Zobrazeno 1 - 2
of 2
pro vyhledávání: '"Anna Bassil"'
Autor:
Rebecca Furze, Judit Molnar, Nigel Parr, Faiz Ahmad, Yvette Henry, David Howe, Rajendra Singh, Martin Toal, Anna Bassil, Sharon Bernard, Robert Davis, Adele Gibson, Claire Maller, Catriona Sharp, David Tough, Rab Prinjha, Huw Lewis
AIM: To improve the tolerability and therapeutic application of histone deacetylase inhibitors (HDACi), by application of an esterase-sensitive motif (ESM), to target pharmacological activity directly to mononuclear myeloid cells expressing the proce
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::b66724da03939ab05a2278fedf0bf4f6
https://doi.org/10.22541/au.164254165.50219816/v1
https://doi.org/10.22541/au.164254165.50219816/v1
Autor:
Lee A, Harrison, Stephen J, Atkinson, Anna, Bassil, Chun-Wa, Chung, Paola, Grandi, James R J, Gray, Etienne, Levernier, Antonia, Lewis, David, Lugo, Cassie, Messenger, Anne-Marie, Michon, Darren J, Mitchell, Alex, Preston, Rab K, Prinjha, Inmaculada, Rioja, Jonathan T, Seal, Simon, Taylor, Ian D, Wall, Robert J, Watson, James M, Woolven, Emmanuel H, Demont
Publikováno v:
Journal of medicinal chemistry. 64(15)
Domain-specific BET bromodomain ligands represent an attractive target for drug discovery with the potential to unlock the therapeutic benefits of antagonizing these proteins without eliciting the toxicological aspects seen with pan-BET inhibitors. W
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid________::29838ca81add590d8ccf661d7c0b5e04
https://pubmed.ncbi.nlm.nih.gov/34232650
https://pubmed.ncbi.nlm.nih.gov/34232650
