Zobrazeno 1 - 3
of 3
pro vyhledávání: '"Cappelli A. 1"'
Autor:
Giuliani G. 1, Cappelli A. 1, Matarrese M. 2, 3, Masiello V. 2, Turolla E.A. 2, Monterisi C. 2, Fazio F. 3, Anzini M. 1, Pericot Mohr G.L. 1, Riitano D. 3, Finetti F. 4, Morbidelli L. 4, Ziche M. 4, Giorgi G. 5, Vomero S. 1
Publikováno v:
Bioorganic & medicinal chemistry
19 (2011): 2242–2251.
info:cnr-pdr/source/autori:Giuliani G. 1, Cappelli A. 1, Matarrese M. 2,3, Masiello V. 2,3, Turolla E.A. 2,3, Monterisi C. 2,3, Fazio F. 3, Anzini M. 1, Pericot Mohr G.L. 1, Riitano D. 3, Finetti F. 4, Morbidelli L. 4, Ziche M. 4, Giorgi G. 5, Vomero S. 1/titolo:Non-peptide NK(1) receptor ligands based on the 4-phenylpyridine moiety./doi:/rivista:Bioorganic & medicinal chemistry (Print)/anno:2011/pagina_da:2242/pagina_a:2251/intervallo_pagine:2242–2251/volume:19
19 (2011): 2242–2251.
info:cnr-pdr/source/autori:Giuliani G. 1, Cappelli A. 1, Matarrese M. 2,3, Masiello V. 2,3, Turolla E.A. 2,3, Monterisi C. 2,3, Fazio F. 3, Anzini M. 1, Pericot Mohr G.L. 1, Riitano D. 3, Finetti F. 4, Morbidelli L. 4, Ziche M. 4, Giorgi G. 5, Vomero S. 1/titolo:Non-peptide NK(1) receptor ligands based on the 4-phenylpyridine moiety./doi:/rivista:Bioorganic & medicinal chemistry (Print)/anno:2011/pagina_da:2242/pagina_a:2251/intervallo_pagine:2242–2251/volume:19
The quinoline nucleus of the previously described 4-phenylquinoline-3-carboxamides NK(1) receptor ligands 7 has been transformed into either substituted or azole-(i.e., triazole or tetrazole) fused pyridine moieties of compounds 9 and 10, respectivel
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=cnr_________::198f0595b462c82e9a680b2aaecb5b43
https://publications.cnr.it/doc/10528
https://publications.cnr.it/doc/10528
Publikováno v:
ICNDST & ADC2006 Joint Conference, Cary (NC-USA), 2006
info:cnr-pdr/source/autori:Ascarelli P.(1), Cappelli E.(1), Conte G.(2), and Trucchi D.M. (1*)./congresso_nome:ICNDST & ADC2006 Joint Conference/congresso_luogo:Cary (NC-USA)/congresso_data:2006/anno:2006/pagina_da:/pagina_a:/intervallo_pagine
info:cnr-pdr/source/autori:Ascarelli P.(1), Cappelli E.(1), Conte G.(2), and Trucchi D.M. (1*)./congresso_nome:ICNDST & ADC2006 Joint Conference/congresso_luogo:Cary (NC-USA)/congresso_data:2006/anno:2006/pagina_da:/pagina_a:/intervallo_pagine
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=cnr_________::effd5c0e08c16792dab941d066f8746c
http://www.cnr.it/prodotto/i/131415
http://www.cnr.it/prodotto/i/131415
Autor:
Cappelli A. 1, Giuliani G. 1, Gallelli A. 1, Valenti S. 1, Anzini M. 1, Mennuni L. 2, Makovec F. 2, Cupello A. 3, Vomero S. 1
Publikováno v:
Bioorganic & medicinal chemistry
13 (2005): 3455–3460.
info:cnr-pdr/source/autori:Cappelli A. 1, Giuliani G. 1, Gallelli A. 1, Valenti S. 1, Anzini M. 1, Mennuni L. 2, Makovec F. 2, Cupello A. 3, Vomero S. 1/titolo:Structure-affinity relationship studies on arylpiperazine derivatives related to quizapine as serotonin transporter ligands. Molecular basis of the selectivity SERT%2F5HT3 receptor/doi:/rivista:Bioorganic & medicinal chemistry (Print)/anno:2005/pagina_da:3455/pagina_a:3460/intervallo_pagine:3455–3460/volume:13
13 (2005): 3455–3460.
info:cnr-pdr/source/autori:Cappelli A. 1, Giuliani G. 1, Gallelli A. 1, Valenti S. 1, Anzini M. 1, Mennuni L. 2, Makovec F. 2, Cupello A. 3, Vomero S. 1/titolo:Structure-affinity relationship studies on arylpiperazine derivatives related to quizapine as serotonin transporter ligands. Molecular basis of the selectivity SERT%2F5HT3 receptor/doi:/rivista:Bioorganic & medicinal chemistry (Print)/anno:2005/pagina_da:3455/pagina_a:3460/intervallo_pagine:3455–3460/volume:13
A series of quipazine derivatives, previously synthesized to probe the 5-HT(3) receptor, was evaluated for its potential interaction with serotonin transporter (SERT). Some of them show nanomolar affinity for the rodent SERT comparable to or slightly
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=cnr_________::cd2543961f8d38abd60b6f5f7cc61891
http://www.cnr.it/prodotto/i/10153
http://www.cnr.it/prodotto/i/10153