Zobrazeno 1 - 7
of 7
pro vyhledávání: '"Anne Vialettes"'
Autor:
Marie Anne Vialettes
Publikováno v:
Adolescence. :127-138
L’image d’une guirlande de bonshommes de papier vient en support au psychologue clinicien exercant en etablissement penitentiaire pour mineurs pour penser des adolescents pris dans une chaine marquee par le fraternel, l’horizontalite et la norm
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::44bd7218e2ac85566487f6b1cfe18a92
https://doi.org/10.3917/ado.087.0127
https://doi.org/10.3917/ado.087.0127
Autor:
Chris Proffitt, Johnny Y. Nagasawa, Levan Darjania, Eric Stefan, Ryan Stansfield, Sean O'Brien, Nicole Streiner, Jeffrey P. Whitten, Joshua R. Bliesath, Peter C. Chua, Caroline B. Ho, Pauline Bourbon, William G. Rice, Fabrice Pierre, Adam Siddiqui-Jain, Ta Kung Chen, Kenna Anderes, Anne Vialettes, Mustapha Haddach, David M. Ryckman, Michael K. Schwaebe, Denis Drygin, Jerome Michaux, May Omori
Publikováno v:
Molecular and Cellular Biochemistry. 356:37-43
In this article we describe the preclinical characterization of 5-(3-chlorophenylamino) benzo[c][2,6]naphthyridine-8-carboxylic acid (CX-4945), the first orally available small molecule inhibitor of protein CK2 in clinical trials for cancer. CX-4945
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8047df7df0af652af52401571f4b18f3
https://doi.org/10.1007/s11010-011-0956-5
https://doi.org/10.1007/s11010-011-0956-5
Autor:
Johnny Y. Nagasawa, Michael K. Schwaebe, Fabrice Pierre, Mustapha Haddach, Anne Vialettes, David M. Ryckman
Publikováno v:
Tetrahedron Letters. 52:1096-1100
Quinolone esters are readily converted into the corresponding amides using aluminum chloride at room temperature in excellent yields and purities. The method is both general and scalable to multi-kilogram quantities.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::c01e22faf3b70c36f997b52049fe13d1
https://doi.org/10.1016/j.tetlet.2010.12.108
https://doi.org/10.1016/j.tetlet.2010.12.108
Autor:
Peter C. Chua, Michael K. Schwaebe, Johnny Y. Nagasawa, Anne Vialettes, Jeffrey P. Whitten, Fabrice Pierre
Publikováno v:
Tetrahedron Letters. 49:4437-4442
A novel and efficient synthesis of 5-oxo-6-carboxy-naphthyridines is reported in this Letter along with a discussion of scope and limitations. Activated 3-nicotinic acids readily acylate the magnesium anion of 2-(benzothiazol-2-yl) or 2-(benzimidazol
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::269ff3db6ed32096f1a6a4ca7c08854c
https://doi.org/10.1016/j.tetlet.2008.05.005
https://doi.org/10.1016/j.tetlet.2008.05.005
Autor:
Jeffrey P. Whitten, Katy Trent, Caroline B. Ho, Kenna Anderes, Anne Vialettes, May Omori, Adam Siddiqui-Jain, Sean O'Brien, Johnny Y. Nagasawa, Michael K. Schwaebe, Eric Stefan, William G. Rice, Pauline Bourbon, Peter C. Chua, Ta Kung Chen, Chris Proffitt, Fabrice Pierre, Denis Drygin, Mustapha Haddach, Jerome Michaux, Nicole Streiner, Levan Darjania, David M. Ryckman, Ryan Stansfield, Josh Bliesath
Publikováno v:
Journal of medicinal chemistry. 54(2)
Herein we chronicle the discovery of CX-4945 (25n), a first-in-class, orally bioavailable ATP-competitive inhibitor of protein kinase CK2 in clinical trials for cancer. CK2 has long been considered a prime cancer drug target because of the roles of d
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::381f31afdb18ac8eca61f6768c660619
https://pubmed.ncbi.nlm.nih.gov/21174434
https://pubmed.ncbi.nlm.nih.gov/21174434
Autor:
Anne Vialettes, Fabrice Pierre, Peter C. Chua, Michael K. Schwaebe, Jeffrey P. Whitten, Johnny Y. Nagasawa
Publikováno v:
ChemInform. 39
A novel and efficient synthesis of 5-oxo-6-carboxy-naphthyridines is reported in this Letter along with a discussion of scope and limitations. Activated 3-nicotinic acids readily acylate the magnesium anion of 2-(benzothiazol-2-yl) or 2-(benzimidazol
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::0fb2575750a69ed00403e5b42a198365
https://doi.org/10.1002/chin.200842138
https://doi.org/10.1002/chin.200842138
Autor:
Fabrice Pierre, Peter C. Chua, Sean E. O’Brien, Adam Siddiqui-Jain, Pauline Bourbon, Mustapha Haddach, Jerome Michaux, Johnny Nagasawa, Michael K. Schwaebe, Eric Stefan, Anne Vialettes, Jeffrey P. Whitten, Ta Kung Chen, Levan Darjania, Ryan Stansfield, Kenna Anderes, Josh Bliesath, Denis Drygin, Caroline Ho, May Omori
Publikováno v:
Journal of Medicinal Chemistry; Jan2011, Vol. 54 Issue 2, p635-654, 20p