Zobrazeno 1 - 3
of 3
pro vyhledávání: '"Arnaldo Nalin"'
Autor:
Daniele Andreotti, Roberto Profeta, Emanuele Miserazzi, Simone Spada, Arnaldo Nalin, Alfonso Pozzan
Publikováno v:
Tetrahedron Letters. 51:6526-6530
Treatment of 2-alkyl pyridine N-oxides with acylating reagents represents an established procedure for the introduction of oxygen functionality into alkyl group at the ortho position of N heteroaromatic rings. We have reported the first example of as
Autor:
William Maton, Fernando Bravo, Paolo Stabile, Daniele Andreotti, Arnaldo Nalin, Simone Spada, Roberto Profeta, Alcide Perboni, Federica Stazi, Damiano Castoldi, Anna Mingardi, Stefano Provera, Emanuele Miserazzi, Nicola Giubellina, Mario Mattioli, Roberta Pachera, Pieter Westerduin, Arianna Ribecai, Simon M. Bryant, Lucilla Turco, Angelo M. Manzo
Publikováno v:
Organic Process Research & Development. 14:1239-1247
An efficient scalable route to synthesize the enantiomerically pure tert-butyl-(1R,4S,6R)-4-(hydroxymethyl)-3-azabicyclo[4.1.0]heptane-3-carboxylate is described. Compared to the original routes, significant improvements were made by using an innovat
Autor:
Stefania Contini, Emiliangelo Ratti, Aldo Feriani, Frank E. Blaney, David G. Trist, Karen L Roberts, Fabio Maria Sabbatini, Romano Di Fabio, Damiano Ghirlanda, Daniele Donati, Angela Worby, Stefano Provera, Mario Mattioli, Yves St-Denis, Roberto Arban, Elettra Fazzolari, Emiliano Castiglioni, Francesca Pavone, Simone Spada, Enza Di Modugno, Carla Marchioro, Giovanni Bernasconi, Arnaldo Nalin, Anna Mingardi, Anna Maria Capelli, Daniele Andreotti, Simone Braggio, Gabriella Gentile
Publikováno v:
Journal of Medicinal Chemistry. 51:7370-7379
To identify new CRF(1) receptor antagonists, an attempt to modify the bis-heterocycle moiety present in the top region of the dihydropyrrole[2,3]pyridine template was made following new pharmacophoric hypothesis on the CRF(1) receptor antagonists bin