Zobrazeno 1 - 6
of 6
pro vyhledávání: '"Berangere Gaucher"'
Publikováno v:
CHIMIA, Vol 57, Iss 5 (2003)
Heterocyclic compounds are an attractive source of screening library structures because they possess varied structural diversity and can exhibit potent biological activity. In this context, we present some of our new and versatile approaches to rapid
Externí odkaz:
https://doaj.org/article/c30efec8a9234b228e2d301c2dad100a
Autor:
Anne-Marie Aubertin, Jacques Greiner, Marielle Rouquayrol, Pierre Vierling, Dominique Roche, Berangere Gaucher
Publikováno v:
Org. Biomol. Chem.. 2:345-357
With the aim of improving the pharmacological properties of current protease inhibitors (PIs), the synthesis of various acyl and carbamate amino acid- or diglyceride-containing prodrugs derived from saquinavir, indinavir and nelfinavir, their in vitr
Publikováno v:
Pharmaceutical Research. 19:1704-1712
Purpose. This study is dedicated to the permeation of various amino acid-, D-glucose-, and PEG-conjugates of indinavir, saquinavir, and nelfinavir across monolayers of Caco-2 cells as models of the intestinal barrier. This screening is aimed at detec
Autor:
Marielle Rouquayrol, Berangere Gaucher, Pierre Vierling, Jacques Greiner, Roger Guedj, Anne-Marie Aubertin
Publikováno v:
ChemInform. 33
With the aim at improving the transport of the current HIV protease inhibitors across the intestinal and blood brain barriers and their penetration into the central nervous system, the synthesis of various acyl and carbamatoyl glucose-containing prod
Autor:
Pierre Vierling, Berangere Gaucher, Dominique Roche, Anne-Marie Aubertin, Marielle Rouquayrol, Jacques Greiner
Publikováno v:
ChemInform. 35
With the aim of improving the pharmacological properties of current protease inhibitors (PIs), the synthesis of various acyl and carbamate amino acid- or diglyceride-containing prodrugs derived from saquinavir, indinavir and nelfinavir, their in vitr
Autor:
Pierre Vierling, Marielle Rouquayrol, Roger Guedj, Berangere Gaucher, Anne-Marie Aubertin, Jacques Greiner
Publikováno v:
Carbohydrate research. 336(3)
With the aim at improving the transport of the current HIV protease inhibitors across the intestinal and blood brain barriers and their penetration into the central nervous system, the synthesis of various acyl and carbamatoyl glucose-containing prod