(Chlorosulfonyl)benzenesulfonyl Fluorides-Versatile Building Blocks for Combinatorial Chemistry: Design, Synthesis and Evaluation of a Covalent Inhibitor Library.

Autor: Tolmachova KA; National Taras Shevchenko University of Kyiv, Volodymyrska Street 60 , Kyiv 01601 , Ukraine.; Institute of Bioorganic Chemistry & Petrochemistry , NAS of Ukraine , Murmanska Street 1 , Kyiv 02660 , Ukraine., Moroz YS; National Taras Shevchenko University of Kyiv, Volodymyrska Street 60 , Kyiv 01601 , Ukraine.; Chemspace , Ilukstes iela 38-5 , Riga , LV-1082 , Latvia., Konovets A; National Taras Shevchenko University of Kyiv, Volodymyrska Street 60 , Kyiv 01601 , Ukraine.; Enamine Ltd. , Chervonotkatska Street 78 , Kyiv 02094 , Ukraine., Platonov MO; Enamine Ltd. , Chervonotkatska Street 78 , Kyiv 02094 , Ukraine., Vasylchenko OV; Enamine Ltd. , Chervonotkatska Street 78 , Kyiv 02094 , Ukraine., Borysko P; Bienta/Enamine Ltd. , Chervonotkatska Street 78 , Kyiv 02094 , Ukraine., Zozulya S; Bienta/Enamine Ltd. , Chervonotkatska Street 78 , Kyiv 02094 , Ukraine., Gryniukova A; Bienta/Enamine Ltd. , Chervonotkatska Street 78 , Kyiv 02094 , Ukraine., Bogolubsky AV; Enamine Ltd. , Chervonotkatska Street 78 , Kyiv 02094 , Ukraine., Pipko S; Enamine Ltd. , Chervonotkatska Street 78 , Kyiv 02094 , Ukraine., Mykhailiuk PK; National Taras Shevchenko University of Kyiv, Volodymyrska Street 60 , Kyiv 01601 , Ukraine., Brovarets VS; Institute of Bioorganic Chemistry & Petrochemistry , NAS of Ukraine , Murmanska Street 1 , Kyiv 02660 , Ukraine., Grygorenko OO; National Taras Shevchenko University of Kyiv, Volodymyrska Street 60 , Kyiv 01601 , Ukraine.; Enamine Ltd. , Chervonotkatska Street 78 , Kyiv 02094 , Ukraine.

Publikováno v: ACS combinatorial science [ACS Comb Sci] 2018 Nov 12; Vol. 20 (11), pp. 672-680. Date of Electronic Publication: 2018 Nov 01.

Expanding Synthesizable Space of Disubstituted 1,2,4-Oxadiazoles.

Autor: Tolmachev A; Enamine Ltd. , 78 Chervonotkatska Street, Kyiv, 02094, Ukraine.; ChemBioCenter, Kyiv National Taras Shevchenko University , 61 Chervonotkatska Street, Kyiv, 02094, Ukraine., Bogolubsky AV; Enamine Ltd. , 78 Chervonotkatska Street, Kyiv, 02094, Ukraine., Pipko SE; ChemBioCenter, Kyiv National Taras Shevchenko University , 61 Chervonotkatska Street, Kyiv, 02094, Ukraine.; UkrOrgSyntez Ltd. (UORSY) , 29 Schorsa Street, Kyiv, 01133, Ukraine., Grishchenko AV; Enamine Ltd. , 78 Chervonotkatska Street, Kyiv, 02094, Ukraine., Ushakov DV; Enamine Ltd. , 78 Chervonotkatska Street, Kyiv, 02094, Ukraine., Zhemera AV; Enamine Ltd. , 78 Chervonotkatska Street, Kyiv, 02094, Ukraine., Viniychuk OO; UkrOrgSyntez Ltd. (UORSY) , 29 Schorsa Street, Kyiv, 01133, Ukraine., Konovets AI; Enamine Ltd. , 78 Chervonotkatska Street, Kyiv, 02094, Ukraine.; The Institute of High Technologies, Kyiv National Taras Shevchenko University , 4 Glushkov Street, Building 5, Kyiv, 03187, Ukraine., Zaporozhets OA; Department of Chemistry, Kyiv National Taras Shevchenko University , 64 Volodymyrska Street, Kyiv, 01601, Ukraine., Mykhailiuk PK; Enamine Ltd. , 78 Chervonotkatska Street, Kyiv, 02094, Ukraine.; Department of Chemistry, Kyiv National Taras Shevchenko University , 64 Volodymyrska Street, Kyiv, 01601, Ukraine., Moroz YS; ChemBioCenter, Kyiv National Taras Shevchenko University , 61 Chervonotkatska Street, Kyiv, 02094, Ukraine.

