Synthesis and Antiproliferative Activity of 2-amino-4-Anilinoquinazoline Derivatives

Autor: Patrick Depreux, Ravez S, Laurence Goossens, Arsenlis S, Castillo Aguilera O, Baldeyrou B, Lansiaux A, Schifano-Faux N, Barczyk A, Jean-François Goossens, Perrine Six

Publikováno v: Medicinal Chemistry. 5

Recently, we have reported a series of 4-anilino-6,7-dimethoxyquinazolines as tyrosine kinase inhibitors with interesting in vitro IC50 values for the Epidermal Growth Factor Receptor (EGFR) and/or for the Vascular Endothelial Growth Factor Receptor-

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::ed244a2b5f1b7c641f45005415767376
https://doi.org/10.4172/2161-0444.1000245

Synthesis and biological evaluation of new penta- and heptacyclic indolo- and quinolinocarbazole ring systems obtained via Pd(0) catalysed reductive N-heteroannulation

Autor: Laronze-Cochard, M., Cochard, F., Daras, E., Lansiaux, Apolline, Brassart, B., Vanquelef, E., Prost, E., Jm, Nuzillard, Baldeyrou, B., Jf, Goosens, Lozach, O., Meijer, L., Jf, Riou, Henon, E., Sapi, J.

Publikováno v: Organic & Biomolecular Chemistry
Organic & Biomolecular Chemistry, 2010, 8 (20), pp.4625-4636
Organic and Biomolecular Chemistry
Organic and Biomolecular Chemistry, Royal Society of Chemistry, 2010, 8 (20), pp.4625-4636

International audience

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=dedup_wf_001::a07dd403c2138f03341ec9e5e325af31
https://hal.science/hal-00554839

DNA intercalation, topisomerase II inhibition and cytotoxic activity of the plant alkaloid neocryptolepine

Autor: Christian BAILLY, Laine, W., Baldeyrou, B., Pauw-Gillet, M. -C, Colson, P., Houssier, C., Cimanga, K., Miert, S., Vlietinck, A. J., Pieters, L.

Publikováno v: Anti-cancer drug design
Publons
Scopus-Elsevier

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=dedup_wf_001::7eb7a39468445b1958dd7ccd01752277
https://hdl.handle.net/10067/338740151162165141

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