Zobrazeno 1 - 10
of 518
pro vyhledávání: '"Casein Kinase Idelta"'
Autor:
Harold RL; Department of Chemistry & Biochemistry, University of California Santa Cruz, Santa Cruz, CA 95064., Tulsian NK; Department of Biological Sciences, National University of Singapore, Singapore 117543, Singapore.; Merck Sharp & Dohme International GmBH (Singapore), Neuros, Singapore 138665, Singapore., Narasimamurthy R; Program in Cancer and Stem Cell Biology, Duke-National University of Singapore Medical School, Singapore 169857, Singapore., Yaitanes N; Department of Chemistry & Biochemistry, University of California Santa Cruz, Santa Cruz, CA 95064., Ayala Hernandez MG; Department of Chemistry & Biochemistry, University of California Santa Cruz, Santa Cruz, CA 95064., Lee HW; Department of Chemistry & Biochemistry, University of California Santa Cruz, Santa Cruz, CA 95064., Crosby P; Department of Chemistry & Biochemistry, University of California Santa Cruz, Santa Cruz, CA 95064., Tripathi SM; Department of Chemistry & Biochemistry, University of California Santa Cruz, Santa Cruz, CA 95064., Virshup DM; Program in Cancer and Stem Cell Biology, Duke-National University of Singapore Medical School, Singapore 169857, Singapore.; Department of Pediatrics, Duke University Medical Center, Durham, NC 27710., Partch CL; Department of Chemistry & Biochemistry, University of California Santa Cruz, Santa Cruz, CA 95064.; Center for Circadian Biology, University of California San Diego, La Jolla, CA 92093.; HHMI, University of California, Santa Cruz, CA 95064.
Publikováno v:
Proceedings of the National Academy of Sciences of the United States of America [Proc Natl Acad Sci U S A] 2024 Oct 08; Vol. 121 (41), pp. e2415567121. Date of Electronic Publication: 2024 Oct 02.
Autor:
Grieco I; Dipartimento di Scienze Chimiche e Farmaceutiche, Università degli Studi di Trieste, Via Licio Giorgieri 1, 34127 Trieste, Italy. Electronic address: ilenia.grieco@phd.units.it., Bassani D; Molecular Modeling Section (MMS), Dipartimento di Scienze del Farmaco, Università di Padova, via Marzolo 5, 35131 Padova, Italy. Electronic address: davide.bassani.1@phd.unipd.it., Trevisan L; Dipartimento di Scienze Chimiche e Farmaceutiche, Università degli Studi di Trieste, Via Licio Giorgieri 1, 34127 Trieste, Italy. Electronic address: letizia.trevisan@phd.units.it., Salmaso V; Molecular Modeling Section (MMS), Dipartimento di Scienze del Farmaco, Università di Padova, via Marzolo 5, 35131 Padova, Italy. Electronic address: veronica.salmaso@unipd.it., Cescon E; Dipartimento di Scienze Chimiche e Farmaceutiche, Università degli Studi di Trieste, Via Licio Giorgieri 1, 34127 Trieste, Italy. Electronic address: eleonora.cescon@phd.units.it., Prencipe F; Dipartimento di Scienze Chimiche e Farmaceutiche, Università degli Studi di Trieste, Via Licio Giorgieri 1, 34127 Trieste, Italy. Electronic address: filippo.prencipe@units.it., Da Ros T; Dipartimento di Scienze Chimiche e Farmaceutiche, Università degli Studi di Trieste, Via Licio Giorgieri 1, 34127 Trieste, Italy. Electronic address: daros@units.it., Martinez-Gonzalez L; Centro de Investigaciones Biologicas, CSIC, Avenida Ramiro de Maeztu 9, 28040 Madrid, Spain; Centro de investigación biomédica en red en enfermedades neurodegenerativas (CIBERNED), Instituto de Salud Carlos III, Spain. Electronic address: loretomg@cib.csic.es., Martinez A; Centro de Investigaciones Biologicas, CSIC, Avenida Ramiro de Maeztu 9, 28040 Madrid, Spain; Centro de investigación biomédica en red en enfermedades neurodegenerativas (CIBERNED), Instituto de Salud Carlos III, Spain. Electronic address: ana.martinez@csic.es., Spalluto G; Dipartimento di Scienze Chimiche e Farmaceutiche, Università degli Studi di Trieste, Via Licio Giorgieri 1, 34127 Trieste, Italy. Electronic address: spalluto@units.it., Moro S; Molecular Modeling Section (MMS), Dipartimento di Scienze del Farmaco, Università di Padova, via Marzolo 5, 35131 Padova, Italy. Electronic address: stefano.moro@unipd.it., Federico S; Dipartimento di Scienze Chimiche e Farmaceutiche, Università degli Studi di Trieste, Via Licio Giorgieri 1, 34127 Trieste, Italy. Electronic address: sfederico@units.it.
