Zobrazeno 1 - 4
of 4
pro vyhledávání: '"Carine Binisti"'
Autor:
Jean-Edouard Ombetta, Françoise Heymans, Chang-Zhi Dong, Jean-Jacques Godfroid, Léon Assogba, Estera Touboul, Catherine Redeuilh, Carine Binisti, Jack Huet, Carine Mounier
Publikováno v:
ChemInform. 33
1-Benzoyl-2-alkyl piperazines are strong inhibitors of Group I and II secreted PLA2s. An improvement of their activity was obtained by replacing the amide function by a sulfamide and by introduction of electrodonor substituents on the para position o
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::53a2236f1aa7156e945647a3cbefc4d3
https://doi.org/10.1002/chin.200212268
https://doi.org/10.1002/chin.200212268
Autor:
Chang-Zhi Dong, Jack Huet, Françoise Heymans, Léon Assogba, Catherine Redeuilh, Carine Mounier, Carine Binisti, Estera Touboul, Jean-Edouard Ombetta, Jean-Jacques Godfroid
Publikováno v:
European journal of medicinal chemistry. 36(10)
1-Benzoyl-2-alkyl piperazines are strong inhibitors of Group I and II secreted PLA2s. An improvement of their activity was obtained by replacing the amide function by a sulfamide and by introduction of electrodonor substituents on the para position o
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c5ac7d887e9ad441ea3d58153e717547
https://pubmed.ncbi.nlm.nih.gov/11738488
https://pubmed.ncbi.nlm.nih.gov/11738488
Autor:
Carine Mounier, Carine Binisti, Cassian Bon, Estera Touboul, Françoise Heymans, Jean-Jacques Godfroid
Publikováno v:
Journal of lipid mediators and cell signalling. 16(3)
Starting from a series of compounds which were known to be PAF antagonists, we have synthesized molecules that are good inhibitors of PLA2s of groups I or II, with IC50 in the micromolar range (Binisti et al., 1997). In this report we investigate the
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::723cf5a22e41b3c992576d9285e5e943
https://pubmed.ncbi.nlm.nih.gov/9246606
https://pubmed.ncbi.nlm.nih.gov/9246606
Autor:
Françoise Heymans, Carine Mounier, Carine Binisti, Cassian Bon, Mina Aitdafoun, Jean-Jacques Godfroid
Publikováno v:
Biochemical pharmacology. 51(6)
A series of 4-alkoxybenzamidines was synthesized, varying the number of carbons of the alkyl chain, and their potency as phospholipase A2 (PLA2) inhibitors was evaluated. The relationship between their capacity to inhibit PLA2 activity and their lipo
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::3c56b1c4deec3d9078b1defb76ef28c6
https://pubmed.ncbi.nlm.nih.gov/8602868
https://pubmed.ncbi.nlm.nih.gov/8602868