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pro vyhledávání: '"Anisa, Gravelle"'
Autor:
Maria Angeles, Martinez-Grau, Isabel C Gonzalez, Valcarcel, Julie V, Early, Richard Klaus, Gessner, Candice Soares, de Melo, Eva Maria Martin, de la Nava, Aaron, Korkegian, Yulia, Ovechkina, Lindsay, Flint, Anisa, Gravelle, Jeff W, Cramer, Prashant V, Desai, Leslie J, Street, Joshua, Odingo, Thierry, Masquelin, Kelly, Chibale, Tanya, Parish
Publikováno v:
Bioorganic & Medicinal Chemistry Letters
Graphical abstract
Highlights • We conducted SAR for the aryl-oxadiazole series with anti-bacterial activity against Mycobacterium tuberculosis. • Improved compounds have sub-micromolar butyrate-specific activity. • Compounds are not cytot
Highlights • We conducted SAR for the aryl-oxadiazole series with anti-bacterial activity against Mycobacterium tuberculosis. • Improved compounds have sub-micromolar butyrate-specific activity. • Compounds are not cytot