Publikováno v: ACS combinatorial science [ACS Comb Sci] 2016 Oct 10; Vol. 18 (10), pp. 616-624. Date of Electronic Publication: 2016 Sep 07.

One-Pot Parallel Synthesis of Alkyl Sulfides, Sulfoxides, and Sulfones.

Autor: Bogolubsky AV; †Enamine, Ltd., 61 Chervonotkatska Street, Kyiv, 02094, Ukraine., Moroz YS; †Enamine, Ltd., 61 Chervonotkatska Street, Kyiv, 02094, Ukraine.; ‡ChemBioCenter, Kyiv National Taras Shevchenko University, 61 Chervonotkatska Street, Kyiv, 02094, Ukraine., Mykhailiuk PK; †Enamine, Ltd., 61 Chervonotkatska Street, Kyiv, 02094, Ukraine.; §Department of Chemistry, Kyiv National Taras Shevchenko University, 64 Volodymyrska Street, Kyiv, 01601, Ukraine., Ostapchuk EN; †Enamine, Ltd., 61 Chervonotkatska Street, Kyiv, 02094, Ukraine.; ‡ChemBioCenter, Kyiv National Taras Shevchenko University, 61 Chervonotkatska Street, Kyiv, 02094, Ukraine., Rudnichenko AV; †Enamine, Ltd., 61 Chervonotkatska Street, Kyiv, 02094, Ukraine., Dmytriv YV; †Enamine, Ltd., 61 Chervonotkatska Street, Kyiv, 02094, Ukraine., Bondar AN; §Department of Chemistry, Kyiv National Taras Shevchenko University, 64 Volodymyrska Street, Kyiv, 01601, Ukraine., Zaporozhets OA; §Department of Chemistry, Kyiv National Taras Shevchenko University, 64 Volodymyrska Street, Kyiv, 01601, Ukraine., Pipko SE; ‡ChemBioCenter, Kyiv National Taras Shevchenko University, 61 Chervonotkatska Street, Kyiv, 02094, Ukraine., Doroschuk RA; §Department of Chemistry, Kyiv National Taras Shevchenko University, 64 Volodymyrska Street, Kyiv, 01601, Ukraine., Babichenko LN; †Enamine, Ltd., 61 Chervonotkatska Street, Kyiv, 02094, Ukraine.; ‡ChemBioCenter, Kyiv National Taras Shevchenko University, 61 Chervonotkatska Street, Kyiv, 02094, Ukraine., Konovets AI; †Enamine, Ltd., 61 Chervonotkatska Street, Kyiv, 02094, Ukraine.; ∥The Institute of High Technologies, Kyiv National Taras Shevchenko University, 4 Glushkov Street, Building 5, Kyiv, 03187, Ukraine., Tolmachev A; †Enamine, Ltd., 61 Chervonotkatska Street, Kyiv, 02094, Ukraine.; ‡ChemBioCenter, Kyiv National Taras Shevchenko University, 61 Chervonotkatska Street, Kyiv, 02094, Ukraine.

Publikováno v: ACS combinatorial science [ACS Comb Sci] 2015 Jun 08; Vol. 17 (6), pp. 348-54. Date of Electronic Publication: 2015 May 13.

Bis(2,2,2-trifluoroethyl) carbonate as a condensing agent in one-pot parallel synthesis of unsymmetrical aliphatic ureas.

Autor: Bogolubsky AV; Enamine Ltd. , 23 Matrosova Street, Kyiv, 01103, Ukraine., Moroz YS, Mykhailiuk PK, Granat DS, Pipko SE, Konovets AI, Doroschuk R, Tolmachev A

Publikováno v: ACS combinatorial science [ACS Comb Sci] 2014 Jun 09; Vol. 16 (6), pp. 303-8. Date of Electronic Publication: 2014 Apr 18.

A solution-phase parallel synthesis of alkylated guanidines from thioisocyanates and amines.

Autor: Bogolubsky AV; Enamine Ltd., 23 Alexandra Matrosova Street, Kiev, 01103, Ukraine., Grishchenko A, Pipko SE, Konovets A, Chuprina A, Tolmachev A, Boyko AN, Chekotylo A, Lukin O

Publikováno v: Molecular diversity [Mol Divers] 2013 Aug; Vol. 17 (3), pp. 471-7. Date of Electronic Publication: 2013 May 01.