Zobrazeno 1 - 10
of 11
pro vyhledávání: '"Andrew W Buesking"'
Publikováno v:
Burger's Medicinal Chemistry and Drug Discovery. :1-30
Autor:
Andrew P Combs, Niu Shin, Laurine Galya, James Hall, Sharon Diamond, Kevin Baptiste, Jason Boer, Yan-ou Yang, Kevin J Bowman, Maryanne B Covington, Yanlong Li, Xin He, Daniel Levy, Brent D Douty, Padmaja Polam, David M Burns, Artem Shvartsbart, Eddy W Yue, Rick Sparks, Nikoo Falahatpisheh, Lixin Shao, Stacey Shepard, Andrew W Buesking
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::68d9b46276e455cc32362364091e1119
https://doi.org/10.1021/scimeetings.0c06483
https://doi.org/10.1021/scimeetings.0c06483
Publikováno v:
The Journal of Organic Chemistry. 77:9593-9600
Arylboroxines, which are easily accessed by drying commercially available arylboronic acids, are added to N-(isopropanesulfinyl)ketimines derived from cyclohexanone, N-Boc-piperidin-4-one, and tetrahydropyran-4-one in high yields and with excellent f
Publikováno v:
Organic Letters. 13:3912-3915
The rhodium-catalyzed addition of readily accessible arylboroxines to N-tert-butanesulfinyl ketimines derived from oxetan-3-one, N-Boc-azetidin-3-one, and isatins proceeds in high yields with excellent functional group compatibility. Moreover, high d
Publikováno v:
Organic Letters. 13:964-967
The MgCl(2)-enhanced addition of benzyl zinc reagents to N-tert-butanesulfinyl imines proceeds readily at room temperature to afford the N-tert-butanesulfinyl-protected amine products in good yields and diastereomeric ratios. This method is functiona
Publikováno v:
ChemInform. 45
The enantioselective synthesis of the title compounds from aldimines uses a low catalyst loading.
Autor:
Jonathan A. Ellman, Andrew W. Buesking
Publikováno v:
ChemInform. 45
Asymmetric addition of electron-rich trifluoromethyl ketones to α-sulfinamido trifluoroborates proceed in good yields and diastereoselectivities.
Publikováno v:
The Journal of organic chemistry. 79(8)
The asymmetric borylation of N-tert-butanesulfinyl imines with bis(pinacolato)diboron is achieved using a Cu(II) catalyst and provides access to synthetically useful and pharmaceutically relevant α-amino boronic acid derivatives. The Cu(II)-catalyze
Publikováno v:
ChemInform. 44
A wide range of cyclic amine products is available and the sulfinyl group can be smoothly removed.
Publikováno v:
ChemInform. 42
Arylboroxines with labile functional groups, that are not compatible with Grignard and organolithium reagents, are converted with moderate to excellent yields.