamo, Italy., Caprini G; Research and Development, Italfarmaco Group, Cinisello Balsamo, Italy., Cordella P; Research and Development, Italfarmaco Group, Cinisello Balsamo, Italy., Cukier C; Department of Biochemistry, Selvita S.A., Kraków, Poland., Fossati G; Research and Development, Italfarmaco Group, Cinisello Balsamo, Italy., Marchini M; Research and Development, Italfarmaco Group, Cinisello Balsamo, Italy., Rocchio I; Research and Development, Italfarmaco Group, Cinisello Balsamo, Italy., Sandrone G; Research and Development, Italfarmaco Group, Cinisello Balsamo, Italy., Vanoni MA; Department of Biosciences, University of Milan, Milan, Italy., Vergani B; Research and Development, Italfarmaco Group, Cinisello Balsamo, Italy., Źrubek K; Department of Biochemistry, Selvita S.A., Kraków, Poland., Stevenazzi A; Research and Development, Italfarmaco Group, Cinisello Balsamo, Italy., Steinkühler C; Research and Development, Italfarmaco Group, Cinisello Balsamo, Italy. Electronic address: C.Steinkuhler@Italfarmacogroup.com.
Publikováno v: The Journal of biological chemistry [J Biol Chem] 2023 Jan; Vol. 299 (1), pp. 102800. Date of Electronic Publication: 2022 Dec 15.
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5
Akademický článek
HDAC6 inhibition disrupts HDAC6-P300 interaction reshaping the cancer chromatin landscape.
Autor: Zamperla, Michela Gottardi1 (AUTHOR), Illi, Barbara2 (AUTHOR), Barbi, Veronica1 (AUTHOR), Cencioni, Chiara3 (AUTHOR), Santoni, Daniele3 (AUTHOR), Gagliardi, Stella4 (AUTHOR), Garofalo, Maria4 (AUTHOR), Zingale, Gabriele Antonio5 (AUTHOR), Pandino, Irene5 (AUTHOR), Sbardella, Diego5 (AUTHOR), Cipolla, Lina6 (AUTHOR), Sabbioneda, Simone6 (AUTHOR), Farsetti, Antonella3 (AUTHOR), Ripamonti, Chiara7 (AUTHOR), Fossati, Gianluca7 (AUTHOR), Steinkühler, Christian7 (AUTHOR), Gaetano, Carlo1 (AUTHOR) carlo.gaetano@icsmaugeri.it, Atlante, Sandra3 (AUTHOR)
Publikováno v: Clinical Epigenetics. 8/20/2024, Vol. 16 Issue 1, p1-20. 20p.
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6
Akademický článek
Novel Benzohydroxamate-Based Potent and Selective Histone Deacetylase 6 (HDAC6) Inhibitors Bearing a Pentaheterocyclic Scaffold: Design, Synthesis, and Biological Evaluation.
Autor: Vergani B; Preclinical R&D , Italfarmaco Group , Via dei Lavoratori 54 , I-20092 Cinisello Balsamo , Milan , Italy., Sandrone G; Preclinical R&D , Italfarmaco Group , Via dei Lavoratori 54 , I-20092 Cinisello Balsamo , Milan , Italy., Marchini M; Preclinical R&D , Italfarmaco Group , Via dei Lavoratori 54 , I-20092 Cinisello Balsamo , Milan , Italy., Ripamonti C; Preclinical R&D , Italfarmaco Group , Via dei Lavoratori 54 , I-20092 Cinisello Balsamo , Milan , Italy., Cellupica E; Preclinical R&D , Italfarmaco Group , Via dei Lavoratori 54 , I-20092 Cinisello Balsamo , Milan , Italy., Galbiati E; Preclinical R&D , Italfarmaco Group , Via dei Lavoratori 54 , I-20092 Cinisello Balsamo , Milan , Italy., Caprini G; Preclinical R&D , Italfarmaco Group , Via dei Lavoratori 54 , I-20092 Cinisello Balsamo , Milan , Italy., Pavich G; Preclinical R&D , Italfarmaco Group , Via dei Lavoratori 54 , I-20092 Cinisello Balsamo , Milan , Italy., Porro G; Preclinical R&D , Italfarmaco Group , Via dei Lavoratori 54 , I-20092 Cinisello Balsamo , Milan , Italy., Rocchio I; Preclinical R&D , Italfarmaco Group , Via dei Lavoratori 54 , I-20092 Cinisello Balsamo , Milan , Italy., Lattanzio M; Preclinical R&D , Italfarmaco Group , Via dei Lavoratori 54 , I-20092 Cinisello Balsamo , Milan , Italy., Pezzuto M; Preclinical R&D , Italfarmaco Group , Via dei Lavoratori 54 , I-20092 Cinisello Balsamo , Milan , Italy., Skorupska M; Preclinical R&D , Italfarmaco Group , Via dei Lavoratori 54 , I-20092 Cinisello Balsamo , Milan , Italy., Cordella P; Preclinical R&D , Italfarmaco Group , Via dei Lavoratori 54 , I-20092 Cinisello Balsamo , Milan , Italy., Pagani P; Preclinical R&D , Italfarmaco Group , Via dei Lavoratori 54 , I-20092 Cinisello Balsamo , Milan , Italy., Pozzi P; Preclinical R&D , Italfarmaco Group , Via dei Lavoratori 54 , I-20092 Cinisello Balsamo , Milan , Italy., Pomarico R; Preclinical R&D , Italfarmaco Group , Via dei Lavoratori 54 , I-20092 Cinisello Balsamo , Milan , Italy., Modena D; Preclinical R&D , Italfarmaco Group , Via dei Lavoratori 54 , I-20092 Cinisello Balsamo , Milan , Italy., Leoni F; Preclinical R&D , Italfarmaco Group , Via dei Lavoratori 54 , I-20092 Cinisello Balsamo , Milan , Italy., Perego R; Preclinical R&D , Italfarmaco Group , Via dei Lavoratori 54 , I-20092 Cinisello Balsamo , Milan , Italy., Fossati G; Preclinical R&D , Italfarmaco Group , Via dei Lavoratori 54 , I-20092 Cinisello Balsamo , Milan , Italy., Steinkühler C; Preclinical R&D , Italfarmaco Group , Via dei Lavoratori 54 , I-20092 Cinisello Balsamo , Milan , Italy., Stevenazzi A; Preclinical R&D , Italfarmaco Group , Via dei Lavoratori 54 , I-20092 Cinisello Balsamo , Milan , Italy.
