Zobrazeno 1 - 2
of 2
pro vyhledávání: '"Ann Yu-Jung Shih"'
Autor:
Kai Nakamura, Qiang Li, Tyzoon K. Nomanbhoy, Ann Yu-Jung Shih, Helge Weissig, Oana Cociorva, Lan Pham, John W. Kozarich, Yi Hu, Melissa C. Zhang, Marek Liyanage, Julia Cajica, Kevin R. Shreder, Arwin Aban, Bei Li
Publikováno v:
Bioorganicmedicinal chemistry letters. 23(18)
As the result of a rhJNK1 HTS, the imidazo[1,2-a]quinoxaline 1 was identified as a 1.6 μM rhJNK1 inhibitor. Optimization of this compound lead to AX13587 (rhJNK1 IC50 = 160 nM) which was co-crystallized with JNK1 to identify key molecular interactio
Autor:
Patrick R. Hof, Brea Midthune, Simone Eggert, Sheue-Houy Tyan, Dara L. Dickstein, Edward H. Koo, Ann Yu-Jung Shih, Jessica J. Walsh
Publikováno v:
Alzheimer's & Dementia. 6