Zobrazeno 1 - 10
of 58
pro vyhledávání: '"Beccari AR"'
Autor:
Bertini, R, Barcelos, Ls, Beccari, Ar, Cavalieri, B, Moriconi, A, Bizzarri, C, DI BENEDETTO, Paola, Di Giacinto, C, Gloaguen, I, Galliera, E, Corsi, Mm, Russo, Rc, Andrade, Sp, Cesta, Mc, Nano, G, Aramini, A, Cutrin, Jc, Locati, M, Allegretti, M, Teixeira, Mm
Publikováno v:
British journal of pharmacology. 165(2)
Background and Purpose: DF 2156A is a new dual inhibitor of IL-8 receptors CXCR1 and CXCR2 with an optimal pharmacokinetic profile. We characterized its binding mode, molecular mechanism of action and selectivity, and evaluated its therapeutic potent
Akademický článek
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Akademický článek
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Autor:
Bertini, R, Barcelos, LS, Beccari, AR, Cavalieri, B, Moriconi, A, Bizzarri, C, Di Benedetto, P, Di Giacinto, C, Gloaguen, I, Galliera, E, Corsi, MM, Russo, RC, Andrade, SP, Cesta, MC, Nano, G, Aramini, A, Cutrin, JC, Locati, M, Allegretti, M, Teixeira, MM
Publikováno v:
British Journal of Pharmacology; Jan2012, Vol. 165 Issue 2, p436-454, 19p, 8 Graphs
Autor:
Vittorio S; Dipartimento di Scienze Farmaceutiche, Università degli Studi di Milano, Via Luigi Mangiagalli 25, I-20133 Milano, Italy., Lunghini F; EXSCALATE, Dompé Farmaceutici SpA, Via Tommaso de Amicis 95, 80123 Naples, Italy., Morerio P; Pattern Analysis and Computer Vision, Fondazione Istituto Italiano di Tecnologia, Via Morego, 30, 16163 Genova, Italy., Gadioli D; Dipartimento di Elettronica Informazione e Bioingegneria, Politecnico di Milano, Via Ponzio 34/5, I-20133 Milano, Italy., Orlandini S; SCAI, SuperComputing Applications and Innovation Department, CINECA, Via dei Tizii 6, Rome 00185, Italy., Silva P; IT4Innovations, VSB - Technical University of Ostrava, 17. listopadu 2172/15, 708 00 Ostrava-Poruba, Czech Republic., Martinovic J; IT4Innovations, VSB - Technical University of Ostrava, 17. listopadu 2172/15, 708 00 Ostrava-Poruba, Czech Republic., Pedretti A; Dipartimento di Scienze Farmaceutiche, Università degli Studi di Milano, Via Luigi Mangiagalli 25, I-20133 Milano, Italy., Bonanni D; Department of Physical and Chemical Sciences, University of L'Aquila, via Vetoio, L'Aquila 67010, Italy., Del Bue A; Pattern Analysis and Computer Vision, Fondazione Istituto Italiano di Tecnologia, Via Morego, 30, 16163 Genova, Italy., Palermo G; Dipartimento di Elettronica Informazione e Bioingegneria, Politecnico di Milano, Via Ponzio 34/5, I-20133 Milano, Italy., Vistoli G; Dipartimento di Scienze Farmaceutiche, Università degli Studi di Milano, Via Luigi Mangiagalli 25, I-20133 Milano, Italy., Beccari AR; EXSCALATE, Dompé Farmaceutici SpA, Via Tommaso de Amicis 95, 80123 Naples, Italy.
Publikováno v:
Computational and structural biotechnology journal [Comput Struct Biotechnol J] 2024 Jul 17; Vol. 23, pp. 2963. Date of Electronic Publication: 2024 Jul 17 (Print Publication: 2024).
Autor:
Vittorio S; Dipartimento di Scienze Farmaceutiche, Università degli Studi di Milano, Via Luigi Mangiagalli 25, I-20133 Milano, Italy., Lunghini F; EXSCALATE, Dompé Farmaceutici SpA, Via Tommaso de Amicis 95, 80123 Naples, Italy., Morerio P; Pattern Analysis and Computer Vision, Fondazione Istituto Italiano di Tecnologia, Via Morego, 30, 16163 Genova, Italy., Gadioli D; Dipartimento di Elettronica Informazione e Bioingegneria, Politecnico di Milano, Via Ponzio 34/5, I-20133 Milano, Italy., Orlandini S; SCAI, SuperComputing Applications and Innovation Department, CINECA, Via dei Tizii 6, Rome 00185, Italy., Silva P; IT4Innovations, VSB - Technical University of Ostrava, 17. listopadu 2172/15, 70800 Ostrava-Poruba, Czech Republic., Jan Martinovic; IT4Innovations, VSB - Technical University of Ostrava, 17. listopadu 2172/15, 70800 Ostrava-Poruba, Czech Republic., Pedretti A; Dipartimento di Scienze Farmaceutiche, Università degli Studi di Milano, Via Luigi Mangiagalli 25, I-20133 Milano, Italy., Bonanni D; Department of Physical and Chemical Sciences, University of L'Aquila, via Vetoio, L'Aquila 67010, Italy., Del Bue A; Pattern Analysis and Computer Vision, Fondazione Istituto Italiano di Tecnologia, Via Morego, 30, 16163 Genova, Italy., Palermo G; Dipartimento di Elettronica Informazione e Bioingegneria, Politecnico di Milano, Via Ponzio 34/5, I-20133 Milano, Italy., Vistoli G; Dipartimento di Scienze Farmaceutiche, Università degli Studi di Milano, Via Luigi Mangiagalli 25, I-20133 Milano, Italy., Beccari AR; EXSCALATE, Dompé Farmaceutici SpA, Via Tommaso de Amicis 95, 80123 Naples, Italy.