Publikováno v: Journal of medicinal chemistry [J Med Chem] 2019 Dec 12; Vol. 62 (23), pp. 10711-10739. Date of Electronic Publication: 2019 Nov 25.
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7
Akademický článek
Vinca alkaloids and analogues as anti-cancer agents: Looking back, peering ahead.
Autor: Martino E; Department of Earth and Environmental Sciences, University of Pavia, Via S. Epifanio 14, 27100 Pavia, Italy., Casamassima G; Department of Drug Sciences, Medicinal Chemistry Section, University of Pavia, Viale Taramelli 12, 27100 Pavia, Italy., Castiglione S; Department of Drug Sciences, Medicinal Chemistry Section, University of Pavia, Viale Taramelli 12, 27100 Pavia, Italy., Cellupica E; Department of Drug Sciences, Medicinal Chemistry Section, University of Pavia, Viale Taramelli 12, 27100 Pavia, Italy., Pantalone S; Department of Drug Sciences, Medicinal Chemistry Section, University of Pavia, Viale Taramelli 12, 27100 Pavia, Italy., Papagni F; Department of Drug Sciences, Medicinal Chemistry Section, University of Pavia, Viale Taramelli 12, 27100 Pavia, Italy., Rui M; Department of Drug Sciences, Medicinal Chemistry Section, University of Pavia, Viale Taramelli 12, 27100 Pavia, Italy., Siciliano AM; Department of Drug Sciences, Medicinal Chemistry Section, University of Pavia, Viale Taramelli 12, 27100 Pavia, Italy., Collina S; Department of Drug Sciences, Medicinal Chemistry Section, University of Pavia, Viale Taramelli 12, 27100 Pavia, Italy. Electronic address: simona.collina@unipv.it.
Publikováno v: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2018 Sep 15; Vol. 28 (17), pp. 2816-2826. Date of Electronic Publication: 2018 Jun 25.
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8
Akademický článek
Novel Piperazine Derivatives of Vindoline as Anticancer Agents.
Autor: Zsoldos, Bernadett1 (AUTHOR), Nagy, Nóra1 (AUTHOR), Donkó-Tóth, Viktória1 (AUTHOR), Keglevich, Péter1 (AUTHOR), Weber, Márton2 (AUTHOR), Dékány, Miklós2 (AUTHOR), Nehr-Majoros, Andrea3,4,5 (AUTHOR), Szőke, Éva3,4,5 (AUTHOR), Helyes, Zsuzsanna3,4,5 (AUTHOR), Hazai, László1 (AUTHOR) hazai.laszlo@vbk.bme.hu
Publikováno v: International Journal of Molecular Sciences. Jul2024, Vol. 25 Issue 14, p7929. 13p.
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9
Akademický článek
Synthesis and Antiproliferative Effect of New Alkyne-Tethered Vindoline Hybrids Containing Pharmacophoric Fragments.
Autor: Ferenczi, Etelka1,2 (AUTHOR) david.papp@ttk.elte.hu, Keglevich, Péter3 (AUTHOR) keglevich.peter@vbk.bme.hu, Tayeb, Bizhar Ahmed4 (AUTHOR) drbat25@gmail.com, Minorics, Renáta4 (AUTHOR) kanizsaine.minorics.renata@szte.hu, Papp, Dávid2,5 (AUTHOR) gitta.schlosser@ttk.elte.hu, Schlosser, Gitta5 (AUTHOR), Zupkó, István4 (AUTHOR) zupko.istvan@szte.hu, Hazai, László3 (AUTHOR) hazai.laszlo@vbk.bme.hu, Csámpai, Antal1 (AUTHOR) antal.csampai@ttk.elte.hu
Publikováno v: International Journal of Molecular Sciences. Jul2024, Vol. 25 Issue 13, p7428. 20p.
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10
Akademický článek
Synthesis of Thiazolidin-4-Ones Derivatives, Evaluation of Conformation in Solution, Theoretical Isomerization Reaction Paths and Discovery of Potential Biological Targets.
Autor: Georgiou, Nikitas1 (AUTHOR) nikitage@chem.uoa.gr, Karta, Danai1 (AUTHOR) danaikarta@gmail.com, Cheilari, Antigoni2 (AUTHOR) cheilarianti@pharm.uoa.gr, Merzel, Franci3 (AUTHOR) franci.merzel@ki.si, Tzeli, Demeter4,5 (AUTHOR) tzeli@chem.uoa.gr, Vassiliou, Stamatia1 (AUTHOR) svassiliou@chem.uoa.gr, Mavromoustakos, Thomas1 (AUTHOR) tmavrom@chem.uoa.gr
Publikováno v: Molecules. Jun2024, Vol. 29 Issue 11, p2458. 19p.
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