Publikováno v:
Bioorganic chemistry [Bioorg Chem] 2024 Oct; Vol. 151, pp. 107659. Date of Electronic Publication: 2024 Jul 17.
Autor:
Ko VI; Neuroscience Graduate Program, University of California, San Diego, 9500 Gilman Drive, La Jolla, CA 92093-0624, USA; Department of Neurosciences, University of California, San Diego, 9500 Gilman Drive, La Jolla, CA 92093-0624, USA., Ong K; Department of Neurosciences, University of California, San Diego, 9500 Gilman Drive, La Jolla, CA 92093-0624, USA., Cleveland DW; Department of Cellular and Molecular Medicine, University of California, San Diego, 9500 Gilman Drive, La Jolla, CA 92093-0624, USA., Yu H; Department of Cellular and Molecular Medicine, University of California, San Diego, 9500 Gilman Drive, La Jolla, CA 92093-0624, USA., Ravits JM; Department of Neurosciences, University of California, San Diego, 9500 Gilman Drive, La Jolla, CA 92093-0624, USA. Electronic address: jravits@ucsd.edu.
Publikováno v:
Neurobiology of disease [Neurobiol Dis] 2024 Jun 15; Vol. 196, pp. 106516. Date of Electronic Publication: 2024 Apr 25.
Autor:
Burger KL; Department of Tumor Biology, H. Lee Moffitt Cancer Center & Research Institute, Tampa, Florida., Fernandez MR; Department of Tumor Biology, H. Lee Moffitt Cancer Center & Research Institute, Tampa, Florida., Meads MB; Department of Malignant Hematology, H. Lee Moffitt Cancer Center & Research Institute, Tampa, Florida., Sudalagunta P; Department of Metabolism & Physiology, H. Lee Moffitt Cancer Center & Research Institute, Tampa, Florida., Oliveira PS; Department of Malignant Hematology, H. Lee Moffitt Cancer Center & Research Institute, Tampa, Florida., Renatino Canevarolo R; Department of Metabolism & Physiology, H. Lee Moffitt Cancer Center & Research Institute, Tampa, Florida., Alugubelli RR; Department of Malignant Hematology, H. Lee Moffitt Cancer Center & Research Institute, Tampa, Florida., Tungsevik A; Department of Malignant Hematology, H. Lee Moffitt Cancer Center & Research Institute, Tampa, Florida., De Avila G; Department of Malignant Hematology, H. Lee Moffitt Cancer Center & Research Institute, Tampa, Florida., Silva M; Department of Metabolism & Physiology, H. Lee Moffitt Cancer Center & Research Institute, Tampa, Florida., Graeter AI; Department of Malignant Hematology, H. Lee Moffitt Cancer Center & Research Institute, Tampa, Florida., Dai HA; Informatics Division, M2Gen®, Tampa, Florida., Vincelette ND; Department of Malignant Hematology, H. Lee Moffitt Cancer Center & Research Institute, Tampa, Florida., Prabhu A; Department of Tumor Biology, H. Lee Moffitt Cancer Center & Research Institute, Tampa, Florida., Magaletti D; Department of Tumor Biology, H. Lee Moffitt Cancer Center & Research Institute, Tampa, Florida.; Department of Malignant Hematology, H. Lee Moffitt Cancer Center & Research Institute, Tampa, Florida., Yang C; Department of Tumor Biology, H. Lee Moffitt Cancer Center & Research Institute, Tampa, Florida., Li W; Department of Tumor Biology, H. Lee Moffitt Cancer Center & Research Institute, Tampa, Florida., Kulkarni A; Informatics Division, M2Gen®, Tampa, Florida., Hampton O; Informatics Division, M2Gen®, Tampa, Florida., Koomen JM; Department of Molecular Oncology, H. Lee Moffitt Cancer Center & Research Institute, Tampa, Florida., Roush WR; Department of Chemistry, Scripps Research, Jupiter, Florida., Monastyrskyi A; Department of Drug Discovery, H. Lee Moffitt Cancer Center & Research Institute, Tampa, Florida., Berglund AE; Department of Biostatistics and Bioinformatics, H. Lee Moffitt Cancer Center & Research Institute, Tampa, Florida., Silva AS; Department of Metabolism & Physiology, H. Lee Moffitt Cancer Center & Research Institute, Tampa, Florida., Cleveland JL; Department of Tumor Biology, H. Lee Moffitt Cancer Center & Research Institute, Tampa, Florida., Shain KH; Department of Tumor Biology, H. Lee Moffitt Cancer Center & Research Institute, Tampa, Florida.; Department of Malignant Hematology, H. Lee Moffitt Cancer Center & Research Institute, Tampa, Florida.
