Zobrazeno 1 - 10
of 10
pro vyhledávání: '"Anelia Mavrova"'
Autor:
Kameliya Anichina, Anelia Mavrova, Dimitar Vuchev, Galya Popova-Daskalova, Giada Bassi, Arianna Rossi, Monica Montesi, Silvia Panseri, Filip Fratev, Emilia Naydenova
Publikováno v:
Pharmaceuticals, Vol 16, Iss 11, p 1518 (2023)
Benzimidazole anthelmintic drugs hold promise for repurposing as cancer treatments due to their interference with tubulin polymerization and depolymerization, manifesting anticancer properties. We explored the potential of benzimidazole compounds wit
Externí odkaz:
https://doaj.org/article/e34ca2f2440e45e59d5be0c45e98282b
Autor:
Ivan Iliev, Anelia Mavrova, Denitsa Yancheva, Stefan Dimov, Galya Staneva, Alexandrina Nesheva, Iana Tsoneva, Biliana Nikolova
Publikováno v:
Molecules, Vol 28, Iss 17, p 6347 (2023)
Thienopyrimidines are structural analogs of quinazolines, and the creation of new 2-alkyl derivatives of ethyl 4-aminothienopyrimidine-6-carboxylates for the study of their anti-proliferative properties is of great pharmacological interest. Some 2-al
Externí odkaz:
https://doaj.org/article/a98861b198aa476fa32ec63321db6283
Autor:
Kameliya Anichina, Nikolai Georgiev, Nikolay Lumov, Dimitar Vuchev, Galya Popova-Daskalova, Georgi Momekov, Emiliya Cherneva, Rositsa Mihaylova, Anelia Mavrova, Stela Atanasova-Vladimirova, Iskra Piroeva, Denitsa Yancheva
Publikováno v:
Molecules, Vol 28, Iss 13, p 5034 (2023)
[1,3,5]Triazino[1,2-a]benzimidazole-2-amines bearing heterocyclic moiety in 4-position were synthesized. The compounds were characterized by elemental analysis, IR, 1H-NMR, 13C-NMR, and HRMS spectroscopy. The molecular geometry and electron structure
Externí odkaz:
https://doaj.org/article/c04206eec0e34954ad744d86912e6ae5
Autor:
Maria Argirova, Maya Guncheva, Georgi Momekov, Emiliya Cherneva, Rositsa Mihaylova, Miroslav Rangelov, Nadezhda Todorova, Petko Denev, Kameliya Anichina, Anelia Mavrova, Denitsa Yancheva
Publikováno v:
Molecules, Vol 28, Iss 1, p 291 (2022)
1H-benzimidazol-2-yl hydrazones with varying hydroxy and methoxy phenyl moieties were designed. Their effect on tubulin polymerization was evaluated in vitro on porcine tubulin. The compounds elongated the nucleation phase and slowed down the tubulin
Externí odkaz:
https://doaj.org/article/6b22eca3d461470f83ff4698263060ff
Autor:
Anelia Mavrova, Stephan Dimov, Inna Sulikovska, Denitsa Yancheva, Ivan Iliev, Iana Tsoneva, Galya Staneva, Biliana Nikolova
Publikováno v:
Molecules, Vol 27, Iss 10, p 3314 (2022)
Novel 4-amino-thieno[2,3-d]pyrimidine-6-carboxylates substituted at the second position were prepared by cyclocondensation of 2-amino-3-cyano-thiophene and aryl nitriles in an acidic medium. The design of the target compounds was based on structural
Externí odkaz:
https://doaj.org/article/9e492df0cfac45439fee3004da9def18
Autor:
Yancheva, Kameliya Anichina, Nikolai Georgiev, Nikolay Lumov, Dimitar Vuchev, Galya Popova-Daskalova, Georgi Momekov, Emiliya Cherneva, Rositsa Mihaylova, Anelia Mavrova, Stela Atanasova-Vladimirova, Iskra Piroeva, Denitsa
Publikováno v:
Molecules; Volume 28; Issue 13; Pages: 5034
[1,3,5]Triazino[1,2-a]benzimidazole-2-amines bearing heterocyclic moiety in 4-position were synthesized. The compounds were characterized by elemental analysis, IR, 1H-NMR, 13C-NMR, and HRMS spectroscopy. The molecular geometry and electron structure
Publikováno v:
Macedonian Pharmaceutical Bulletin. 68:405-406
Autor:
Jelena Lazarević, Jelena Zvezdanović, Neda Anastassova, Anelia Mavrova, Denitsa Yancheva, Andrija Šmelcerović
Publikováno v:
Acta Facultatis Medicae Naissensis (2022) 39(4):443-450
Introduction: Oxidative stress and resulting lipid peroxidation are involved in numerous pathological conditions. For this reason, the role of antioxidants attracts attention and the radical-scavenging capacity of many natural and synthetic supplemen
Publikováno v:
Acta Facultatis Medicae Naissensis (2020) 37(4):381-386
Antioxidant properties of 2-[2-imino-5-nitro-3-(2-oxo-2-phenylethyl)-2,3-dihydro-1H-benzimidazol1-yl]-1-phenylethanone (compound 1) and 2-(4-fluorobenzylidene)-6-(phenylcarbonyl)[1,3]thiazolo[3,2a]benzimidazol-3(2H)-one (compound 2) were evaluated in
Autor:
Vutchev, D., Marinova, I., Harizanov, R., Blagoeva, V., Massarlieva, A., Anichina, K., Anelia Mavrova
Publikováno v:
Scopus-Elsevier
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=dedup_wf_001::945d18597ddb9c1fdb58a1bb46115213
http://www.scopus.com/inward/record.url?eid=2-s2.0-67549088145&partnerID=MN8TOARS
http://www.scopus.com/inward/record.url?eid=2-s2.0-67549088145&partnerID=MN8TOARS