Publikováno v:
Computational and structural biotechnology journal [Comput Struct Biotechnol J] 2024 May 18; Vol. 23, pp. 2141-2151. Date of Electronic Publication: 2024 May 18 (Print Publication: 2024).
Autor:
Filograna A; Institute of Experimental Endocrinology and Oncology 'G. Salvatore'(IEOS), National Research Council (CNR), 80131, Naples, Italy., De Tito S; Molecular Cell Biology of Autophagy, The Francis Crick Institute, London, UK. The Study Has Been Previously Performed at IEOS-CNR, Naples, Italy., Monte ML; Institute of Experimental Endocrinology and Oncology 'G. Salvatore'(IEOS), National Research Council (CNR), 80131, Naples, Italy., Oliva R; Department of Chemical Sciences, University of Naples Federico II, 80126, Naples, Italy., Bruzzese F; Animal Facility Unit, Istituto Nazionale Tumori-IRCCS-Fondazione G. Pascale, 80131, Naples, Italy., Roca MS; Experimental Pharmacology Unit, Istituto Nazionale Tumori-IRCCS-Fondazione G. Pascale, Naples, 80131, Italy., Zannetti A; Institute of Biostructures and Bioimaging (IBB), National Research Council (CNR), Naples, 80145, Italy., Greco A; Interdepartmental Service Center of Veterinary Radiology, University of Naples Federico II, 80137, Naples, Italy., Spano D; Institute of Experimental Endocrinology and Oncology 'G. Salvatore'(IEOS), National Research Council (CNR), 80131, Naples, Italy., Ayala I; Institute of Experimental Endocrinology and Oncology 'G. Salvatore'(IEOS), National Research Council (CNR), 80131, Naples, Italy., Liberti A; National Research Council (CNR), Piazzale Aldo Moro, 700185, Rome, Italy.; Biology and Evolution of Marine Organisms (BEOM), Stazione Zoologica Anton Dohrn, Naples, Italy., Petraccone L; Department of Chemical Sciences, University of Naples Federico II, 80126, Naples, Italy., Dathan N; Institute of Experimental Endocrinology and Oncology 'G. Salvatore'(IEOS), National Research Council (CNR), 80131, Naples, Italy., Catara G; Institute of Biochemistry and Cell Biology, National Research Council (CNR), 80131, Naples, Italy., Schembri L; National Research Council (CNR), Piazzale Aldo Moro, 700185, Rome, Italy.; Department of Pharmacy, University of Naples Federico II, 80131, Naples, Italy., Colanzi A; Institute of Experimental Endocrinology and Oncology 'G. Salvatore'(IEOS), National Research Council (CNR), 80131, Naples, Italy., Budillon A; Scientific Directorate, Istituto Nazionale Tumori-IRCCS-Fondazione G. Pascale, 80131, Naples, Italy., Beccari AR; EXSCALATE, Dompé Farmaceutici S.P.A, Naples, Italy., Del Vecchio P; Department of Chemical Sciences, University of Naples Federico II, 80126, Naples, Italy., Luini A; Institute of Experimental Endocrinology and Oncology 'G. Salvatore'(IEOS), National Research Council (CNR), 80131, Naples, Italy., Corda D; Institute of Experimental Endocrinology and Oncology 'G. Salvatore'(IEOS), National Research Council (CNR), 80131, Naples, Italy. daniela.corda@cnr.it., Valente C; Institute of Experimental Endocrinology and Oncology 'G. Salvatore'(IEOS), National Research Council (CNR), 80131, Naples, Italy. carmen.valente@cnr.it.; Present address: Dompé Farmaceutici S.P.A, L'Aquila, Italy. carmen.valente@cnr.it.
Publikováno v:
Journal of experimental & clinical cancer research : CR [J Exp Clin Cancer Res] 2024 May 06; Vol. 43 (1), pp. 137. Date of Electronic Publication: 2024 May 06.
