Zobrazeno 1 - 10
of 20
pro vyhledávání: '"Aydın Salman"'
Publikováno v:
ARKIVOC, Vol 2006, Iss 12, Pp 98-110 (2006)
Externí odkaz:
https://doaj.org/article/a5331abc25d944da9b97e4d6089b7c9d
Publikováno v:
Acta Crystallographica Section E, Vol 64, Iss 10, Pp o1919-o1919 (2008)
In the title compound, C24H28N2O3S, the pendant methyl C atom bonded to the cyclohexane ring is disordered over two sites in a 0.580 (11):0.420 (11) ratio. The cyclohexane ring adopts a distorted chair conformation while the thiazolidine ring has an
Externí odkaz:
https://doaj.org/article/2a864d224cee43d286945bf94d5133fc
Publikováno v:
European Journal of Medicinal Chemistry. 45:1068-1077
3H-Spiro[1,3-benzothiazole-2,3'-indol]-2'(1'H)-ones 3a-c and 4a-e were synthesized from treating the 5-substituted 1H-indole-2,3-diones with 2-aminothiophenol in ethanol. The structures were confirmed by elemental analyses, spectrometry (IR, (1)H NMR
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ad871a6fd44696e2c084f8351f9bec98
https://doi.org/10.1016/j.ejmech.2009.12.001
https://doi.org/10.1016/j.ejmech.2009.12.001
Autor:
Claudiu T. Supuran, Alfonso Maresca, Aydın Salman, Alexandru T. Balaban, Özlen Güzel, Andrea Scozzafava
Publikováno v:
Journal of Medicinal Chemistry. 52:4063-4067
A series of 2-(hydrazinocarbonyl)-3-aryl-1H-indole-5-sulfonamides has been derivatized by reaction with 2,4,6-trimethylpyrylium perchlorate, leading to pyridinium derivatives. The new sulfonamides were evaluated as inhibitors of two beta-carbonic anh
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::aba77f3161511207bfa84d142a48bba4
https://doi.org/10.1021/jm9004016
https://doi.org/10.1021/jm9004016
Publikováno v:
Bioorganic & Medicinal Chemistry. 16:8976-8987
New series of 5-methyl/trifluoromethoxy-1H-indole-2,3-dione 3-thiosemicarbazones 3a-t, 1-methyl-5-methyl/trifluoromethoxy-1H-indole-2,3-dione 3-thiosemicarbazones 4a-y and 5-trifluoromethoxy-1-morpholinomethyl-1H-indole-2,3-dione 3-thiosemicarbazones
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c2eeea3495169bd5cf66740d964c3a20
https://doi.org/10.1016/j.bmc.2008.08.050
https://doi.org/10.1016/j.bmc.2008.08.050
Autor:
Claudia Temperini, Andrea Scozzafava, Aydın Salman, Claudiu T. Supuran, Alessio Innocenti, Özlen Güzel
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 18:152-158
2-(Hydrazinocarbonyl)-3-phenyl-1 H -indole-5-sulfonamide was tested for its interaction with 12 carbonic anhydrase (CA, EC 4.2.1.1) isoforms in the search of compounds with good inhibitory activity against isozymes with medicinal chemistry applicatio
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5bccb56af1ceea666a30351d50195d5c
https://doi.org/10.1016/j.bmcl.2007.10.110
https://doi.org/10.1016/j.bmcl.2007.10.110
Autor:
Aydın Salman, Özlen Güzel
Publikováno v:
Bioorganic & Medicinal Chemistry. 14:7804-7815
Reaction of 2-chloromethylsaccharin with substituted potassium dithiocarbamates and substituted potassium dithiocarbonates furnished (1,1-dioxido-3-oxo-1,2-benzisothiazol-2(3 H )-yl)methyl N , N -disubstituted dithiocarbamates ( 4 – 15 ) and (1,1-d
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ab2ba7b182c234c124e3d45f90552457
https://doi.org/10.1016/j.bmc.2006.07.065
https://doi.org/10.1016/j.bmc.2006.07.065
Publikováno v:
Monatshefte für Chemie - Chemical Monthly. 137:795-801
2-Hydroxy-2,2-diphenylacetohydrazide (2), cyclic ketones, and mercaptoalkanoic acids were converted into 2-hydroxy-N-(3-oxo-1-thia-4-azaspiro[4.4]non/[4.5]dec-4-yl)-2,2-diphenylacetamide derivatives (3, 4) in a one pot procedure. Compounds 3 and 4 we
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::df6261c035bcc128b1a52bbb5ed07605
https://doi.org/10.1007/s00706-006-0475-3
https://doi.org/10.1007/s00706-006-0475-3
Autor:
Aydın Salman, Özlen Güzel
Publikováno v:
Journal of enzyme inhibition and medicinal chemistry. 24(4)
A series of new 2-aryl-4-thiazolidinones (3 and 4) was synthesized from 2-hydroxy-2,2-diphenyl-N'-[(substituted phenyl)methylene]acetohydrazides (2) and mercaptoacetic acid or 2-mercaptopropionic acid. The antimycobacterial activity of these compound
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0406abf36819d521c6dd221b346f8339
https://pubmed.ncbi.nlm.nih.gov/19624255
https://pubmed.ncbi.nlm.nih.gov/19624255
Autor:
Andrea Scozzafava, Özlen Güzel, Alfonso Maresca, Aydın Salman, Claudiu T. Supuran, Alexandru T. Balaban
Publikováno v:
Bioorganicmedicinal chemistry letters. 19(11)
A series of 2-(hydrazinocarbonyl)-3-aryl-1H-indole-5-sulfonamides possessing various 2-, 3- or 4- substituted phenyl groups with methyl-, halogeno- and methoxy-functionalities, or a perfluorophenyl moiety, has been derivatized by reaction with 2,4,6-
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5b018c1ec52fc9d8134fe43f632c4e52
https://pubmed.ncbi.nlm.nih.gov/19410461
https://pubmed.ncbi.nlm.nih.gov/19410461