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Autor:
Robert L. Hudkins, Joanne R. Mathiasen, Reddeppa reddy Dandu, Lisa D. Aimone, Rita Raddatz, Val R. Marcy, Greg A. Hostetler, John A. Gruner, Caitlyn Benfield, Robert J. Bendesky
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 21:6362-6365
A series of pyridazinone-phenethylamine derivatives with moderate to low nanomolar affinity for rat and human H(3)R are described. These analogs exhibited excellent selectivity and metabolic stability, with acceptable rat pharmacokinetic properties.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5059cea68a269120cb488864e8573a91
https://doi.org/10.1016/j.bmcl.2011.08.104
https://doi.org/10.1016/j.bmcl.2011.08.104
