Zobrazeno 1 - 10
of 86
pro vyhledávání: '"Castelhano, A L"'
Autor:
Stewart, Mike, Steinig, Arno G, Ma, Chienling, Song, Jian-Ping, McKibben, Bryan, Castelhano, Arlindo L, MacLennan, Stephen J
Publikováno v:
In Biochemical Pharmacology 2004 68(2):305-312
Akademický článek
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Autor:
David, Thomas K., Prashanth, Nayak K., Rajendraswami, M., Pallalu, Devendrareddy, Castelhano, Arlindo L., Kates, Michael J., Blobaum, Anna L., Jones, Carrie K., Emmitte, Kyle A., Conn, P. Jeffrey, Lindsley, Craig W.
Publikováno v:
In Tetrahedron Letters 6 September 2017 58(36):3554-3558
Publikováno v:
In Tetrahedron Letters 23 July 1999 40(30):5471-5474
Autor:
Campbell, Robert M., Cartwright, Craig, Chen, Wei, Chen, Yong, Duzic, Emir, Fu, Jian-Min, Loveland, Michelle, Manning, Ron, McKibben, Bryan, Pleiman, Christopher M., Silverman, Lauren, Trueheart, Joshua, Webb, David R., Wilkinson, Vicki, Witter, David J., Xie, Xiaobing, Castelhano, Arlindo L.
Publikováno v:
In Bioorganic & Medicinal Chemistry Letters 1999 9(16):2413-2418
Autor:
Panarese, Joseph D., Engers, Darren W., Wu, Yong-Jin, Bronson, Joanne J., Macor, John E., Chun, Aspen, Rodriguez, Alice L., Felts, Andrew S., Engers, Julie L., Loch, Matthew T., Emmitte, Kyle A., Castelhano, Arlindo L., Kates, Michael J., Nader, Michael A., Jones, Carrie K., Blobaum, Anna L., Conn, P. Jeffrey, Niswender, Colleen M., Hopkins, Corey R., Lindsley, Craig W.
Publikováno v:
ACS Medicinal Chemistry Letters; 2019, Vol. 10 Issue 3, p255-260, 6p
Publikováno v:
Tetrahedron Letters. 40:5471-5474
Tetrasubstituted thiophenes, obtained by optimizing the multi-component reaction originally developed by Gewald, served as key templates for structural diversification and semi-automated library synthesis. Conditions were developed to carry out Gewal
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::3d40633bfb111ded20db0a84400707d6
https://doi.org/10.1016/s0040-4039(99)01108-9
https://doi.org/10.1016/s0040-4039(99)01108-9
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 8:3137-3142
Spirolactam-based Pro-Pro mimetics incorporated in the consensus sequence XPpXP, lead to effective nonpeptidic ligands of SH3 domains.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7936263f987821c3e508c859bfae9846
https://doi.org/10.1016/s0960-894x(98)00577-0
https://doi.org/10.1016/s0960-894x(98)00577-0
Autor:
Xiaohong Lin, Scott M Hammond, Castelhano Arlindo L, Yiping Zhang, Michelle F. Browner, Teresa Ho, Nolan James Dewdney, Jian Jeffrey Chen
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 6:1601-1606
A novel series of hydrozamate-based inhibitors of matrix metalloproteinases containing benzimidazole and imidazole heterocyles as amide bond isosteres have been prepared. Potent inhibition (in the low nanomolar range) and selectivity (> 100-fold) can
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::e942f851518dc7708ae7b94566495a0a
https://doi.org/10.1016/s0960-894x(96)00283-1
https://doi.org/10.1016/s0960-894x(96)00283-1
Autor:
Roland J. Billedeau, Castelhano Arlindo L, Allen Krantz, Robert L. Martin, Nolan James Dewdney, Rhonda Uppington, T.J. Liak, Sheila L. Donnelly, Horne Stephen, Yuan Zhengyu, Lilia J. Kurz
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 5:1415-1420
Potent collagenase inhibitors incorporating a novel indolactam macrocycle, which are accessible by the intramolecular alkylation of N-t-Boc-L-Trp-NH(CH 2 ) 6 OTs under phase transfer conditions, show enhanced activity compared to their acyclic analog
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::82e1d14ac54c54b608da6ad96422c376
https://doi.org/10.1016/0960-894x(95)00233-j
https://doi.org/10.1016/0960-894x(95)00233-j