Zobrazeno 1 - 2
of 2
pro vyhledávání: '"Bingliu Lu"'
Publikováno v:
Bioorganicmedicinal chemistry letters. 27(21)
A series of hydroxamic acid-based HDACIs with 4-aminoquinazolinyl moieties as capping groups was profiled. Most compounds showed more potent HDACs inhibition activity than clinically used drug SAHA. Among them, compounds 5f and 5h selectively inhibit
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2a860a466adaf927a4a30a4e254a4788
https://pubmed.ncbi.nlm.nih.gov/28947154
https://pubmed.ncbi.nlm.nih.gov/28947154
Publikováno v:
Bioorganicmedicinal chemistry letters. 27(14)
The synthesis and biological evaluation of a variety of 4-piperazinyl-containing Chidamide derivatives is described. Some of these compounds were shown to inhibit HDAC1 with IC50 values below micromolar range, and inhibited proliferation of several h
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d2e2e66d05b75f3ee059734d05908a2b
https://pubmed.ncbi.nlm.nih.gov/28532668
https://pubmed.ncbi.nlm.nih.gov/28532668