Photochemical Metal-Free synthesis and biological Assessment of isocryptolepine analogues targeting estrogen receptor Alpha in breast cancer cells.

Autor: Bogdanov FB; Department of Experimental Tumor Biology, N.N. Blokhin National Medical Research Center of Oncology, Kashirskoye shosse 24 bldg.15, 115522 Moscow, Russia; Faculty of Medicine, Moscow State University, Lomonosov prospect 27 bldg.1, 119991 Moscow, Russia. Electronic address: f.bogdanov.f@yandex.ru., Balakhonov RY; N.D. Zelinsky Institute of Organic Chemistry, Russian Academy of Sciences, Leninsky prospect 47, 119991 Moscow, Russia. Electronic address: balakhnvrman3@gmail.com., Volkov ES; N.D. Zelinsky Institute of Organic Chemistry, Russian Academy of Sciences, Leninsky prospect 47, 119991 Moscow, Russia. Electronic address: esvolkov@inbox.ru., Sonin IV; N.D. Zelinsky Institute of Organic Chemistry, Russian Academy of Sciences, Leninsky prospect 47, 119991 Moscow, Russia. Electronic address: igors3112@list.ru., Andreeva OE; Department of Experimental Tumor Biology, N.N. Blokhin National Medical Research Center of Oncology, Kashirskoye shosse 24 bldg.15, 115522 Moscow, Russia. Electronic address: o.andreeva@ronc.ru., Sorokin DV; Department of Experimental Tumor Biology, N.N. Blokhin National Medical Research Center of Oncology, Kashirskoye shosse 24 bldg.15, 115522 Moscow, Russia. Electronic address: d.sorokin@ronc.ru., Piven YA; Institute of Bioorganic Chemistry, National Academy of Sciences of Belarus, Akad. Kuprevicha st. 5/2, Minsk 220084, Belarus. Electronic address: piven.ya@gmail.com., Scherbakov AM; Department of Experimental Tumor Biology, N.N. Blokhin National Medical Research Center of Oncology, Kashirskoye shosse 24 bldg.15, 115522 Moscow, Russia; Gause Institute of New Antibiotics, Bol'shaya Pirogovskaya ulitsa 11, 119021 Moscow, Russia. Electronic address: alex.scherbakov@gmail.com., Shirinian VZ; N.D. Zelinsky Institute of Organic Chemistry, Russian Academy of Sciences, Leninsky prospect 47, 119991 Moscow, Russia. Electronic address: svbegunt@mail.ru.

Publikováno v: Bioorganic chemistry [Bioorg Chem] 2024 Dec; Vol. 153, pp. 107942. Date of Electronic Publication: 2024 Nov 05.

Light-driven photoswitching of quinazoline analogues of combretastatin A-4 as an effective approach for targeting skin cancer cells.

Autor: Scherbakov AM; Department of Experimental Tumor Biology, Blokhin N.N. National Medical Research Center of Oncology, Kashirskoye sh. 24, Moscow 115522, Russian Federation., Balakhonov RY; N. D. Zelinsky Institute of Organic Chemistry, RAS, Moscow, Russian Federation. svbegunt@mail.ru., Salnikova DI; Department of Experimental Tumor Biology, Blokhin N.N. National Medical Research Center of Oncology, Kashirskoye sh. 24, Moscow 115522, Russian Federation.; Faculty of Medicine, Lomonosov Moscow State University, Moscow, Russian Federation., Sorokin DV; Department of Experimental Tumor Biology, Blokhin N.N. National Medical Research Center of Oncology, Kashirskoye sh. 24, Moscow 115522, Russian Federation., Yadykov AV; N. D. Zelinsky Institute of Organic Chemistry, RAS, Moscow, Russian Federation. svbegunt@mail.ru., Markosyan AI; Scientific Technological Center of Organic and Pharmaceutical Chemistry, NAS RA, Yerevan, Armenia., Shirinian VZ; N. D. Zelinsky Institute of Organic Chemistry, RAS, Moscow, Russian Federation. svbegunt@mail.ru.

Publikováno v: Organic & biomolecular chemistry [Org Biomol Chem] 2021 Sep 15; Vol. 19 (35), pp. 7670-7677. Date of Electronic Publication: 2021 Sep 15.