Zobrazeno 1 - 8
of 8
pro vyhledávání: '"Béranger Duthion"'
Publikováno v:
ARKIVOC, Vol 2014, Iss 3, Pp 239-255 (2014)
Externí odkaz:
https://doaj.org/article/8cf00b7567b540a6bb407be605f46c73
Publikováno v:
ARKIVOC, Vol 2014, Iss 3, Pp 239-255 (2014)
LY503430, an optically active β-fluoroamine, is a potential therapeutic agent for the Parkinson's disease. Different strategies have been studied to synthesize this molecule using a regioselective and stereospecific rearrangement of β-amino alcohol
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6cb7b2d32553b7ac7da21824f785f363
https://doi.org/10.3998/ark.5550190.p008.252
https://doi.org/10.3998/ark.5550190.p008.252
Publikováno v:
Organic Letters. 12:4620-4623
N,N-Dialkyl-β-amino alcohols were enantiospecifically and regioselectively rearranged by using N,N-diethylaminosulfur trifluoride (DAST) to give optically active β-fluoroamines in excellent yields and enantiomeric excesses. This rearrangement was a
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d79fec63d58a0825415ffca0489d684f
https://doi.org/10.1021/ol1019579
https://doi.org/10.1021/ol1019579
Publikováno v:
ChemInform. 42
β-Amino alcohols of type (I), (III), and (V) undergo a stereospecific reaction with DAST to give rearranged β-fluoroamines with no or very low degree of racemization.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::34557311ca4e714ba07fe501caa62eb6
https://doi.org/10.1002/chin.201106051
https://doi.org/10.1002/chin.201106051
Publikováno v:
ChemInform. 41
This tutorial review focuses on the rearrangement of β-amino alcohols via aziridinium intermediates. It covers the literature from 1947 to January 2009 (55 references). The rearrangement of β-amino alcohols can be performed by activation of the hyd
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::a49231ec72106f217f3b3ca02fa7b8d1
https://doi.org/10.1002/chin.201019248
https://doi.org/10.1002/chin.201019248
Publikováno v:
Chemical Society Reviews
Chemical Society Reviews, Royal Society of Chemistry, 2010, 39, pp.89-102. ⟨10.1039/b806985a⟩
Chemical Society Reviews, Royal Society of Chemistry, 2010, 39, pp.89-102. ⟨10.1039/b806985a⟩
International audience; This tutorial review focuses on the rearrangement of b-amino alcohols via aziridinium intermediates. It covers the literature from 1947 to January 2009 (55 references). The rearrangement of b-amino alcohols can be performed by
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0727b7491989cc64656dc98801812620
https://hal.archives-ouvertes.fr/hal-03228884
https://hal.archives-ouvertes.fr/hal-03228884
Publikováno v:
ChemInform. 40
N-alkyl 1,2-amino alcohols were rearranged stereospecifically by using TFAA/Et3N. This rearrangement has been used to synthesize N-isopropyl-3-(aryloxy)-2-hydroxypropylamines, β-adrenergic blocking agents such as (S)-toliprolol and (S)-propanolol.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::5197571efc9d135d4e6bdbe492c1f305
https://doi.org/10.1002/chin.200951066
https://doi.org/10.1002/chin.200951066
Publikováno v:
Synfacts. 2011:0013-0013
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::dc3c94eaea2cef700f6344dc45a8eef4
https://doi.org/10.1055/s-0030-1258979
https://doi.org/10.1055/s-0030-1258979