Zobrazeno 1 - 5
of 5
pro vyhledávání: '"Balaji Vitukudi Narayanaiyenga"'
Autor:
Ilya Okun, Ming Fai Chan, Rosario Silvestre Castillo, Fiona Stavros, Raju Bore Gowda, Emily Hwang, Balaji Vitukudi Narayanaiyenga, Adam Kois, Chengde Wu, Erik Verner
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 6:2393-2398
Replacement of the 4-methyl group in a series of N-(3,4-dimethylisoxazolyl)benzenesulfonamide endothelin antagonists with a bromine or chlorine atom resulted in a three- to ten-fold increase in the binding affinity for both the ETA and ETB receptors.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::4f5becdfc4f23bbb9e55cc361edb527c
https://doi.org/10.1016/0960-894x(96)00441-6
https://doi.org/10.1016/0960-894x(96)00441-6
Autor:
Adam Kois, Kottayil I. Varughese, Balaji Vitukudi Narayanaiyenga, Raju Bore Gowda, Jay I. Varughese, Ming Fai Chan
Publikováno v:
ChemInform. 30
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::a56cc189887616c27b72e0c370a1fdb1
https://doi.org/10.1002/chin.199926162
https://doi.org/10.1002/chin.199926162
Autor:
Raju Bore Gowda, Adam Kois, Chengde Wu, Erik Verner, Ming Fai Chan, Balaji Vitukudi Narayanaiyenga, Fiona Stavros, Rosario Silvestre Castillo, Ilya Okun
Publikováno v:
Bioorganicmedicinal chemistry. 6(12)
The systematic modification of the ETA selective N-(5-isoxazolyl)benzene-sulfonamide endothelin antagonists to give ETB selective antagonists is reported. The reversal in selectivity was brought about by substitution of the 4-position with aryl and s
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::424e0120a12677485b3f0d9c47e2f814
https://pubmed.ncbi.nlm.nih.gov/9925292
https://pubmed.ncbi.nlm.nih.gov/9925292
Autor:
Rosario Silverstre Castillo, Ming Fai Chan, Mengfen Lin, Balaji Vitukudi Narayanaiyenga, Cynthia K. Larive
Publikováno v:
International journal of peptide and protein research. 48(3)
Two endothelin antagonists cyclo(D-Leu-D-Val-Pro-D-Asp-Trp) (IPI-147), and cyclo (D-Trp-D-Asp-Ac3c-D-Val-Leu) (IPI-725) have been synthetized. Their solution conformations have been studied in aqueous solution by NMR spectroscopy and dynamics simulat
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2e422810a0e88d3f2eb1e3a5c83c7700
https://pubmed.ncbi.nlm.nih.gov/8897090
https://pubmed.ncbi.nlm.nih.gov/8897090
Autor:
Balaji Vitukudi Narayanaiyenga, Raju Bore Gowda, Ming Fai Chan, Jay I. Varughese, Adam Kois, Kottayil I. Varughese
Publikováno v:
HETEROCYCLES. 51:5
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::1c5a435a7aa3f86ca1d3e3b681275d19
https://doi.org/10.3987/com-98-8343
https://doi.org/10.3987/com-98-8343