Zobrazeno 1 - 10
of 29
pro vyhledávání: '"Bela Ternai"'
Autor:
Gideon M. Polya, Bela Ternai, Mery Hasmeda, Wilawan Mahabusarakam, Zhe Xiong Lu, Prapaipit Chamsuksai Ternai
Publikováno v:
Chemico-Biological Interactions. 114:121-140
A series of prenylated xanthones are variously potent inhibitors of the catalytic subunit (cAK) of rat liver cyclic AMP-dependent protein kinase (PKA), rat brain Ca2+ and phospholipid-dependent protein kinase C (PKC), chicken gizzard myosin light cha
Publikováno v:
Biological Chemistry Hoppe-Seyler. 375:527-536
The phenanthrenemethanol antimalarial halofantrine is a potent inhibitor of bovine heart and rat liver cyclic AMP-dependent protein kinase catalytic subunit (cAK) (IC50 values 2.1 microM and 0.6 microM, respectively). The inhibition of rat liver cAK
Publikováno v:
Planta Medica. 59:525-528
Methanolic extracts of leaves, flowers, stems, bark, and other parts of representative plants of the Myrtaceae, specifically of the EUCALYPTUS, MELALEUCA, THRYPTOMENA, CALLISTOMEN, ACMENA, AND ANGOPHORA genera, variously contain high levels of inhibi
Publikováno v:
Biological Chemistry Hoppe-Seyler. 373:205-212
Rat liver cyclic AMP-dependent protein kinase catalytic subunit (cAK), assayed using the synthetic peptide substrate, LRRASLG, is inhibited by a range of plant-derived flavonoids. In general, maximal inhibitory effectiveness (IC50 values 1 to 2 micro
Publikováno v:
Plant Science. 78:165-175
Wheat embryo Ca2+-dependent protein kinase (CDPK) is inhibited by a variety of long chain amphiphilic compounds that also inhibit avian myosin light chain kinase (MLCK), namely by straight chain alkylamines, alkyltrimethylammonium halides and N- alky
Publikováno v:
Phytochemistry. 44(5)
The prenylated isoflavone warangalone from the insecticidal plant Derris scandens is a selective and potent inhibitor of rat liver cyclic AMP-dependent protein kinase catalytic subunit (cAK) (IC50 3.5 microM). The inhibition of rat liver cAK by waran
Publikováno v:
Biological chemistry Hoppe-Seyler. 373(9)
A variety of anthraquinone (anthracene-9,10-dione) derivatives inhibits rat brain Ca(2+)- and phospholipid-activated protein kinase C (PKC) of which the most potent inhibitors are mitoxantrone (1,4-dihydroxy-5,8-bis[2-(hydroxyethylamino)-ethylamino]-
Publikováno v:
Biological chemistry Hoppe-Seyler. 372(9)
Avian myosin light chain kinase (MLCK) is inhibited by a range of plant-derived flavonoids. Maximal inhibition requires 2,3-unsaturation and polyhydroxylation of two of the three flavonoid rings. Phosphorylation of a synthetic myosin light chain-rela
Publikováno v:
Medical Journal of Australia. 152:54-54
Autor:
Luisa Cook, Bela Ternai
Publikováno v:
Biological Chemistry Hoppe-Seyler. 370:11-20
Inhibition of human leucocyte elastase by oleic acid and the structurally related 3-(1'-oxo-7'-carboxyheptyl)-4-hydroxy-6-octyl-2-pyrone is considerably enhanced by the addition of Cu2+, Zn2+ and, to a lesser extent, Co2+ and Ca2+. Sulindac sulfide a