Publikováno v:
Cancer research [Cancer Res] 2023 Dec 01; Vol. 83 (23), pp. 3901-3919.
Autor:
Francucci B; Medicinal Chemistry Unit, School of Pharmacy, University of Camerino, 62032 Camerino, Italy., Angeloni S; Medicinal Chemistry Unit, School of Pharmacy, University of Camerino, 62032 Camerino, Italy., Dal Ben D; Medicinal Chemistry Unit, School of Pharmacy, University of Camerino, 62032 Camerino, Italy., Lambertucci C; Medicinal Chemistry Unit, School of Pharmacy, University of Camerino, 62032 Camerino, Italy., Ricciutelli M; Medicinal Chemistry Unit, School of Pharmacy, University of Camerino, 62032 Camerino, Italy., Spinaci A; Medicinal Chemistry Unit, School of Pharmacy, University of Camerino, 62032 Camerino, Italy., Smirnov A; Medicinal Chemistry Unit, School of Pharmacy, University of Camerino, 62032 Camerino, Italy., Volpini R; Medicinal Chemistry Unit, School of Pharmacy, University of Camerino, 62032 Camerino, Italy., Buccioni M; Medicinal Chemistry Unit, School of Pharmacy, University of Camerino, 62032 Camerino, Italy., Marucci G; Medicinal Chemistry Unit, School of Pharmacy, University of Camerino, 62032 Camerino, Italy.
Publikováno v:
Molecules (Basel, Switzerland) [Molecules] 2023 Jun 14; Vol. 28 (12). Date of Electronic Publication: 2023 Jun 14.
Structure-Based Development of Isoform-Selective Inhibitors of Casein Kinase 1ε vs Casein Kinase 1δ.
Autor:
Choi JY; Department of Chemistry, The Scripps Research Institute, Scripps Florida, Jupiter, Florida 33458, United States.; Department of Chemistry and Biochemistry, Queens College, Queens, New York 11367, United States.; Ph.D. Programs in Chemistry and Biochemistry, The Graduate Center of the City University of New York, New York, New York 10016, United States., Noguchi Y; Department of Chemistry, The Scripps Research Institute, Scripps Florida, Jupiter, Florida 33458, United States., Alburger JM; Department of Chemistry, The Scripps Research Institute, Scripps Florida, Jupiter, Florida 33458, United States., Bayle S; Department of Drug Discovery, Moffitt Cancer Center, Tampa, Florida 33612, United States., Chung E; Department of Chemistry and Biochemistry, Queens College, Queens, New York 11367, United States., Grant W; Department of Molecular Therapeutics, The Scripps Research Institute, Scripps Florida, Jupiter, Florida 33458, United States., Chaikuad A; Institute of Pharmaceutical Chemistry, Goethe University, Frankfurt am Main 60438, Germany.; Structural Genomics Consortium, BMLS, Goethe University, Frankfurt am Main 60438, Germany., Knapp S; Institute of Pharmaceutical Chemistry, Goethe University, Frankfurt am Main 60438, Germany.; Structural Genomics Consortium, BMLS, Goethe University, Frankfurt am Main 60438, Germany., Duckett DR; Department of Drug Discovery, Moffitt Cancer Center, Tampa, Florida 33612, United States., Roush WR; Department of Chemistry, The Scripps Research Institute, Scripps Florida, Jupiter, Florida 33458, United States.
