Zobrazeno 1 - 10
of 170
pro vyhledávání: '"B. Hochberg"'
Autor:
Timothy A. Coulther, David Labaree, Jessa L. Silver, Robert Dilis, Edward Hua, Richard B. Hochberg, Emmett McCaskill, Robert N. Hanson, Mary Jo Ondrechen, Pakamas Tongcharoensirikul
Publikováno v:
Steroids. 144:15-20
A series consisting of substituted benzoylbenzamide derivatives of 17α-E-vinyl estradiol 6a-i and 7a-d was prepared in good overall yields from the corresponding novel iodinated benzoylbenzamide precursors using Pd(0)-catalyzed Stille coupling. Biol
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::bd16f6deaa0e9a5ccb0c5f49b75c6cfc
https://doi.org/10.1016/j.steroids.2019.02.003
https://doi.org/10.1016/j.steroids.2019.02.003
Publikováno v:
Cytotherapy. 24:S55
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::5d01f252287360d9e61e9f9a4b9bfeaf
https://doi.org/10.1016/s1465-3249(22)00186-4
https://doi.org/10.1016/s1465-3249(22)00186-4
Publikováno v:
Neuroendocrinology. 103:538-551
Background/Aims: The contributions of the three principal ovarian steroid hormones (estradiol, progesterone and testosterone) to the regulation of estrogen receptor alpha (ERα) levels in the rat brain were examined during the estrous cycle. Methods:
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::d2754458c7a4ca3d8a298d3b84292664
https://doi.org/10.1159/000441077
https://doi.org/10.1159/000441077
Publikováno v:
Chinese Chemical Letters. 25:567-570
We have previously found that several families of nonpolar short chain 11 β -ethers and esters of estradiol are selective estrogen receptor modulators (SERMs). Surprisingly, the transformation from potent estrogen to anti-estrogen occurs when the 11
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::08a287c825eef5f04fc96df16b126890
https://doi.org/10.1016/j.cclet.2014.01.015
https://doi.org/10.1016/j.cclet.2014.01.015
Autor:
Robert Dilis, Emmett McCaskill, David Labaree, Robert N. Hanson, Pakamas Tongcharoensirikul, Richard B. Hochberg
Publikováno v:
Steroids. 77:471-476
As part of our program to explore the influence of small structural modifications on the biological response of the estrogen receptor-α (ERα), we prepared and evaluated a series of mono-and di-substituted phenyl vinyl estradiols. The target compoun
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a9e2a36dbf45d8de5937d49724e7a65c
https://doi.org/10.1016/j.steroids.2012.01.003
https://doi.org/10.1016/j.steroids.2012.01.003
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Publikováno v:
Neuroendocrinology. 103(5)
The contributions of the three principal ovarian steroid hormones (estradiol, progesterone and testosterone) to the regulation of estrogen receptor alpha (ERα) levels in the rat brain were examined during the estrous cycle.Receptor concentrations we
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid________::bb1b7040c7fe78e05b53a083b5662f17
https://pubmed.ncbi.nlm.nih.gov/26422138
https://pubmed.ncbi.nlm.nih.gov/26422138
Autor:
Nick Z. Lu, Kerry L. Burnstein, Donald P. McDonnell, Peter J. Fuller, John A. Cidlowski, Suzanne E. Wardell, Jack Michel Renoir, Donald B. DeFranco, Elizabeth M. Wilson, Richard B. Hochberg, Vincent Giguère, Lorraine I. McKay, Nancy L. Weigel
Publikováno v:
Pharmacological Reviews. 58:782-797
The glucocorticoid receptor (GR[1][1]), mineralocorticoid receptor (MR), progesterone receptor (PR), and androgen receptor (AR) are classic members of the nuclear receptor superfamily, composing subfamily 3C. Members of this subfamily are among those
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5a8eb12213002b4cdae3e23eaf8d33ab
https://doi.org/10.1124/pr.58.4.9
https://doi.org/10.1124/pr.58.4.9
Autor:
David Labaree, Richard B. Hochberg, Robert A. Stockland, Mark C. Kohler, John A. Bawiec, Ilia A. Guzei, Margaret E. Kastner
Publikováno v:
Organometallics. 25:2475-2485
Gold complexes of 17-ethynyl-17β-hydroxyandrost-4-en-3-one, 17-ethynyl-3-methoxyestra-1,3,5(10)-trien-17β-ol, and 17α-ethynylestra-1,3,5(10)-triene-3,17β-diol have been prepared and characterized. The title compounds were prepared by treatment of
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::6d53794a1022baa66e31867456c1670e
https://doi.org/10.1021/om051064r
https://doi.org/10.1021/om051064r
Publikováno v:
Journal of Medicinal Chemistry. 48:1428-1447
We have previously found that esters of 11beta-estradiol carboxylates are transformed from an estrogen into an antiestrogen when the 11beta-side chain is increased in length from four to five non-hydrogen atoms (nor = 5). To understand the structural
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4eab4d7538bfdcdf0c25d01d37d0a963
https://doi.org/10.1021/jm049352x
https://doi.org/10.1021/jm049352x