Zobrazeno 1 - 10
of 95
pro vyhledávání: '"Antonio J. Moreno-Vargas"'
Publikováno v:
Catalysts, Vol 12, Iss 8, p 876 (2022)
Iminosugar derivatives containing a pyrrolidine-phosphine moiety were prepared from carbohydrates and used as catalysts in the [3 + 2] cycloaddition reaction between alkyl allenoates and electron-deficient imines. The corresponding 1,2,3,5-tetrasubst
Externí odkaz:
https://doaj.org/article/65af786b14ae45aeb5a494f733123ad2
Autor:
Camilla Matassini, Stefania Mirabella, Andrea Goti, Inmaculada Robina, Antonio J. Moreno-Vargas, Francesca Cardona
Publikováno v:
Beilstein Journal of Organic Chemistry, Vol 11, Iss 1, Pp 2631-2640 (2015)
The synthesis of new multivalent architectures based on a trihydroxypiperidine α-fucosidase inhibitor is reported herein. Tetravalent and nonavalent dendrimers were obtained by means of the click chemistry approach involving the copper azide-alkyne-
Externí odkaz:
https://doaj.org/article/4f72bfa8b0294aa59ed0eeef97c7a692
Autor:
Pilar Elías-Rodríguez, Elena Moreno-Clavijo, Sebastián Carrión-Jiménez, Ana T. Carmona, Antonio J. Moreno-Vargas, Irene Caffa, Fabrizio Montecucco, Michele Cea, Alessio Nencioni, Inmaculada Robina
Publikováno v:
ARKIVOC, Vol 2014, Iss 3, Pp 197-214 (2014)
Externí odkaz:
https://doaj.org/article/f17bc83cfa244c88aba7b15fdd996842
Publikováno v:
CHIMIA, Vol 65, Iss 1-2 (2011)
Since the discovery of the 'formose reaction' by Butlerow,[1] total synthesis of carbohydrates has undergone rapid development. The most important methods for the asymmetric synthesis of monosaccharides and analogues of biological importance are pres
Externí odkaz:
https://doaj.org/article/fa03de143c9a4d6c802699198311f1c9
Publikováno v:
CHIMIA, Vol 65, Iss 1-2 (2011)
We present herein a selection of ingenious methods that have been developed to convert inexpensive furan, pyrrole and unsaturated hydrocarbons into enantiomerically enriched monosaccharides and analogues of biological interest.
Externí odkaz:
https://doaj.org/article/323d73966526480c9813456e874f3131
Autor:
Elena Moreno-Clavijo, Ana T. Carmona, Antonio J. Moreno-Vargas, Lidia Molina, Inmaculada Robina
Publikováno v:
CHIMIA, Vol 65, Iss 1-2 (2011)
A review dealing with 1,4-iminoalditol (hydroxylated pyrrolidine) derivatives as inhibitors of ?-L-fucosidases including the different synthetic approaches for their preparation as well as their inhibitory properties is presented.
Externí odkaz:
https://doaj.org/article/60015e07918d488cbbaaccb369fbefca
Autor:
Simone Fratta, Paulina Biniecka, Antonio J. Moreno-Vargas, Ana T. Carmona, Aimable Nahimana, Michel A. Duchosal, Francesco Piacente, Santina Bruzzone, Irene Caffa, Alessio Nencioni, Inmaculada Robina
Publikováno v:
European Journal of Medicinal Chemistry. 250:115170
Cancer cells are highly dependent on Nicotinamide phosphoribosyltransferase (NAMPT) activity for proliferation, therefore NAMPT represents an interesting target for the development of anti-cancer drugs. Several compounds, such as FK866 and CHS828, we
Autor:
Jian-Fei Bai, Somi Reddy Majjigapu, Bernard Sordat, Sophie Poty, Pierre Vogel, Pilar Elías-Rodríguez, Antonio J. Moreno-Vargas, Ana T. Carmona, Irene Caffa, Moustafa Ghanem, Amr Khalifa, Fiammetta Monacelli, Michele Cea, Inmaculada Robina, Consuelo Gajate, Faustino Mollinedo, Axel Bellotti, Aimable Nahimana, Michel Duchosal, Alessio Nencioni
Publikováno v:
Digital.CSIC. Repositorio Institucional del CSIC
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11 p.- 2 fig.-4 tab.-8 schem.-1 graph. abst.
Pancreatic ductal adenocarcinoma (PDAC) is one of the most lethal diseases for which chemotherapy has not been very successful yet. FK866 ((E)-N-(4-(1-benzoylpiperidin-4-yl)butyl)-3-(pyridin-3-yl)acry
Pancreatic ductal adenocarcinoma (PDAC) is one of the most lethal diseases for which chemotherapy has not been very successful yet. FK866 ((E)-N-(4-(1-benzoylpiperidin-4-yl)butyl)-3-(pyridin-3-yl)acry
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7c4ff75c600149bbef14b882ef0bbb10
http://hdl.handle.net/10261/274793
http://hdl.handle.net/10261/274793
Autor:
Valeria Pingitore, Macarena Martínez-Bailén, Ana T. Carmona, Zuzana Mészáros, Natalia Kulik, Kristýna Slámová, Vladimír Křen, Pavla Bojarová, Inmaculada Robina, Antonio J. Moreno-Vargas
Publikováno v:
idUS. Depósito de Investigación de la Universidad de Sevilla
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Two libraries of mono- and dimeric pyrrolidine iminosugars were synthesized by CuAAC and (thio)urea-bond-forming reactions from the respective azido/aminohexylpyrrolidine iminosugar precursors. The resulting monomeric and dimeric compounds were scree
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7a1c411d14bd2626201a144f2b08835a
Autor:
Emily A. Hoyt, Gonzalo Jiménez-Osés, Claudio D. Navo, Ester Jiménez-Moreno, Antonio J. Moreno-Vargas, Alena Istrate, Inmaculada Robina, Enrique Gil de Montes, Gonçalo J. L. Bernardes, Francisco Corzana
Publikováno v:
Angewandte Chemie International Edition. 59:6196-6200
An azanorbornadiene bromovinyl sulfone reagent for cysteine-selective bioconjugation has been developed. Subsequent reaction with dipyridyl tetrazine leads to bond cleavage and formation of a pyrrole-linked conjugate. The latter involves ligation of