Syntheses and antiproliferative effects of d-homo- and d-secoestrones

Autor: Mernyák, Erzsébet, Szabó, Johanna, Bacsa, Ildikó, Huber, Judit, Schneider, Gyula, Minorics, Renáta, Bózsity, Noémi, Zupkó, István, Varga, Mónika, Bikádi, Zsolt, Hazai, Eszter, Wölfling, János

Publikováno v: In Steroids September 2014 87:128-136

Synthesis and in vitro pharmacological evaluation of N -[(1-benzyl-1,2,3-triazol-4-yl)methyl]-carboxamides on d -secoestrone scaffolds.

Autor: Szabó, Johanna¹ (AUTHOR), Bacsa, Ildikó¹ (AUTHOR), Wölfling, János¹ (AUTHOR), Schneider, Gyula¹ (AUTHOR), Zupkó, István² (AUTHOR), Varga, Mónika³ (AUTHOR), Herman, Bianka E.⁴ (AUTHOR), Kalmár, László⁵ (AUTHOR), Szécsi, Mihály⁴ (AUTHOR), Mernyák, Erzsébet¹ (AUTHOR) bobe@chem.u-szeged.hu

Publikováno v: Journal of Enzyme Inhibition & Medicinal Chemistry. Aug2016, Vol. 31 Issue 4, p574-579. 6p.

Comparative investigation of the in vitro inhibitory potencies of 13-epimeric estrones and D-secoestrones towards 17β-hydroxysteroid dehydrogenase type 1

Autor: Herman, Bianka Edina, Szabó, Johanna, Bacsa, Ildikó, Wölfling, János, Schneider, Gyula, Bálint, Mónika, Hetényi, Csaba, Mernyák, Erzsébet, Szécsi, Mihály

The inhibitory effects of 13-epimeric estrones, D-secooxime and D-secoalcohol estrone compounds on human placental 17β-hydroxysteroid dehydrogenase type 1 isozyme (17β-HSD1) were investigated. The transformation of estrone to 17β-estradiol was stu

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The first Pd-catalyzed Buchwald-Hartwig aminations at C-2 or C-4 in the estrone series.

Autor: Bacsa I; Department of Organic Chemistry, University of Szeged, Dóm tér 8, H-6720 Szeged, Hungary., Szemerédi D; Department of Organic Chemistry, University of Szeged, Dóm tér 8, H-6720 Szeged, Hungary., Wölfling J; Department of Organic Chemistry, University of Szeged, Dóm tér 8, H-6720 Szeged, Hungary., Schneider G; Department of Organic Chemistry, University of Szeged, Dóm tér 8, H-6720 Szeged, Hungary., Fekete L; Department of Medicinal Chemistry, University of Szeged, Dóm tér 8, H-6720 Szeged, Hungary., Mernyák E; Department of Organic Chemistry, University of Szeged, Dóm tér 8, H-6720 Szeged, Hungary.

Publikováno v: Beilstein journal of organic chemistry [Beilstein J Org Chem] 2018 May 04; Vol. 14, pp. 998-1003. Date of Electronic Publication: 2018 May 04 (Print Publication: 2018).