Publikováno v:
Journal of medicinal chemistry [J Med Chem] 2023 Jun 08; Vol. 66 (11), pp. 7162-7178. Date of Electronic Publication: 2023 May 19.
Autor:
Qi F; Department of Urologic Surgery, Jiangsu Cancer Hospital and Jiangsu Institute of Cancer Research and Affiliated Cancer Hospital of Nanjing Medical University, Nanjing, 210009, China., Shen W; Department of Hematology, The First Affiliated Hospital of Nanjing Medical University, Nanjing, China., Wei X; State Key Laboratory of Reproductive Medicine, Department of Urology, The First Affiliated Hospital of Nanjing Medical University, Nanjing, 210029, China., Cheng Y; Department of Urology, The First Affiliated Hospital of Nanjing Medical University, Nanjing, 210029, China., Xu F; Jiangsu Cancer Hospital & Jiangsu Institute of Cancer Research & Affiliated Cancer Hospital of Nanjing Medical University, Nanjing, 210009, China., Zheng Y; Department of Urologic Surgery, Jiangsu Cancer Hospital and Jiangsu Institute of Cancer Research and Affiliated Cancer Hospital of Nanjing Medical University, Nanjing, 210009, China., Li L; State Key Laboratory of Translational Medicine and Innovative Drug Development, Jiangsu Simcere Diagnostics Co., Ltd, Nanjing, China.; Nanjing Simcere Medical Laboratory Science Co., Ltd, Nanjing, China., Qin C; State Key Laboratory of Reproductive Medicine, Department of Urology, The First Affiliated Hospital of Nanjing Medical University, Nanjing, 210029, China. qinchao@njmu.edu.cn., Li X; Department of Urologic Surgery, Jiangsu Cancer Hospital and Jiangsu Institute of Cancer Research and Affiliated Cancer Hospital of Nanjing Medical University, Nanjing, 210009, China. leex91@163.com.; Department of Scientific Research, Jiangsu Cancer Hospital and Jiangsu Institute of Cancer Research and Affiliated Cancer Hospital of Nanjing Medical University, Nanjing, China. leex91@163.com.
Publikováno v:
Cellular and molecular life sciences : CMLS [Cell Mol Life Sci] 2023 May 19; Vol. 80 (6), pp. 156. Date of Electronic Publication: 2023 May 19.
Autor:
Yang M; Department of Biochemistry and Molecular Biology, School of Medicine, Key Laboratory of Neuroregeneration of Jiangsu and Ministry of Education of China, Co-innovation Center of Neuroregeneration, Nantong University, Nantong, Jiangsu, China., Qi R; Department of Biochemistry and Molecular Biology, School of Medicine, Key Laboratory of Neuroregeneration of Jiangsu and Ministry of Education of China, Co-innovation Center of Neuroregeneration, Nantong University, Nantong, Jiangsu, China., Liu Y; Department of Biochemistry and Molecular Biology, School of Medicine, Key Laboratory of Neuroregeneration of Jiangsu and Ministry of Education of China, Co-innovation Center of Neuroregeneration, Nantong University, Nantong, Jiangsu, China., Shen X; Department of Biochemistry and Molecular Biology, School of Medicine, Key Laboratory of Neuroregeneration of Jiangsu and Ministry of Education of China, Co-innovation Center of Neuroregeneration, Nantong University, Nantong, Jiangsu, China., Zhao Y; Department of Biochemistry and Molecular Biology, School of Medicine, Key Laboratory of Neuroregeneration of Jiangsu and Ministry of Education of China, Co-innovation Center of Neuroregeneration, Nantong University, Nantong, Jiangsu, China., Jin N; Department of Biochemistry and Molecular Biology, School of Medicine, Key Laboratory of Neuroregeneration of Jiangsu and Ministry of Education of China, Co-innovation Center of Neuroregeneration, Nantong University, Nantong, Jiangsu, China.; Department of Neurochemistry, Inge Grundke-Iqbal Research Floor, New York State Institute for Basic Research in Developmental Disabilities, Staten Island, NY, USA., Wu R; Department of Biochemistry and Molecular Biology, School of Medicine, Key Laboratory of Neuroregeneration of Jiangsu and Ministry of Education of China, Co-innovation Center of Neuroregeneration, Nantong University, Nantong, Jiangsu, China., Liu F; Department of Neurochemistry, Inge Grundke-Iqbal Research Floor, New York State Institute for Basic Research in Developmental Disabilities, Staten Island, NY, USA., Gu J; Department of Biochemistry and Molecular Biology, School of Medicine, Key Laboratory of Neuroregeneration of Jiangsu and Ministry of Education of China, Co-innovation Center of Neuroregeneration, Nantong University, Nantong, Jiangsu, China.; Department of Neurochemistry, Inge Grundke-Iqbal Research Floor, New York State Institute for Basic Research in Developmental Disabilities, Staten Island, NY, USA.
