Zobrazeno 1 - 10
of 29
pro vyhledávání: '"Baijayantimala Swain"'
Autor:
Mohammed Arifuddin, Claudiu T. Supuran, Srinivas Nanduri, Krishna Kartheek Chinchilli, Priti Singh, Baijayantimala Swain, Nerella Sridhar Goud, Dilep Kumar Sigalapalli, Abhishek Choli, Andrea Angeli, Venkata Madhavi Yaddanapudi
Publikováno v:
Anti-Cancer Agents in Medicinal Chemistry. 23:1225-1233
Background: Carbonic anhydrases (CAs, EC 4.2.1.1) catalyze the reversible hydration of carbon dioxide to bicarbonate and a proton. Inhibition of isoforms IX and XII has induced potent anticancer effects. Objective: A series of indole-3-sulfonamide-he
Autor:
Baijayantimala Swain, Abrar Khan, Priti Singh, Vaibhav S. Marde, Andrea Angeli, Krishna Kartheek Chinchilli, Venkata Madhavi Yaddanapudi, Simone Carradori, Claudiu T. Supuran, Mohammed Arifuddin
Publikováno v:
Molecules, Vol 27, Iss 22, p 8028 (2022)
A novel series of twenty-five rhodamine-linked benzenesulfonamide derivatives (7a–u and 9a–d) were synthesized and screened for their inhibitory action against four physiologically relevant human (h) carbonic anhydrase (CA) isoforms, namely hCA I
Externí odkaz:
https://doaj.org/article/a422a55ee080449dab1df6c758b9bb1d
Autor:
Baijayantimala Swain, Andrea Angeli, Srinivas Angapelly, Pavitra S. Thacker, Priti Singh, Claudiu T. Supuran, Mohammed Arifuddin
Publikováno v:
Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 34, Iss 1, Pp 1199-1209 (2019)
The synthesis of a novel series of 3-functionalised benzenesulfonamides incorporating phenyl-1,2,3-triazole with an amide linker was achieved by using the “click-tail” approach. The new compounds, including the intermediates, were assayed as inhi
Externí odkaz:
https://doaj.org/article/b2f5c8215efe4eb08c2a2b7477d7b20d
Autor:
Mohammed Arifuddin, Claudiu T. Supuran, Venkata Madhavi Yaddanapudi, Baijayantimala Swain, Priti Singh, Andrea Angeli, Santosh Kumar Sahoo
Publikováno v:
Anti-Cancer Agents in Medicinal Chemistry. 22:2358-2366
Background: A high yielding green protocol has been developed and delineated for the synthesis of 3,3- di(indolyl)indolin-2-ones, potentially bioactive compounds, involving one pot aqueous medium condensation of isatin with indole in the presence of
Autor:
Pavitra S. Thacker, Prerna L. Tiwari, Andrea Angeli, Danaboina Srikanth, Baijayantimala Swain, Mohammed Arifuddin, Claudiu T. Supuran
Publikováno v:
Metabolites, Vol 11, Iss 4, p 225 (2021)
A series of coumarin-linked 4-anilinomethyl-1,2,3-triazoles (6a–t) was synthesized via a molecular hybridization approach, through carbon C-6 of the coumarin moiety. The synthesized compounds were evaluated for their inhibition of carbonic anhydras
Externí odkaz:
https://doaj.org/article/9cb8f55cf7294bf59c050f2eea9d143b
Autor:
Priti Singh, Santosh Kumar Sahoo, Nerella Sridhar Goud, Baijayantimala Swain, Venkata Madhavi Yaddanapudi, Mohammed Arifuddin
Publikováno v:
Asian Journal of Organic Chemistry. 11
Autor:
Baijayantimala Swain, Santosh Kumar Sahoo, Priti Singh, Andrea Angeli, Venkata Madhavi Yaddanapudi, Claudiu T. Supuran, Mohammed Arifuddin
Publikováno v:
European journal of medicinal chemistry. 234
A novel series of 32 sulfonamide containing quinolines (5a-j, 7a-k and 9a-k) were synthesized using tail approach and assayed for their carbonic anhydrase inhibitory potency against four human (h) carbonic anhydrase (CA) isoforms hCA I, II, IX and XI
Autor:
Priti Singh, Dilep Kumar Sigalapalli, Nerella Sridhar Goud, Baijayantimala Swain, Santosh Kumar Sahoo, Andrea Angeli, Afzal B. Shaik, Venkata Madhavi Yaddanapudi, Claudiu T. Supuran, Mohammed Arifuddin
Publikováno v:
ChemMedChem. 17(5)
Owing to severe allergic reactions (anaphylaxis) and resistance exhibited by sulfonamide-based carbonic anhydrase (CA) inhibitors, non-classical or non-sulfonamide CA inhibitors are gaining increased attention by medicinal chemists. In this context,
Autor:
Priti Singh, Nerella Sridhar Goud, Baijayantimala Swain, Santosh Kumar Sahoo, Abhishek Choli, Andrea Angeli, Bhoopendra Singh Kushwah, Venkata Madhavi Yaddanapudi, Claudiu T. Supuran, Mohammed Arifuddin
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 70:128809
In this manuscript, design, rational, synthesisand carbonic anhydrases (CAs) inhibitory profile of the quinoline/pyridine linked indole-3-sulfonamide derivatives were reported. The library of 29newly quinoline/pyridine indole-3-sulfonamide derivative
Autor:
Venkata M. Yaddanapudi, Claudiu T. Supuran, Abhay Kothari, Andrea Angeli, Kamtam Aashritha, Mohammed Arifuddin, Dilep Kumar Sigalapalli, Priti Singh, Baijayantimala Swain
Publikováno v:
Archiv der PharmazieREFERENCES. 354(7)
A novel series of imidazothiadiazole-linked benzenesulfonamide derivatives (5a-t) was synthesized and subjected for screening against the four physiologically and pharmacologically relevant human carbonic anhydrase (hCA) isoforms: hCA I, II, VA, and