Zobrazeno 1 - 10
of 69
pro vyhledávání: '"Angelo Scatturin"'
Autor:
Angelo Scatturin, Vertuani Gianni, Rita Pecoraro, Alessandro Dalpiaz, Marisa Boggian, Maria Ferretti, Susanna Spisani
Publikováno v:
Arzneimittelforschung. 49:873-877
The conformation of several Phe-D-Leu-Phe-D-Leu-Phe analogues was analyzed using infrared absorption and circular dichroism. Their effect on human neutrophils was verified by receptor binding and chemotaxis assays. The results demonstrate that the co
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::75f954584cba3321037cc71e264386ba
https://doi.org/10.1055/s-0031-1300519
https://doi.org/10.1055/s-0031-1300519
Publikováno v:
International Journal of Peptide and Protein Research. 34:409-415
The tripeptide N-formyl-L-Met-L-Leu-L-Phe-OMe (FMLP-OMe) crystallizes in the orthorhombic system, space group P 2(1)2(1)2(1), with the following unit-cell parameters: a = 21.727, b = 21.836, c = 5.133 A, Z = 4. The structure has been solved and refin
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e8f52a48a5f849e10ec43c65efbfceeb
https://doi.org/10.1111/j.1399-3011.1989.tb00710.x
https://doi.org/10.1111/j.1399-3011.1989.tb00710.x
Autor:
C. Falcomer, G. Pochetti, Vertuani G, Maurizio Ricci, M. Boggian, C. Ross, Angelo Scatturin, S. Cerrini
Publikováno v:
Scopus-Elsevier
The conformational behaviour of the peptide antibiotic leucinostatin A has been studied in solvents of different polarity using circular dichroism (CD) and infrared (i.r.) absorption. I.r. studies provided evidence of an intramolecularly hydrogen-bon
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b3140552afbedd611ef8172401069cbe
https://doi.org/10.1111/j.1399-3011.1989.tb00205.x
https://doi.org/10.1111/j.1399-3011.1989.tb00205.x
Autor:
Gaia Colombo, Fabrizio Bortolotti, Sergio Tanganelli, Luca Ferraro, Paolo Giunchedi, Angelo Scatturin, Alessandro Dalpiaz, Paola Russo, Enea Menegatti, Elisabetta Gavini
Publikováno v:
Journal of Pharmaceutical Sciences. 97:4889-4903
N(6)-cyclopentyladenosine (CPA) has neuronal anti-ischemic properties, but it is not absorbed into the brain from the bloodstream, where it shows poor stability and induces side effects. Microparticulate drug delivery systems designed for CPA nasal a
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9e8a5f4709d216cf1535d934718048f8
https://doi.org/10.1002/jps.21335
https://doi.org/10.1002/jps.21335
Autor:
Francesca Corradini, Markus Drechsler, Elisa Sivieri, Alessandra Rossi, Elisabetta Esposito, Rita Cortesi, Enea Menegatti, Angelo Scatturin
Publikováno v:
International Journal of Pharmaceutics. 339:52-60
In the present study, the preparation, characterization and activity of non-phospholipid vesicles (NPV) containing three aminoacid-based molecules were described. As model compounds trypsin, bovine basic pancreatic inhibitor and polylysine rich pepti
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::97553bea044762915230a72769abcfbc
https://doi.org/10.1016/j.ijpharm.2007.02.024
https://doi.org/10.1016/j.ijpharm.2007.02.024
Autor:
F. Vitali, Martina Scaglianti, Fabrizio Bortolotti, Alessandro Dalpiaz, Barbara Pavan, Stefano Manfredini, Angelo Scatturin, Carla Biondi
Publikováno v:
International Journal of Pharmaceutics. 291:171-181
Diclofenac (Diclo), its ascorbic acid (AA) or 6-amino-AA (AA-NH2) pro-drugs (AA-Diclo or AA-NH-Diclo) were prepared and evaluated on human retinal pigment epithelium (HRPE) cells to investigate their ability to interact with the vitamin C transporter
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::323467ac310fcb9688484f29c25e5a30
https://doi.org/10.1016/j.ijpharm.2004.07.054
https://doi.org/10.1016/j.ijpharm.2004.07.054
Autor:
Silvia Vertuani, Stefano Manfredini, Martina Scaglianti, Giuliano Marzola, Angelo Scatturin, Federica Vitali, Luca Ferraro, Carla Biondi, Barbara Pavan, Alessandro Dalpiaz, Puttur D. Prasad, Fabrizio Bortolotti, Sergio Tanganelli
Publikováno v:
European Journal of Pharmaceutical Sciences. 24:259-269
Ascorbic acid (AA) or 6-Br-ascorbate (BrAA) conjugation has been investigated as a tool to improve brain drug delivery by the Vitamin C transporter SVCT2. To this aim, the effects of AA- or BrAA-conjugation on drug affinity and uptake have been asses
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9fde07739b263186a464f21741e505d2
https://doi.org/10.1016/j.ejps.2004.10.014
https://doi.org/10.1016/j.ejps.2004.10.014
Autor:
Federica Vitali, Martina Scaglianti, Puttur D. Prasad, Sergio Tanganelli, Carla Biondi, Luca Ferraro, Fabrizio Bortolotti, Stefano Manfredini, Angelo Scatturin, Barbara Pavan, Alessandro Dalpiaz
Publikováno v:
Journal of Pharmaceutical Sciences. 93:78-85
Continuing our studies on SVCT2 ascorbic acid (AA) transporter-mediated drug delivery of neurotropic agents, we have now investigated the in vitro intracellular uptake of Diclofenac (Diclo) and its conjugate (AA-Diclo), both characterized by high aff
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::3677a3263be52b131f510dca6f1e25e8
https://doi.org/10.1002/jps.10532
https://doi.org/10.1002/jps.10532
Autor:
Barbara Malawska, Angelo Scatturin
Publikováno v:
Mini-Reviews in Medicinal Chemistry. 3:341-348
The chemical diversity and various mechanisms of action of anticonvulsants make it difficult to identify a common pharmacophore. The present review outlines different pharmacophore models for anticonvulsant activity with emphasis on the development o
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b309609e0e37c9681febb742fa291c51
https://doi.org/10.2174/1389557033488088
https://doi.org/10.2174/1389557033488088
Autor:
A. Dalpiaz, Maria Angela Vandelli, Angelo Scatturin, Carla Biondi, Barbara Pavan, Flavio Forni
Publikováno v:
International Journal of Pharmaceutics. 242:115-120
We report a preliminary study evaluating the encapsulation modalities in microparticles of the antiischemic drug N(6)-cyclopentyladenosine (CPA). The effects of release systems have been evaluated on the stability in human whole blood of CPA and its
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e527a7a4289af484640bddefea4ffe41
https://doi.org/10.1016/s0378-5173(02)00179-5
https://doi.org/10.1016/s0378-5173(02)00179-5