Zobrazeno 1 - 10
of 21
pro vyhledávání: '"Anita Gulbe"'
Autor:
Ilona Domracheva, Ruslan Muhamadejev, Marina Petrova, Edvards Liepinsh, Anita Gulbe, Irina Shestakova, Gunars Duburs, Pavel Arsenyan
Publikováno v:
Toxicology Reports, Vol 2, Iss C, Pp 377-383 (2015)
Addition of DMPC considerably inhibits the degradation of Carmofur in neutral phosphate buffer solutions and this drug becomes less influenced by pH. Carmofur stabilization at neutral pH caused by DMPC addition for in vitro studies was characterized
Externí odkaz:
https://doaj.org/article/2efb2ea3afd140c9b3a1669e338b32b8
Autor:
Martins Rucins, Pavels Dimitrijevs, Klavs Pajuste, Oksana Petrichenko, Ludmila Jackevica, Anita Gulbe, Signe Kibilda, Krisjanis Smits, Mara Plotniece, Dace Tirzite, Karlis Pajuste, Arkadij Sobolev, Janis Liepins, Ilona Domracheva, Aiva Plotniece
Publikováno v:
Pharmaceutics, Vol 11, Iss 3, p 115 (2019)
The design of nanoparticle delivery materials possessing biological activities is an attractive strategy for the development of various therapies. In this study, 11 cationic amphiphilic 4-(N-alkylpyridinium)-1,4-dihydropyridine (1,4-DHP) derivatives
Externí odkaz:
https://doaj.org/article/e6bb0efd137046cc8539b508b29ed21d
Autor:
Tatjana Beresneva, Anatoly Mishnev, Elina Jaschenko, Irina Shestakova, Anita Gulbe, Edgars Abele
Publikováno v:
ARKIVOC, Vol 2012, Iss 9, Pp 185-194 (2012)
Externí odkaz:
https://doaj.org/article/baef39b3bf4d4bd7a18a3cb9d6e64bbf
Autor:
Edgars Abele, Lena Golomba, Tatjana Beresneva, Julija Visnevska, Elina Jaschenko, Irina Shestakova, Anita Gulbe, Solveiga Grinberga, Sergey Belyakov, Ramona Abele
Publikováno v:
ARKIVOC, Vol 2012, Iss 8, Pp 49-61 (2012)
Externí odkaz:
https://doaj.org/article/782f224901894bcdb1dfb7fdb8b8e5ff
Publikováno v:
New Journal of Chemistry. 43:11851-11864
The general aim of the current research is to find novel non-toxic small molecules with antimetastatic activity. Herein we present a series of novel selenopheno[2,3-f]coumarins with low cytotoxicity profiles against cancer cells with different nature
Autor:
L. Golomba, Edgars Abele, Elina Jaschenko, Anita Gulbe, Ilona Domracheva, T. Beresneva, Ramona Abele
Publikováno v:
Current Organic Synthesis. 15:1154-1160
Aims and Objectives: The aim of the research is to obtain and to investigate the cytotoxicity of a novel class of non-toxic oximes – derivatives of N-(benzo[4,5]imidazo[2,1-b]thiazol-3-ylmethoxy)-ω- (hetarylsulfanyl)-alkanamidines. Materials and M
Autor:
Janis Liepins, Pavels Dimitrijevs, Mara Plotniece, Dace Tirzite, Signe Kibilda, Anita Gulbe, Ilona Domracheva, Arkadij Sobolev, Oksana Petrichenko, Ludmila Jackevica, Karlis Pajuste, Klavs Pajuste, Martins Rucins, Aiva Plotniece, Krisjanis Smits
Publikováno v:
Pharmaceutics
Volume 11
Issue 3
Pharmaceutics, Vol 11, Iss 3, p 115 (2019)
Volume 11
Issue 3
Pharmaceutics, Vol 11, Iss 3, p 115 (2019)
The design of nanoparticle delivery materials possessing biological activities is an attractive strategy for the development of various therapies. In this study, 11 cationic amphiphilic 4-(N-alkylpyridinium)-1,4-dihydropyridine (1,4-DHP) derivatives
Publikováno v:
Chemistry of Heterocyclic Compounds. 52:551-554
The antioxidant activity of selenium-containing analogs of raloxifene was studied by the ability to scavenge 2,2-diphenyl-1-picrylhydrazyl, superoxide, nitric oxide, and peroxyl radicals. These compounds exhibited similar scavenging properties as res
Autor:
Luba Ignatovich, Anita Gulbe, Sergey Belyakov, Zhanna Rudevica, I. Shestakova, Juris Popelis, Jana Spura, Ilona Domrachova, Ainars Leonchiks, Velta Muravenko
Publikováno v:
Applied Organometallic Chemistry. 29:756-763
New 6,6-dimethyl-2-oxo-4-{2-[5-alkylsilyl(germyl)]furan(thiophen)-2-yl}vinyl-5,6-dihydro-2H-pyran-3-carbonitriles (IC50: 1–6 µg ml−1) have been prepared by the condensation of corresponding silicon- and germanium-containing furyl(thienyl)-2-carb
Autor:
Anita Gulbe, Edvards Liepinsh, Ruslan Muhamadejev, Pavel Arsenyan, Ilona Domracheva, Gunars Duburs, I. Shestakova, Marina Petrova
Publikováno v:
Toxicology Reports
Toxicology Reports, Vol 2, Iss C, Pp 377-383 (2015)
Toxicology Reports, Vol 2, Iss C, Pp 377-383 (2015)
Graphical abstract
Highlights • DMPC addition stabilizes Carmofur at neutral pH. • We report considerable increase of Carmofur cytotoxicity. • It opens a way for the drug delivery of Carmofur in neutral and basic media.
Addition of DM
Highlights • DMPC addition stabilizes Carmofur at neutral pH. • We report considerable increase of Carmofur cytotoxicity. • It opens a way for the drug delivery of Carmofur in neutral and basic media.
Addition of DM