Immunoproteasome inhibition and bioactivity of thiasyrbactins

Autor: Bakas, NA, Schultz, CR, Yco, LP, Roberts, CC, Chang, C-EA, Bachmann, AS, Pirrung, MC

Publikováno v: Bakas, NA; Schultz, CR; Yco, LP; Roberts, CC; Chang, C-EA; Bachmann, AS; et al.(2018). Immunoproteasome inhibition and bioactivity of thiasyrbactins. BIOORGANIC & MEDICINAL CHEMISTRY, 26(2), 401-412. doi: 10.1016/j.bmc.2017.11.048. UC Riverside: Retrieved from: http://www.escholarship.org/uc/item/9r33c48t

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=od_______325::6b313c1e30f46dafe581831fc696b985
http://www.escholarship.org/uc/item/9r33c48t

Inhibitors of the Hippo Pathway Kinases STK3/MST2 and STK4/MST1 Have Utility for the Treatment of Acute Myeloid Leukemia.

Autor: Bata N; Cell and Molecular Biology of Cancer Program, NCI-Designated Cancer Center, Sanford Burnham Prebys Medical Discovery Institute, 10901 North Torrey Pines Road, La Jolla, California 92037, United States., Chaikuad A; Buchmann Institute for Molecular Life Sciences, Structural Genomics Consortium, Johann Wolfgang Goethe-University, D-60438 Frankfurt am Main, Germany.; Institute for Pharmaceutical Chemistry, Max von Lauestrasse 9, Johann Wolfgang Goethe-University, D-60438 Frankfurt am Main, Germany., Bakas NA; Cell and Molecular Biology of Cancer Program, NCI-Designated Cancer Center, Sanford Burnham Prebys Medical Discovery Institute, 10901 North Torrey Pines Road, La Jolla, California 92037, United States., Limpert AS; Cell and Molecular Biology of Cancer Program, NCI-Designated Cancer Center, Sanford Burnham Prebys Medical Discovery Institute, 10901 North Torrey Pines Road, La Jolla, California 92037, United States., Lambert LJ; Cell and Molecular Biology of Cancer Program, NCI-Designated Cancer Center, Sanford Burnham Prebys Medical Discovery Institute, 10901 North Torrey Pines Road, La Jolla, California 92037, United States., Sheffler DJ; Cell and Molecular Biology of Cancer Program, NCI-Designated Cancer Center, Sanford Burnham Prebys Medical Discovery Institute, 10901 North Torrey Pines Road, La Jolla, California 92037, United States., Berger LM; Buchmann Institute for Molecular Life Sciences, Structural Genomics Consortium, Johann Wolfgang Goethe-University, D-60438 Frankfurt am Main, Germany.; Institute for Pharmaceutical Chemistry, Max von Lauestrasse 9, Johann Wolfgang Goethe-University, D-60438 Frankfurt am Main, Germany., Liu G; Chemistry Department, Viva Biotech Ltd., 581 Shen Kuo Road, Shanghai 201203, China., Yuan C; Chemistry Department, Viva Biotech Ltd., 581 Shen Kuo Road, Shanghai 201203, China., Wang L; Chemistry Department, Viva Biotech Ltd., 581 Shen Kuo Road, Shanghai 201203, China., Peng Y; Chemistry Department, Viva Biotech Ltd., 581 Shen Kuo Road, Shanghai 201203, China., Dong J; Chemistry Department, Viva Biotech Ltd., 581 Shen Kuo Road, Shanghai 201203, China., Celeridad M; Cell and Molecular Biology of Cancer Program, NCI-Designated Cancer Center, Sanford Burnham Prebys Medical Discovery Institute, 10901 North Torrey Pines Road, La Jolla, California 92037, United States., Layng F; Cell and Molecular Biology of Cancer Program, NCI-Designated Cancer Center, Sanford Burnham Prebys Medical Discovery Institute, 10901 North Torrey Pines Road, La Jolla, California 92037, United States., Knapp S; Buchmann Institute for Molecular Life Sciences, Structural Genomics Consortium, Johann Wolfgang Goethe-University, D-60438 Frankfurt am Main, Germany.; Institute for Pharmaceutical Chemistry, Max von Lauestrasse 9, Johann Wolfgang Goethe-University, D-60438 Frankfurt am Main, Germany.; Translational cancer network DKTK site Frankfurt/Mainz and Frankfurt Cancer Institute (FCI), Johann Wolfgang Goethe-University, D-60438 Frankfurt am Main, Germany., Cosford NDP; Cell and Molecular Biology of Cancer Program, NCI-Designated Cancer Center, Sanford Burnham Prebys Medical Discovery Institute, 10901 North Torrey Pines Road, La Jolla, California 92037, United States.

Publikováno v: Journal of medicinal chemistry [J Med Chem] 2022 Jan 27; Vol. 65 (2), pp. 1352-1369. Date of Electronic Publication: 2021 Nov 22.

Autophagy in Cancer: Regulation by Small Molecules.

Autor: Limpert AS; NCI Designated Cancer Center, Sanford-Burnham Prebys Medical Discovery Institute, La Jolla, CA, USA; These authors contributed equally., Lambert LJ; NCI Designated Cancer Center, Sanford-Burnham Prebys Medical Discovery Institute, La Jolla, CA, USA; These authors contributed equally., Bakas NA; NCI Designated Cancer Center, Sanford-Burnham Prebys Medical Discovery Institute, La Jolla, CA, USA., Bata N; NCI Designated Cancer Center, Sanford-Burnham Prebys Medical Discovery Institute, La Jolla, CA, USA., Brun SN; Department of Molecular and Cell Biology, The Salk Institute for Biological Studies, San Diego, La Jolla, CA, USA., Shaw RJ; Department of Molecular and Cell Biology, The Salk Institute for Biological Studies, San Diego, La Jolla, CA, USA., Cosford NDP; NCI Designated Cancer Center, Sanford-Burnham Prebys Medical Discovery Institute, La Jolla, CA, USA. Electronic address: ncosford@sbpdiscovery.org.

Publikováno v: Trends in pharmacological sciences [Trends Pharmacol Sci] 2018 Dec; Vol. 39 (12), pp. 1021-1032.

Immunoproteasome inhibition and bioactivity of thiasyrbactins.

Autor: Bakas NA; Department of Chemistry, University of California, Riverside, CA 92521, USA., Schultz CR; Department of Pediatrics and Human Development, College of Human Medicine, Michigan State University, Grand Rapids, MI 49503, USA., Yco LP; Department of Pediatrics and Human Development, College of Human Medicine, Michigan State University, Grand Rapids, MI 49503, USA., Roberts CC; Department of Chemistry, University of California, Riverside, CA 92521, USA., Chang CA; Department of Chemistry, University of California, Riverside, CA 92521, USA., Bachmann AS; Department of Pediatrics and Human Development, College of Human Medicine, Michigan State University, Grand Rapids, MI 49503, USA. Electronic address: andre.bachmann@hc.msu.edu., Pirrung MC; Department of Chemistry, University of California, Riverside, CA 92521, USA; Department of Pharmaceutical Sciences, University of California, Irvine, CA 92697, USA. Electronic address: Michael.pirrung@ucr.edu.

Publikováno v: Bioorganic & medicinal chemistry [Bioorg Med Chem] 2018 Jan 15; Vol. 26 (2), pp. 401-412. Date of Electronic Publication: 2017 Dec 07.