Zobrazeno 1 - 10
of 71
pro vyhledávání: '"Armin Walser"'
Autor:
Armin Walser, Silke Herok, Uwe Heinelt, Peter-Michael Blohm, Hans Matter, Detlev Schneider, Volker Brachvogel, Petra Lönze, Alexander Liesum, Elisabeth Defossa, Andrea Müller, Herman Schreuder, Peter Wildgoose, Fahad Al-Obeidi
Publikováno v:
Journal of Medicinal Chemistry. 45:2749-2769
A series of 138 nonchiral 3-amidinobenzyl-1H-indole-2-carboxamides and analogues as inhibitors of the blood coagulation enzyme factor Xa (fXa) were designed, synthesized, and investigated by X-ray structure analysis and 3D quantitative structure-acti
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a726565af642ccfaba27630b1476d74a
https://doi.org/10.1021/jm0111346
https://doi.org/10.1021/jm0111346
Autor:
James A. Ostrem, Michal Lebl, Peter Strop, Fahad Al-Obeidi, Armin Walser, Pavel Safar, Alena Stierandova
Publikováno v:
Expert Opinion on Therapeutic Patents. 9:931-953
The invention provides compounds which specifically inhibit factor Xa activity. The compounds consist of the structure X1 -YIR-X2, wherein X1 is H, acyl, alkyl, acylalkyl, arylalkyl or one or more amino acids, and X2 is a modified C-terminal group, o
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::524f02e9b3202161fcf9377de414d147
https://doi.org/10.1517/13543776.9.7.931
https://doi.org/10.1517/13543776.9.7.931
Autor:
Carl J. Mason, Armin Walser, Bob Yaremko, Herman J. Crowley, T. Flynn, Margaret O'Donnell, Catherine Maresca
Publikováno v:
ChemInform. 22
A series of [1,2,4]triazolo[4,3-alpha][1,4]benzodiazepines bearing an ethynyl functionality at the 8-position and the isosteric thieno[3,2-f][1,2,4]triazolo[4,3-alpha][1,4]diazepines were prepared and evaluated as antagonists of platelet activating f
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::dc9ac877d5a8a2f09df3badd02e3557e
https://doi.org/10.1002/chin.199127208
https://doi.org/10.1002/chin.199127208
Publikováno v:
ChemInform. 22
The syntheses of two novel pentacyclic ring systems, the thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepino-[4,5-a]benzimidazole and the indazolo[2,3-d][1,2,4]triazolo[4,3-a][1,4]benzodiazepine are described. Attachment of a propargyl linked quinolino
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::333361a7b13fec7e77e6fe9fb5535550
https://doi.org/10.1002/chin.199147204
https://doi.org/10.1002/chin.199147204
Autor:
T. Flynn, Armin Walser
Publikováno v:
ChemInform. 24
The syntheses of two enantiomeric tetracyclic compounds, the thieno[3,2-f][pyrrolo[2,1-c][1,2,4]triazolo[4,3-a][1,4]diazepines 10a and 10b are described. Testing of these enantiomers as inhibitors of platelet activating factor (PAF) revealed good ena
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::f9598d3c91e7248095b3ba1731bc5e58
https://doi.org/10.1002/chin.199318235
https://doi.org/10.1002/chin.199318235
Autor:
T. Flynn, Armin Walser
Publikováno v:
Journal of Heterocyclic Chemistry. 29:1477-1480
The syntheses of two enantiomeric tetracyclic compounds, the thieno[3,2-f][pyrrolo[2,1-c][1,2,4]triazolo[4,3-a][1,4]diazepines 10a and 10b are described. Testing of these enantiomers as inhibitors of platelet activating factor (PAF) revealed good ena
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::af46ac51b648f7e72349799b6b5d6f02
https://doi.org/10.1002/jhet.5570290619
https://doi.org/10.1002/jhet.5570290619
Publikováno v:
Journal of Heterocyclic Chemistry. 28:1121-1125
The syntheses of two novel pentacyclic ring systems, the thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepino-[4,5-a]benzimidazole and the indazolo[2,3-d][1,2,4]triazolo[4,3-a][1,4]benzodiazepine are described. Attachment of a propargyl linked quinolino
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::25e58c6e3dc2de1cad6315be4bdf71d6
https://doi.org/10.1002/jhet.5570280448
https://doi.org/10.1002/jhet.5570280448
Autor:
Armin Walser, R. Ian Fryer
Publikováno v:
Chemistry of Heterocyclic Compounds: Bicyclic Diazepines: Diazepines with an Additional Ring, Volume 50
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::e6393725e5517f3eba2e557fdb29e11a
https://doi.org/10.1002/9780470187371.ch3
https://doi.org/10.1002/9780470187371.ch3
Autor:
Armin Walser, R. Ian Fryer
Publikováno v:
Chemistry of Heterocyclic Compounds: Bicyclic Diazepines: Diazepines with an Additional Ring, Volume 50
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::3c1cc5853ec9d69b537ad0ddf17cba56
https://doi.org/10.1002/9780470187371.ch1
https://doi.org/10.1002/9780470187371.ch1
Autor:
R. Ian Fryer, Armin Walser
Publikováno v:
Chemistry of Heterocyclic Compounds: A Series Of Monographs ISBN: 9780470187371
Chemistry of Heterocyclic Compounds: Bicyclic Diazepines: Diazepines with an Additional Ring, Volume 50
Chemistry of Heterocyclic Compounds: Bicyclic Diazepines: Diazepines with an Additional Ring, Volume 50
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::521465997672a74354c5647f7bdf2b3d
https://doi.org/10.1002/9780470187371.ch8
https://doi.org/10.1002/9780470187371.ch8