Výsledky vyhledávání - "B. F. Garifullin"

Autor: B. F. Garifullin, Vladimir E. Kataev

Publikováno v: Chemistry of Heterocyclic Compounds. 57:326-341

The minireview surveys the modification of native nucleosides as a result of which huge libraries of nucleoside analogs of various structures were synthesized. Particular attention is paid to the synthesis of the so-called prodrug forms of nucleoside

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::51ebf6efe7d3e998fe7d2577bcbacd57
https://doi.org/10.1007/s10593-021-02912-8

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Synthesis of 1,2,3-triazolyl nucleoside analogues and their antiviral activity

Autor: Iana L Yesaulkova, Vladimir E. Kataev, Olga V. Andreeva, Vladimir V. Zarubaev, Alexander V. Slita, B. F. Garifullin, Maya G. Belenok, M. M. Shulaeva, Liliya F. Saifina, Vyacheslav E. Semenov

Publikováno v: Molecular Diversity

Based on the fact that a search for influenza antivirals among nucleoside analogues has drawn very little attention of chemists, the present study reports the synthesis of a series of 1,2,3-triazolyl nucleoside analogues in which a pyrimidine fragmen

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::60842714558eb48a28e9f3462914d4b0
https://doi.org/10.1007/s11030-020-10141-y

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Synthesis and Antiviral Evaluation of Nucleoside Analogues Bearing One Pyrimidine Moiety and Two D-Ribofuranosyl Residues

Autor: Olga V. Andreeva, Liliya F. Saifina, M. M. Shulaeva, Anna P. Lyubina, Maria A Man'kova, Iana L Yesaulkova, Alexandrina S. Volobueva, Alexander V. Slita, B. F. Garifullin, Vyacheslav E. Semenov, Vladimir V. Zarubaev, Alexandra D. Voloshina, Mayya G Belenok, Vladimir E. Kataev

Publikováno v: Molecules
Molecules, Vol 26, Iss 3678, p 3678 (2021)
Volume 26
Issue 12

A series of 1,2,3-triazolyl nucleoside analogues in which 1,2,3-triazol-4-yl-β-d-ribofuranosyl fragments are attached via polymethylene linkers to both nitrogen atoms of the heterocycle moiety (uracil, 6-methyluracil, thymine, quinazoline-2,4-dione,

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c84a88e67f3506817018c8dad811e2a0
http://europepmc.org/articles/PMC8234143

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Synthesis and cytotoxicity of the conjugates of diterpenoid isosteviol and N-acetyl-D-glucosamine

Autor: R. R. Sharipova, A. S. Sapunova, A. D. Voloshina, Irina Yu. Strobykina, B. F. Garifullin, Leysan R Khabibulina, Bulat I. Khairutdinov, Yuriy F. Zuev, Vladimir E. Kataev

Publikováno v: Natural Product Research. 35:1372-1378

A series of conjugates of diterpenoid isosteviol (16-oxo-ent-beyeran-19-oic acid) and N-acetyl-D-glucosamine was synthesised and their cytotoxicity against several human cancer cell lines (M-Hela, ...

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::468a1c92a9ddca973815d0e117829b5b
https://doi.org/10.1080/14786419.2019.1650355

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Synthesis and Biological Activity of 3,4,-Tri-О-Acetyl-N-Acetylglucosamine and Tetraacetylglucopyranose Conjugated with Alkyl Phosphates

Autor: A. S. Sapunova, A. D. Voloshina, Vladimir E. Kataev, R. R. Sharipova, M. A. Kravchenko, B. F. Garifullin

Publikováno v: Russian Journal of Bioorganic Chemistry. 45:155-164

Conjugates of 3,4,6-tri-О-acetyl-N-acetylglucosamine and tetraacetyl glucopyranose with alkyl phosphates were synthesized. The dependence of their antibacterial and antituberculosis activities on the length of the alkyl substituent at the phosphate

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::d8c470f68c08e0d685dbe2d48994e51b
https://doi.org/10.1134/s1068162019020110

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Synthesis and Biological Activity of Alkane-1,1-diylbis(phosphonates) of Diterpenoid Isosteviol

Autor: A. S. Sapunova, A. D. Voloshina, Vladimir E. Kataev, I. Yu. Strobykina, A. V. Nemtarev, B. F. Garifullin

Publikováno v: Russian Journal of Organic Chemistry. 55:17-24

Isosteviol reacted with α,ω-dibromoalkanes to give 19-(ω-bromoahkyl) esters which were treated with tetraethyl methylenebis(phosphonate) to obtain bis(phosphonates) conjugated to the deterpenoid skeleton through a polymethylene spacer. The bis(pho

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::13f0a68e1f1c49399e6f21de0ce1a782
https://doi.org/10.1134/s1070428019010044

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Glycosides and Glycoconjugates of the Diterpenoid Isosteviol with a 1,2,3-Triazolyl Moiety: Synthesis and Cytotoxicity Evaluation

Autor: Irina Yu. Strobykina, B. F. Garifullin, Alexey B. Dobrynin, Olga V. Andreeva, Leysan R Khabibulina, R. R. Sharipova, Alexandra D. Voloshina, Mayya G Belenok, Vladimir E. Kataev, A. S. Sapunova

Publikováno v: Journal of natural products. 83(8)

Several glycoconjugates of the diterpenoid isosteviol (16-oxo-ent-beyeran-19-oic acid) with a 1,2,3-triazolyl moiety were synthesized, and their cytotoxicity was evaluated against some human cancer and normal cell lines. Most of the synthesized compo

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2e77193ba94b39c32ece72c1ee21b252
https://pubmed.ncbi.nlm.nih.gov/32786882

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Synthesis and Antitubercular and Antibacterial Activities of Triethylammonium 2-Acetamido-3,4,6-tri-O-acetyl-2-deoxy-D-glucopyranosyl Decyl Phosphate

Autor: R. R. Sharipova, Vladimir E. Kataev, M. A. Kravchenko, A. D. Voloshina, B. F. Garifullin

Publikováno v: Russian Journal of Organic Chemistry. 54:1333-1336

Phosphorylation of 2-acetamido-3,4,6-tri-O-acetyl-2-deoxy-D-glucose at the anomeric hydroxy group gave previously unknown triethylammonium 2-acetamido-3,4,6-tri-O-acetyl-2-deoxy-D-glucopyranosyl phosphonate, and successive treatment of the latter wit

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::e7270618b2080cb3045c264e191dfcb6
https://doi.org/10.1134/s1070428018090117

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New Targets for Growth Inhibition of Mycobacterium tuberculosis: Why Do Natural Terpenoids Exhibit Antitubercular Activity?

Autor: B. F. Garifullin, Vladimir E. Kataev, R. N. Khaybullin, R. R. Sharipova

Publikováno v: Russian Journal of Bioorganic Chemistry. 44:438-452

The article draws the attention of chemists to the literature data reporting the discovery of new targets for growth inhibition of Mycobacterium tuberculosis, namely, diterpene cyclase (Rv3377c) and tuberculosinol phosphatase (Rv3378c), which produce

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::4640975ba464632b7fcfe1a18db30640
https://doi.org/10.1134/s1068162018040106

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