Zobrazeno 1 - 6
of 6
pro vyhledávání: '"Bridgette Craig"'
Autor:
Perry Michael David, James Saenz, Kim Albizati, Sami Bahmanyar, Billie J. Kline, Mark A. Mitchell, Bridgette Craig-Woods, Nebojsa Stankovic, Shu Yu
Publikováno v:
Organic Process Research & Development. 11:30-38
A practical process for the synthesis of PPARγ agonist AG035029 was developed which involved six steps along the longest linear path. The process development utilized automated technology and compu...
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::1b6305e05034118858e1838077f3c0de
https://doi.org/10.1021/op0601621
https://doi.org/10.1021/op0601621
Autor:
Ramon J. Alabaster, Roger N. Farr, Simon A Johnson, Guo-Jie Ho, John Y. L. Chung, Bridgette Craig, Andrew W. Gibson, Guy R. Humphrey, John S Edwards, Edward J. J. Grabowski
Publikováno v:
Tetrahedron: Asymmetry. 14:3503-3515
An efficient, high yield process for the synthesis of a GnRH antagonist has been developed. We have demonstrated that under boron trifluoride mediation, nosyl aziridines will react with 2-arylindole derivatives to afford β-substituted tryptamines in
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::4c6c88ed48ed0a6d6e183872fc1b51b7
https://doi.org/10.1016/j.tetasy.2003.08.038
https://doi.org/10.1016/j.tetasy.2003.08.038
Autor:
Jing Li, David J. Mathre, Joseph F. Payack, James M. McNamara, Nancy N. Tsou, David M. Tschaen, Karel M. J. Brands, Karl B. Hansen, Paul J. Reider, Bridgette Craig, Peter G. Dormer, Mark A. Huffman, Philip J. Pye, Todd D. Nelson, Kai Rossen, Robert A. Reamer, Alexander Candelario, Jonathan D. Rosen, Christopher J. Welch, Zhiguo J. Song, Paul N. Devine, Matthew M. Zhao
Publikováno v:
Journal of the American Chemical Society. 125:2129-2135
An efficient stereoselective synthesis of the orally active NK(1) receptor antagonist Aprepitant is described. A direct condensation of N-benzyl ethanolamine with glyoxylic acid yielded a 2-hydroxy-1,4-oxazin-3-one which was activated as the correspo
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e40c18512e9aa7684b8f1a518ae347f5
https://doi.org/10.1021/ja027458g
https://doi.org/10.1021/ja027458g
Autor:
Jacqueline H. Smitrovich, Mark A. Huffman, Joseph F. Payack, Louis Matty, Jonathan D. Rosen, James M. McNamara, Todd D. Nelson, Bridgette Craig
Publikováno v:
ChemInform. 36
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::c5bef914e03678b3f12dd7a49a57a45b
https://doi.org/10.1002/chin.200517138
https://doi.org/10.1002/chin.200517138
Autor:
Mark A. Huffman, Todd D. Nelson, Jacqueline H. Smitrovich, James M. McNamara, Bridgette Craig, Joseph F. Payack, Louis Matty, Jonathan D. Rosen
Publikováno v:
Organic letters. 7(1)
The concise synthesis of a stereochemically rich hNK-1 receptor antagonist is described. The synthesis is highlighted by an S(N)2 reaction of an enantiomerically pure alpha-alkoxy sulfonate (orthogonally protected butane triol), which was prepared by
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4462c9978e0459ddd09411474381da7d
https://pubmed.ncbi.nlm.nih.gov/15624976
https://pubmed.ncbi.nlm.nih.gov/15624976
Autor:
James Saenz, Mark Mitchell, Sami Bahmanyar, Nebojsa Stankovic, Michael Perry, Bridgette Craig-Woods, Billie Kline, Shu Yu, Kim Albizati
Publikováno v:
Organic Process Research & Development; Jan2007, Vol. 11 Issue 1, p30-38, 9p