Zobrazeno 1 - 9
of 9
pro vyhledávání: '"Bérengère Sauvagnat"'
Autor:
Michael Garrigou, Bérengère Sauvagnat, Ruchia Duggal, Nicole Boo, Pooja Gopal, Jennifer M. Johnston, Anthony Partridge, Tomi Sawyer, Kaustav Biswas, Nicolas Boyer
Publikováno v:
Journal of medicinal chemistry. 65(13)
Macrocyclic peptides can disrupt previously intractable protein-protein interactions (PPIs) relevant to oncology targets such as KRAS. Early hits often lack cellular activity and require meticulous improvement of affinity, permeability, and metabolic
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::491831c740f73f2615b446cf167b05cf
https://pubmed.ncbi.nlm.nih.gov/35707970
https://pubmed.ncbi.nlm.nih.gov/35707970
Publikováno v:
Tetrahedron Letters. 41:6371-6375
A Schiff base protected glycine supported on a soluble polymer such as poly(ethylene glycol) reacted readily with various electrophiles in the presence of an inorganic base under microwave activation. It was shown in this study that the polymer suppo
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::497170f13144b4dee24ea54a0f3092bb
https://doi.org/10.1016/s0040-4039(00)01067-4
https://doi.org/10.1016/s0040-4039(00)01067-4
Publikováno v:
Comptes Rendus de l'Académie des Sciences - Series IIC - Chemistry. 1:777-780
A poly(ethylene glycol) (PEG) supported substrate bearing a methyl acrylate moiety has been subjected to a palladium-catalyzed Heck reaction with phenyl iodide to afford an analogue of glutamic acid with a good regio- and stereoselectivity of the dou
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::cba1fe3509fc88df917b714e67ed93c5
https://doi.org/10.1016/s1251-8069(99)80045-0
https://doi.org/10.1016/s1251-8069(99)80045-0
Autor:
Bérengère Sauvagnat, J.-L. Aubagnac, Christine Enjalbal, Frédéric Lamaty, René Lazaro, Jean Martinez
Publikováno v:
Rapid Communications in Mass Spectrometry. 12:1034-1037
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::f84f8ed46ebc147bfb092b78c1518783
https://doi.org/10.1002/(sici)1097-0231(19980815)12:15<1034::aid-rcm264>3.0.co
https://doi.org/10.1002/(sici)1097-0231(19980815)12:15<1034::aid-rcm264>3.0.co
Publikováno v:
Tetrahedron Letters. 39:821-824
α-substituted α-amino esters were synthesized in liquid-phase by polyethylene glycol (ce:simple-paraEG) promoted alkylation of a polyethylene glycol-supported Schiff base activated glycine ester.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::57913574541f8c58c6cb5dfaba2a90ad
https://doi.org/10.1016/s0040-4039(97)10722-5
https://doi.org/10.1016/s0040-4039(97)10722-5
Publikováno v:
ChemInform. 33
Analogues of the neurotransmitter glutamic acid were synthesized by performing a Heck reaction on 4-methylene glutamic acid analogue. This reaction has proved to be highly regio- and stereoselective in the formation of trisubstituted olefin derivativ
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::d1012cce3b1f5ea72677f141d4af7aec
https://doi.org/10.1002/chin.200212230
https://doi.org/10.1002/chin.200212230
Autor:
René Lazaro, Christine Gauzy, Jean Martinez, Stéphane Varray, Frédéric Lamaty, Bérengère Sauvagnat
Publikováno v:
Proceedings of The 4th International Electronic Conference on Synthetic Organic Chemistry.
Ring closing metathesis has been performed for the first time on a soluble poly(ethylene glycol) supported substrate in the presence of Grubbs' catalyst and provided in good yields 6-, 7- and 8-membered ring aminoacid derivatives. The presence of the
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::1f503e9e760e607b321ddb04b4698be1
https://doi.org/10.3390/ecsoc-4-01890
https://doi.org/10.3390/ecsoc-4-01890
Publikováno v:
Journal of Combinatorial Chemistry
Journal of Combinatorial Chemistry, American Chemical Society, 2000, 2 (2), pp.134-142. ⟨10.1021/cc9900605⟩
Scopus-Elsevier
Journal of Combinatorial Chemistry, American Chemical Society, 2000, 2 (2), pp.134-142. ⟨10.1021/cc9900605⟩
Scopus-Elsevier
International audience; A Schiff base activated glycine supported on a soluble polymer (poly(ethylene glycol) (PEG)) was readily alkylated with a wide variety of electrophiles in the presence of a carbonate base in acetonitrile. The presence of the p
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::130e243352e4d57066ce000ee4eb5a49
https://hal.archives-ouvertes.fr/hal-03125693
https://hal.archives-ouvertes.fr/hal-03125693
Autor:
Jean-Alain Fehrentz, N. Mai, J.-L. Aubagnac, Bérengère Sauvagnat, Valérie Rolland, Catherine Pothion, M. L. Roumestant, José Luis Martínez, M. Sadoune, Monique Calmes, J. Daunis, Ph. Viallefont, Y. Vidal, Frédéric Lamaty, Muriel Amblard, René Lazaro, Marielle Paris, Jean-Pierre Lavergne, C. Drouot, Farhate Guenoun, S. Bouifraden, M. El Hadrami, L. Lecointe, P. Chevallet, Christine Enjalbal
Publikováno v:
Amino Acids
Amino Acids, Springer Verlag, 1999, 16, pp.345-379
HAL
Amino Acids, Springer Verlag, 1999, 16, pp.345-379
HAL
Some of the chemistry of amino acids going on in our laboratory (Laboratoire des Amino acides Peptides et Protéines) is described as well as some mass spectrometry methodology for their characterization particularly on solid supports. Several aspect
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c50b3bc557c7ead77260efb8527000da
https://pubmed.ncbi.nlm.nih.gov/10399020
https://pubmed.ncbi.nlm.nih.gov/10399020