Autor:
Manelfi C; EXSCALATE, Dompé Farmaceutici SpA, Via Tommaso de Amicis 95, 80123, Napoli, Italy., Tazzari V; EXSCALATE, Dompé Farmaceutici SpA, Via Tommaso de Amicis 95, 80123, Napoli, Italy., Lunghini F; EXSCALATE, Dompé Farmaceutici SpA, Via Tommaso de Amicis 95, 80123, Napoli, Italy., Cerchia C; Department of Pharmacy, University of Naples 'Federico II', Via D. Montesano 49, 80131, Napoli, Italy., Fava A; EXSCALATE, Dompé Farmaceutici SpA, Via Tommaso de Amicis 95, 80123, Napoli, Italy., Pedretti A; Dipartimento di Scienze Farmaceutiche, Università degli Studi di Milano, Via Mangiagalli, 25, 20133, Milano, Italy., Stouten PFW; EXSCALATE, Dompé Farmaceutici SpA, Via Tommaso de Amicis 95, 80123, Napoli, Italy.; Stouten Pharma Consultancy BV, Kempenarestraat 47, 2860, Sint-Katelijne-Waver, Belgium., Vistoli G; Dipartimento di Scienze Farmaceutiche, Università degli Studi di Milano, Via Mangiagalli, 25, 20133, Milano, Italy., Beccari AR; EXSCALATE, Dompé Farmaceutici SpA, Via Tommaso de Amicis 95, 80123, Napoli, Italy. andrea.beccari@dompe.com.
Publikováno v:
Journal of cheminformatics [J Cheminform] 2024 Feb 23; Vol. 16 (1), pp. 21. Date of Electronic Publication: 2024 Feb 23.
Autor:
Gervasoni S; Dipartimento di Scienze Farmaceutiche, Università Degli Studi di Milano, Via Mangiagalli, 25, I-20133 Milano, Italy.; Department of Physics, Università di Cagliari, I-09042 Monserrato, Italy., Manelfi C; EXSCALATE, Dompé Farmaceutici S.p.A., Via Tommaso De Amicis, 95, I-80131 Napoli, Italy., Adobati S; Dipartimento di Scienze Farmaceutiche, Università Degli Studi di Milano, Via Mangiagalli, 25, I-20133 Milano, Italy., Talarico C; EXSCALATE, Dompé Farmaceutici S.p.A., Via Tommaso De Amicis, 95, I-80131 Napoli, Italy., Biswas AD; EXSCALATE, Dompé Farmaceutici S.p.A., Via Tommaso De Amicis, 95, I-80131 Napoli, Italy., Pedretti A; Dipartimento di Scienze Farmaceutiche, Università Degli Studi di Milano, Via Mangiagalli, 25, I-20133 Milano, Italy., Vistoli G; Dipartimento di Scienze Farmaceutiche, Università Degli Studi di Milano, Via Mangiagalli, 25, I-20133 Milano, Italy., Beccari AR; EXSCALATE, Dompé Farmaceutici S.p.A., Via Tommaso De Amicis, 95, I-80131 Napoli, Italy.
Publikováno v:
International journal of molecular sciences [Int J Mol Sci] 2023 Dec 29; Vol. 25 (1). Date of Electronic Publication: 2023 Dec 29.
Autor:
Palchevskyi S; Laboratory of Protein Structure, International Institute of Molecular and Cell Biology in Warsaw, 02-109, Warsaw, Poland.; Cell Signalling Department, Institute of Molecular Biology and Genetics NASU, 03143, Kyiv, Ukraine., Czarnocki-Cieciura M; Laboratory of Protein Structure, International Institute of Molecular and Cell Biology in Warsaw, 02-109, Warsaw, Poland., Vistoli G; Dipartimento di Scienze Farmaceutiche, Università degli Studi di Milano, Via Mangiagalli, 25, I-20133, Milano, Italy., Gervasoni S; Dipartimento di Scienze Farmaceutiche, Università degli Studi di Milano, Via Mangiagalli, 25, I-20133, Milano, Italy.; Department of Physics, University of Cagliari, I-09042, Monserrato, Italy., Nowak E; Laboratory of Protein Structure, International Institute of Molecular and Cell Biology in Warsaw, 02-109, Warsaw, Poland., Beccari AR; Dompé Farmaceutici SpA, EXSCALATE, Via Tommaso De Amicis, 95, I-80131, Napoli, Italy., Nowotny M; Laboratory of Protein Structure, International Institute of Molecular and Cell Biology in Warsaw, 02-109, Warsaw, Poland. mnowotny@iimcb.gov.pl., Talarico C; Dompé Farmaceutici SpA, EXSCALATE, Via Tommaso De Amicis, 95, I-80131, Napoli, Italy. carmine.talarico@dompe.com.
Publikováno v:
Communications biology [Commun Biol] 2023 Oct 19; Vol. 6 (1), pp. 1065. Date of Electronic Publication: 2023 Oct 19.