Publikováno v:
Journal of Alzheimer's disease : JAD [J Alzheimers Dis] 2023; Vol. 91 (4), pp. 1527-1539.
Autor:
Kishino Y; Department of Neuropathology, Graduate School of Medicine, The University of Tokyo, Tokyo, Japan; Department of Pathology, Graduate School of Medicine, The University of Tokyo, Tokyo, Japan; Department of Degenerative Neurological Diseases, National Institute of Neuroscience, National Center of Neurology and Psychiatry, Kodaira, Japan., Matsukawa K; Department of Neuropathology, Graduate School of Medicine, The University of Tokyo, Tokyo, Japan., Matsumoto T; Department of Neuropathology, Graduate School of Medicine, The University of Tokyo, Tokyo, Japan., Miyazaki R; Department of Neuropathology, Graduate School of Medicine, The University of Tokyo, Tokyo, Japan; Department of Degenerative Neurological Diseases, National Institute of Neuroscience, National Center of Neurology and Psychiatry, Kodaira, Japan., Wakabayashi T; Department of Neuropathology, Graduate School of Medicine, The University of Tokyo, Tokyo, Japan; Department of Innovative Dementia Prevention, Graduate School of Medicine, The University of Tokyo, Tokyo, Japan., Nonaka T; Dementia Research Project, Tokyo Metropolitan Institute of Medical Science, Tokyo, Japan., Kametani F; Dementia Research Project, Tokyo Metropolitan Institute of Medical Science, Tokyo, Japan., Hasegawa M; Dementia Research Project, Tokyo Metropolitan Institute of Medical Science, Tokyo, Japan., Hashimoto T; Department of Neuropathology, Graduate School of Medicine, The University of Tokyo, Tokyo, Japan; Department of Degenerative Neurological Diseases, National Institute of Neuroscience, National Center of Neurology and Psychiatry, Kodaira, Japan; Department of Innovative Dementia Prevention, Graduate School of Medicine, The University of Tokyo, Tokyo, Japan. Electronic address: tonchan@ncnp.go.jp., Iwatsubo T; Department of Neuropathology, Graduate School of Medicine, The University of Tokyo, Tokyo, Japan. Electronic address: iwatsubo@m.u-tokyo.ac.jp.
Publikováno v:
The Journal of biological chemistry [J Biol Chem] 2022 Aug; Vol. 298 (8), pp. 102191. Date of Electronic Publication: 2022 Jun 24.
Autor:
Schulte AM; Stratingh Institute for Chemistry, University of Groningen, 9747 AG Groningen, The Netherlands., Kolarski D; Stratingh Institute for Chemistry, University of Groningen, 9747 AG Groningen, The Netherlands., Sundaram V; Discipline of Biological Engineering, Indian Institute of Technology Gandhinagar, Gandhinagar 382355, India., Srivastava A; Discipline of Biological Engineering, Indian Institute of Technology Gandhinagar, Gandhinagar 382355, India., Tama F; Institute of Transformative BioMolecules (WPI-ITbM), Nagoya University, Chikusa, Nagoya 464-8601, Japan.; Department of Physics, Graduate School of Science, Nagoya University, Chikusa, Nagoya 464-8602, Japan.; Computational Structural Biology Unit, RIKEN-Center for Computational Science, Chuo, Kobe 650-0047, Japan., Feringa BL; Stratingh Institute for Chemistry, University of Groningen, 9747 AG Groningen, The Netherlands., Szymanski W; Stratingh Institute for Chemistry, University of Groningen, 9747 AG Groningen, The Netherlands.; Department of Radiology, Medical Imaging Center, University Medical Center Groningen, University of Groningen, 9713 GZ Groningen, The Netherlands.
Publikováno v:
International journal of molecular sciences [Int J Mol Sci] 2022 May 10; Vol. 23 (10). Date of Electronic Publication: 2022 May 10.