Zobrazeno 1 - 9
of 9
pro vyhledávání: '"Brigitte Illel"'
Autor:
Caroline, Twarog, Elias, Fattal, Magali, Noiray, Brigitte, Illel, David J, Brayden, Myriam, Taverna, Hervé, Hillaireau
Publikováno v:
International journal of pharmaceutics. 626
A common approach to tackle the poor intestinal membrane permeability of peptides after oral administration is to formulate them with a permeation enhancer (PE). Increased oral bioavailability for oral peptide candidates has been reported from clinic
Autor:
David J. Brayden, Kai Liu, Kenneth A. Dawson, Caroline Twarog, Brigitte Illel, Peter J. O'Brien, Elias Fattal
Publikováno v:
European Journal of Pharmaceutics and Biopharmaceutics. 152:95-107
Salcaprozate sodium (SNAC) and sodium caprate (C10) are the two leading intestinal permeation enhancers (PEs) in oral peptide formulations in clinical trials. There is debate over their mechanism of action on intestinal epithelia. The aims were: (i)
Autor:
Caroline Twarog, Elias Fattal, Magali Noiray, Brigitte Illel, David J. Brayden, Myriam Taverna, Hervé Hillaireau
Publikováno v:
International Journal of Pharmaceutics. 626:122131
Autor:
Caroline, Twarog, Fiona, McCartney, Sabine M, Harrison, Brigitte, Illel, Elias, Fattal, David J, Brayden
Publikováno v:
European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences. 158
SNAC and C
Autor:
Caroline, Twarog, Kai, Liu, Peter J, O'Brien, Kenneth A, Dawson, Elias, Fattal, Brigitte, Illel, David J, Brayden
Publikováno v:
European journal of pharmaceutics and biopharmaceutics : official journal of Arbeitsgemeinschaft fur Pharmazeutische Verfahrenstechnik e.V. 152
Salcaprozate sodium (SNAC) and sodium caprate (C
Autor:
Torsten Haack, Laurent Hortala, Ulrich Werner, Priscilla Brun, Harivardhan Reddy Lakkireddy, Didier Bazile, Rachel Vogel, Melissa Besenius, Brigitte Illel, Matthias Urmann, Jean Alié
Publikováno v:
Advanced Drug Delivery Reviews. 106:196-222
While some orally delivered diabetes peptides are moving to late development with standard formulations incorporating functional excipients, the demonstration of the value of nanotechnology in clinic is still at an early stage. The goal of this revie
Autor:
Fiona McCartney, Sabine M. Harrison, Brigitte Illel, Elias Fattal, Caroline Twarog, David J. Brayden
Publikováno v:
European Journal of Pharmaceutical Sciences. 158:105685
SNAC and C10 are intestinal permeation enhancers (PEs) used in formulations of peptides for oral delivery in clinical trials. Our aims were to compare their: (i) mechanism of action in isolated rat intestinal mucosae mounted in Ussing chambers and in
Autor:
Brigitte Illel
Publikováno v:
Critical reviews in therapeutic drug carrier systems. 14(3)
The percutaneous administration of drug products is of current therapeutic interest, mainly with regard to reduction of hepatic metabolism and systemic toxicity, and delivery to specific sites. Hair follicles and sebaceous glands can be privileged pa
Publikováno v:
Journal of pharmaceutical sciences. 80(5)
The relative importance of stratum corneum and follicles in percutaneous absorption is not fully understood. In order to quantitatively investigate the importance of the transappendageal route, we have previously developed a model of skin without fol