Zobrazeno 1 - 10 of 12 pro vyhledávání: '"Carol Elaine Pasini"'
2
[Untitled]
Autor: Carol Elaine Pasini, Joseph M. Indelicato
Publikováno v: Pharmaceutical Research. :250-254
Loracarbef is an oral 1-carba-l-dethiacephalosporin antibiotic structurally related to cefaclor. Like many β-lactam antibiotics, loracar-bef exists in several hydrated crystalline forms. The pH–solubility profile curve for loracarbef monohydrate i
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::7a7fc4ac1c7e2e2933c06b64f0cd5f6f
https://doi.org/10.1023/a:1018949709797
Zobrazit plný text záznamu
6
3-Quaternary ammonium 1-carba-1-dethiacephems
Autor: Jeffrey S. Kasher, Joseph M. Indelicato, David A. Preston, Donald B. Boyd, G. K. Cook, J H McDonald rd, William E. Alborn, Carol Elaine Pasini, J. A. Eudaly, R Johnson
Publikováno v: Journal of Medicinal Chemistry. 32:2442-2450
A series of structurally unique 1-carba-1-dethiacephems is described. The structural stability of the 1-carba-1-dethiacephem nucleus was essential for the preparation of this series of 3-quaternary ammonium carbacephems. The known p-nitrobenzyl 7 bet
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c90b27c1c60fa4bddf02234df45371ee
https://doi.org/10.1021/jm00131a006
Zobrazit plný text záznamu
7
Heteroatom-activated .beta.-lactam antibiotics: considerations of differences in the biological activity of [[3(S)-(acylamino)-2-oxo-1-azetidinyl]oxy]acetic acids (oxamazins) and the corresponding sulfur analogs (thiamazins)
Autor: Donald B. Boyd, Carol Elaine Pasini, Charles Eigenbrot, Steven R. Woulfe, Marvin J. Miller, Joseph M. Indelicato
Publikováno v: Journal of Medicinal Chemistry. 30:528-536
The considerable antibacterial activity of [[3(S)-(acylamino)-2-oxo-1-azetidinyl]oxy]acetic acids (oxamazins) in contrast to the lack of activity of the corresponding sulfur analogues (thiamazins) is examined in terms of physicochemical parameters, i
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::62e698533525c6cd6c0335675e9b2149
https://doi.org/10.1021/jm00386a015
Zobrazit plný text záznamu
8
3-Sulfonyl-1-carba-1-dethiacephems
Autor: Basil D. Halliday, Thomas Alan Crowell, John H. McDonald, Joseph M. Indelicato, Carol Elaine Pasini, Ernie C. Y. Wu
Publikováno v: Journal of Medicinal Chemistry. 32:2436-2442
The stability of the 1-carba-1-dethiacephalosporin framework has allowed the synthesis of a range of 3-sulfonyl-1-carba-1-dethiacephems unavailable for a variety of reasons in the cephem arena. The known p-nitrobenzyl 7 beta-(phenoxyacetamido)-3-[[(t
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::dd4b45f68be0d942ad540260a76d4a07
https://doi.org/10.1021/jm00131a005
Zobrazit plný text záznamu
9
Intramolecular Nucleophilic Amino Attack in a Monobactam: Synthesis and Stability of (S,3S(-3-[(2R)-2-Amino-2-phenylacetamido[-2-methyl-4-oxo-1-Azetidinesulfonic Acid
Autor: Joseph M. Indelicato, Carol Elaine Pasini, Fisher Jack Wayne
Publikováno v: Journal of Pharmaceutical Sciences. 75:304-306
The potentially orally bioavailable arylglycine-substituted monobactam, (2S,3S)- 3-[(2R)-2-amino-2-phenylacetamido]-2-methyl-4-oxo-1- azetidinesulfonic acid, was prepared as a crystalline solid. No significant antibacterial activity [i.e., MICs were
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::c10da6984dba267196a876b9d28a9ce0
https://doi.org/10.1002/jps.2600750321
Zobrazit plný text záznamu

Vyhledávací nástroje:

Upřesnit hledání

Omezení vyhledávání
Plný text Recenzováno Digitální knihovna AV ČR
Zdroje