Zobrazeno 1 - 10
of 47
pro vyhledávání: '"B, Thirupataiah"'
Akademický článek
Tento výsledek nelze pro nepřihlášené uživatele zobrazit.
K zobrazení výsledku je třeba se přihlásit.
K zobrazení výsledku je třeba se přihlásit.
Autor:
Jetta, Sandeep Kumar, Rapaka, Naimisha, B, Thirupataiah, Gangireddy, Sujeevan Reddy, Navneet, Bung, Arijit, Roy, Gopalakrishnan, Bulusu, Ankita, Mishra, Prem N, Yadav, Parimal, Misra, Manojit, Pal
Publikováno v:
Bioorganic chemistry. 129
Efforts have been devoted for the discovery and development of positive allosteric modulators (PAMs) of 5-HT
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid________::b2ce6cce7ee40df7e58e45459b795009
https://pubmed.ncbi.nlm.nih.gov/36272252
https://pubmed.ncbi.nlm.nih.gov/36272252
Autor:
Gangireddy Sujeevan Reddy, Jetta Sandeep Kumar, B. Thirupataiah, Harshavardhan Bhuktar, Sharda Shukla, Manojit Pal
Publikováno v:
Bioorganic chemistry. 129
The importance of the quinoxaline framework is exemplified by its presence in the well-known drugs such as varenicline, brimonidine, quinacillin, etc. In the past few years, preparation of a variety of organic compounds containing the quinoxaline fra
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::886382e764fd344e80e8937bccbf438b
https://pubmed.ncbi.nlm.nih.gov/36274386
https://pubmed.ncbi.nlm.nih.gov/36274386
Autor:
Jetta Sandeep Kumar, B. Thirupataiah, Jayesh Mudgal, Gangireddy Sujeevan Reddy, Guntipally Mounika, Kazi Amirul Hossain, Marina Rajadurai, Jessy Elizabeth Mathew, Gautham G. Shenoy, Kishore V. L. Parsa, Manojit Pal
Publikováno v:
Chemical Communications. 57:10091-10094
A Pd-catalysed regioselective synthesis of 4,5-disubstituted 7-membered N/O-heterocycles was achieved via the 7-endo-dig cyclization followed by C–C bond formation of 2-(1-alkynyl)phenylacetamide. The ligand/additive free cascade reaction proceeded
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1c47dc332e07b7b9ffdfb20caeab9f3a
https://doi.org/10.1039/d1cc04140a
https://doi.org/10.1039/d1cc04140a
Autor:
B, Thirupataiah, Guntipally, Mounika, Gangireddy, Sujeevan Reddy, Jetta, Sandeep Kumar, Ravikumar, Kapavarapu, Raghavender, Medishetti, Jayesh, Mudgal, Jessy E, Mathew, Gautham G, Shenoy, C, Mallikarjuna Rao, Kiranam, Chatti, Kishore, V L Parsa, Manojit, Pal
Publikováno v:
Bioorganic chemistry. 115
In spite of possessing a wide range of pharmacological properties the anti-inflammatory activities of isoquinolin-1(2H)-ones were rarely known or explored earlier. PDE4 inhibitors on the other hand in addition to their usefulness in treating inflamma
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid________::fab6367eae7262d990036a230948cf98
https://pubmed.ncbi.nlm.nih.gov/34426160
https://pubmed.ncbi.nlm.nih.gov/34426160
Autor:
Kishore V. L. Parsa, Jayesh Mudgal, E.V.V. Shivaji Ramarao, Jetta Sandeep Kumar, Ramudu Bankala, Hari Maduri Doss, Mahaboobkhan Rasool, Manojit Pal, Rajnikanth Sunke, Pushkar Kulkarni, B. Thirupataiah, Ravikumar Kapavarapu, Gautham G. Shenoy, Raghavender Medishetti, Jessy Elizabeth Mathew
Publikováno v:
European Journal of Medicinal Chemistry. 174:198-215
A new class of PDE4 inhibitors were designed and synthesized via the InCl3 mediated heteroarylation of indoles and their further derivatization through the Pd(II)-catalyzed C H activation strategy. This effort allowed us to discover a series of 2-(1H
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::5aec68d5d4d21d2e7d1057a76f345800
https://doi.org/10.1016/j.ejmech.2019.04.020
https://doi.org/10.1016/j.ejmech.2019.04.020
Autor:
Jetta Sandeep, Kumar, Gangireddy Sujeevan, Reddy, Raghavender, Medishetti, Kazi, Amirul Hossain, B, Thirupataiah, Jhansi, Edelli, Shilpak, Dilip Bele, Rebecca, Kristina Edwin, Alex, Joseph, Gautham G, Shenoy, C, Mallikarjuna Rao, Manojit, Pal
Publikováno v:
Bioorganic Chemistry. 124:105857
Addressing the increasing incidences of cancer worldwide along with the multifaceted problem of drug resistance via development of new anticancer agents has become an essential goal. Due to the known cytotoxic effects and reported Akt inhibitory pote
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0a387ad6cbe4e19cbbdaec9295533147
https://doi.org/10.1016/j.bioorg.2022.105857
https://doi.org/10.1016/j.bioorg.2022.105857
Autor:
Gangireddy Sujeevan, Reddy, Rajamanikkam, Kamaraj, Kazi Amirul, Hossain, Jetta Sandeep, Kumar, B, Thirupataiah, Raghavender, Medishetti, N, Sushma Sri, Parimal, Misra, Manojit, Pal
Publikováno v:
Bioorganic chemistry. 116
A series of indole based novel Schiff bases was designed as potential agonists of 5-HT
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid________::f5d0901a08364ac6872ed580ad9bf3ed
https://pubmed.ncbi.nlm.nih.gov/34670330
https://pubmed.ncbi.nlm.nih.gov/34670330
Autor:
B, Thirupataiah, Guntipally, Mounika, Gangireddy Sujeevan, Reddy, Jetta Sandeep, Kumar, Kazi Amirul, Hossain, Raghavender, Medishetti, Snigdha, Samarpita, Mahaboobkhan, Rasool, Jayesh, Mudgal, Jessy E, Mathew, Gautham G, Shenoy, C Mallikarjuna, Rao, Kiranam, Chatti, Kishore V L, Parsa, Manojit, Pal
Publikováno v:
European journal of medicinal chemistry. 221
While anti-inflammatory properties of isocoumarins are known their PDE4 inhibitory potential was not explored previously. In our effort the non-PDE4 inhibitor isocoumarins were transformed into the promising inhibitors via introducing an aminosulfony
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid________::65e763f432a55d48daf040d57ef951bd
https://pubmed.ncbi.nlm.nih.gov/33992926
https://pubmed.ncbi.nlm.nih.gov/33992926
Autor:
B. Thirupataiah, Harshavardhan Bhuktar, Guntipally Mounika, Gangireddy Sujeevan Reddy, Jetta Sandeep Kumar, Sharda Shukla, Kazi Amirul Hossain, Raghavender Medishetti, Snigdha Samarpita, Mahaboobkhan Rasool, P.C. Jagadish, Gautham G. Shenoy, Kishore V.L. Parsa, Manojit Pal
Publikováno v:
Bioorganic Chemistry. 121:105667
In search of potent and new anti-inflammatory agents, we explored a new class of isocoumarin derivatives possessing the 3-oxoalkyl moiety at C-4 position. These compounds were synthesized via the FeCl
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::166deade5a5ccc889bcae0d4b03426d3
https://doi.org/10.1016/j.bioorg.2022.105667
https://doi.org/10.1016/j.bioorg.2022.105667