Zobrazeno 1 - 10
of 10
pro vyhledávání: '"Benzazepines/*pharmacology"'
Autor:
Mahin Abad Dar, Franziska Maiwald, Diego Benítez, Laurent Meijer, Nadège Loaëc, Conrad Kunick, Lutz Preu, Hanna Erdmann, Marcelo A. Comini, Oliver Koch, Diego Charquero, Christoph Hölscher
Publikováno v:
European Journal of Medicinal Chemistry
European Journal of Medicinal Chemistry, Elsevier, 2014, 83, pp.274-283. ⟨10.1016/j.ejmech.2014.06.020⟩
European Journal of Medicinal Chemistry, Elsevier, 2014, 83, pp.274-283. ⟨10.1016/j.ejmech.2014.06.020⟩
International audience; Trypanosomes from the "brucei" complex are pathogenic parasites endemic in sub-Saharan Africa and causative agents of severe diseases in humans and livestock. In order to identify new antitrypanosomal chemotypes against Africa
Drug dependence is a chronic brain disease characterized by recurrent episodes of relapse, even when the person is motivated to quit. Relapse is a major problem and new pharmacotherapies are needed to prevent relapse episodes. The nicotinic acetylcho
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9ac4a1d397964437ab50b62a2a6f7372
https://hdl.handle.net/20.500.14017/dea1fdfd-8553-4d68-b02f-ec00b923ed5f
https://hdl.handle.net/20.500.14017/dea1fdfd-8553-4d68-b02f-ec00b923ed5f
Publikováno v:
Pharmacological Research, vol. 61, no. 1, pp. 85-91
The hyperpolarization-activated cyclic nucleotide-gated (HCN) channels are expressed in pacemaker cells very early during cardiogenesis. This work aimed at determining to what extent these channels are implicated in the electromechanical disturbances
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::49227053769d10cd7230a73d71104145
https://serval.unil.ch/resource/serval:BIB_E2217744245B.P001/REF.pdf
https://serval.unil.ch/resource/serval:BIB_E2217744245B.P001/REF.pdf
Autor:
Spiridon Konitsiotis, E. Kafetzopoulos
Publikováno v:
European Journal of Pharmacology. 179:201-205
Naive rats were challenged systematically with apomorphine after receiving unilateral dorsal or ventral intracaudate injections of the dopamine D-1 receptor antagonist, SCH23390, or the D-2 receptor antagonist, sulpiride. Sulpiride injections into bo
Autor:
Arai Takashi, Katsunori Iwasaki, Izzettin Hatip-Al-Khatib, Nobuaki Egashira, Michihiro Fujiwara
The effects of zanapezil (TAK-147) and donepezil (E2020) on extracellular acetylcholine (ACh) levels were investigated by HPLC-microdialysis of ventral hippocampus (VH) in freely moving intact rats. The results showed that the basal ACh release rate
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1d2ecd4e43b346f6effbadb7b7830e65
http://acikerisim.pau.edu.tr:8080/xmlui/handle/11499/5088
http://acikerisim.pau.edu.tr:8080/xmlui/handle/11499/5088
Publikováno v:
Grodum, E, Andersen, M, Hangaard, J, Koldkjaer, O & Hagen, C 1998, ' Lack of effect of the dopamine D1 antagonist, NNC 01-0687, on unstimulated and stimulated release of anterior pituitary hormones in males ', Journal of Endocrinological Investigation, vol. 21, no. 5, pp. 291-297 . https://doi.org/10.1007/BF03350331
Scopus-Elsevier
Scopus-Elsevier
Dopamine in humans inhibits the secretion of luteinizing hormone (LH), follicular stimulating hormone (FSH), thyroid stimulating hormone (TSH) and prolactin (PRL), and is a stimulator of growth hormone (GH) secretion. Dopamine-D1 receptor stimulation
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f506b0c974ec648d6cfd0c5f81817a75
https://portal.findresearcher.sdu.dk/da/publications/27fb301a-ffc5-464d-a450-7f3067989491
https://portal.findresearcher.sdu.dk/da/publications/27fb301a-ffc5-464d-a450-7f3067989491
Publikováno v:
Journal of cardiovascular pharmacology. 12(6)
Under control conditions a primary culture containing about 80-90% of granular juxtaglomerular (JG) cells prepared from rat kidneys continuously released renin into the culture medium at a rate of 17.9 +/- 1.4 ng angiotensin I/h per mg of cell protei
Publikováno v:
Nature, Vol. 310, No 5973 (1984) pp. 140-1
In response to stress, adrenocorticotropic hormone (ACTH) is released by corticotrophs in the anterior pituitary under the control of several central and peripheral factors including corticotropin-releasing factor (CRF), which was recently isolated f
Publikováno v:
European journal of pharmacology. 162(3)
In human blood platelet membranes, 5-HT displaced the binding of the putative selective D-1 dopamine receptor antagonist [ 3 H]SCH 23390 in a competitive manner with a K i value of 5.7 ± 0.8 nM, which was about 1000-fold lower than the K i value for
Publikováno v:
ETSU Faculty Works.
Myeloid-derived suppressor cells (MDSCs) prolong sepsis by promoting immunosuppression. We reported that sepsis MDSC development requires long non-coding RNA Hotairm1 interactions with S100A9. Using a mouse model that simulates the immunobiology of s
Externí odkaz:
https://dc.etsu.edu/etsu-works-2/210