Zobrazeno 1 - 10
of 25
pro vyhledávání: '"Ayad Kareem, Khan"'
Publikováno v:
Al-Mustansiriyah Journal of Pharmaceutical Sciences, Vol 24, Iss 3 (2024)
Molecular docking simulation and synthesis of five compounds of N2, N4-bis (2-(4-substituted phenyl)-4-oxothiazolidin-3-yl)-3,5-dimethyl-1H-pyrrole-2,4-dicarboxamide was carried out to evaluate their theoretical binding affinities, targeting acute my
Externí odkaz:
https://doaj.org/article/c91f049ac3a14635bb3989309204928c
Publikováno v:
Al-Mustansiriyah Journal of Pharmaceutical Sciences, Vol 24, Iss 1 (2024)
A series of novel 1,3-diazetidin-2-one derivatives were designed, synthesized, and evaluated preliminary (In Vitro) for their cytotoxic activity against the lung (A549) cancer cell line. GOLD software (version 2021.2.0) was used to conduct a molecula
Externí odkaz:
https://doaj.org/article/064ada82445448e7ae5357b745f1a60f
Publikováno v:
Journal of Advanced Pharmaceutical Technology & Research, Vol 14, Iss 3, Pp 176-184 (2023)
A series of eight novels' 1,3-diazetidin-2-ones have been proposed to assess their potential activities. They are intended to examine antiproliferative effects through inhibition of epidermal growth factor receptor (EGFR) expression. These eight comp
Externí odkaz:
https://doaj.org/article/93c7b68a8b0b438fb8c214a990bc8010
Publikováno v:
Al-Mustansiriyah Journal of Pharmaceutical Sciences, Vol 22, Iss 3 (2022)
This review is about 1,2,4-triazoles include their synthesis; their physio-chemical properties, SAR, reactions, derivatives. Finally, their biological activities with a demonstrated showing different requirements to achieve different activity
Externí odkaz:
https://doaj.org/article/1d1ce4072821408c893e890964352c13
Publikováno v:
Al-Mustansiriyah Journal of Pharmaceutical Sciences, Vol 21, Iss 3 (2022)
Infections caused by bacteria have a significant impact on public health. Chemical synthesis of new derivatives of cephalexin inked to amino acid (tryptophan or histidine) through an amide bond at the acyl side chain is achieved. This is a new app
Externí odkaz:
https://doaj.org/article/f84a67dfc69349219dbf11c1d823cda0
Publikováno v:
Al-Mustansiriyah Journal of Pharmaceutical Sciences, Vol 19, Iss 4 (2019)
New two derivatives of 2- methyl benzoimidazole were designed, synthesized and evaluated as a potential cyclooxygenase-2 [COX-2] inhibitors. The synthesized compounds have been recognized according to their spectral FT-IR, 1H-NMR data and physical pr
Externí odkaz:
https://doaj.org/article/b092fce57536454fa99726410acb6082
Autor:
Ayad Kareem Khan
Publikováno v:
Al-Mustansiriyah Journal of Science, Vol 28, Iss 3, Pp 122-133 (2018)
In the present research, a series of some azo compounds (5-9) and 1,2,3-triazoles derived from 2-methyl quinazolin-4(3H)-one were synthesized successfully by stepwise routes includes the following: 3-amino-2-methylquinazolin-4(3H)-one (3) prepared fi
Externí odkaz:
https://doaj.org/article/0a4bc7fa1e964b329f62b29113c814de
Publikováno v:
Al Mustansiriyah Journal of Pharmaceutical Sciences. 22:65-81
This review is about 1,2,4-triazoles include their synthesis; their physio-chemical properties, SAR, reactions, derivatives. Finally, their biological activities with a demonstrated showing different requirements to achieve different activity
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::4474e7b5c088d0afa619221d99120807
https://doi.org/10.32947/ajps.v22i3.890
https://doi.org/10.32947/ajps.v22i3.890
Publikováno v:
Al Mustansiriyah Journal of Pharmaceutical Sciences. 21:25-34
Infections caused by bacteria have a significant impact on public health. Chemical synthesis of new derivatives of cephalexin inked to amino acid (tryptophan or histidine) through an amide bond at the acyl side chain is achieved. This is a new approa
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::04258e47623fedc88771522a0e9c4e99
https://doi.org/10.32947/ajps.v21i3.794
https://doi.org/10.32947/ajps.v21i3.794
Publikováno v:
Al-Mustansiriyah Journal of Pharmaceutical Sciences, Vol 18, Iss 1 (2018)
The synthesis of new NSAIDs with improved efficacy and selectivity towards COX2, which encouraged by the various biological activities of 1,2,4-triazoles and 1,3,4-thiadiazoles. In this experiment, the production of 1,2,4-triazolothiadiazoles deriva
Externí odkaz:
https://doaj.org/article/9ed15369805c419f9a4570acb48fbdee