Zobrazeno 1 - 10
of 122
pro vyhledávání: '"Andrea Medeiros"'
Autor:
Cristina Quiroga, Marcelo Incerti, Diego Benitez, Eduardo Manta, Andrea Medeiros, Marcelo A. Comini
Publikováno v:
Frontiers in Chemical Biology, Vol 3 (2024)
Trypanosoma cruzi is the etiologic agent of Chagas’ disease, a debilitating and mortal zoonotic illness that threatens the lives of several millions of people in the American continent. The acute phase is underdiagnosed and there is no curative tre
Externí odkaz:
https://doaj.org/article/53e87e20ac534bea9c4c565a318587a7
Autor:
Estefanía Dibello, Natalia Oddone, Jaime Franco, Tünde-Zita Illyés, Andrea Medeiros, Attila Kiss, Fanni Hőgye, Katalin E. Kövér, László Szilágyi, Marcelo A. Comini
Publikováno v:
International Journal for Parasitology: Drugs and Drug Resistance, Vol 24, Iss , Pp 100529- (2024)
Earlier evidences showed that diglycosyl diselenides are active against the infective stage of African trypanosomes (top hits IC50 0.5 and 1.5 μM) but poorly selective (selectivity index 38-folds vs. murine and human macrohages). For the glycosyl se
Externí odkaz:
https://doaj.org/article/128999b6d1494de5a7542cec9311668e
Autor:
Santiago M. Ruatta, Denis N. Prada Gori, Martín Fló Díaz, Franca Lorenzelli, Karen Perelmuter, Lucas N. Alberca, Carolina L. Bellera, Andrea Medeiros, Gloria V. López, Mariana Ingold, Williams Porcal, Estefanía Dibello, Irina Ihnatenko, Conrad Kunick, Marcelo Incerti, Martín Luzardo, Maximiliano Colobbio, Juan Carlos Ramos, Eduardo Manta, Lucía Minini, María Laura Lavaggi, Paola Hernández, Jonas Šarlauskas, César Sebastian Huerta García, Rafael Castillo, Alicia Hernández-Campos, Giovanni Ribaudo, Giuseppe Zagotto, Renzo Carlucci, Noelia S. Medrán, Guillermo R. Labadie, Maitena Martinez-Amezaga, Carina M. L. Delpiccolo, Ernesto G. Mata, Laura Scarone, Laura Posada, Gloria Serra, Theodora Calogeropoulou, Kyriakos Prousis, Anastasia Detsi, Mauricio Cabrera, Guzmán Alvarez, Adrián Aicardo, Verena Araújo, Cecilia Chavarría, Lucija Peterlin Mašič, Melisa E. Gantner, Manuel A. Llanos, Santiago Rodríguez, Luciana Gavernet, Soonju Park, Jinyeong Heo, Honggun Lee, Kyu-Ho Paul Park, Mariela Bollati-Fogolín, Otto Pritsch, David Shum, Alan Talevi, Marcelo A. Comini
Publikováno v:
Frontiers in Pharmacology, Vol 14 (2023)
Introduction: The identification of chemical compounds that interfere with SARS-CoV-2 replication continues to be a priority in several academic and pharmaceutical laboratories. Computational tools and approaches have the power to integrate, process
Externí odkaz:
https://doaj.org/article/37a7aaacc38c4e40801eaddd5b8743ba
Autor:
Hellen Daghero, Romina Pagotto, Cristina Quiroga, Andrea Medeiros, Marcelo A. Comini, Mariela Bollati-Fogolín
Publikováno v:
Frontiers in Cellular and Infection Microbiology, Vol 13 (2023)
Chagas disease (CD) is a life-threatening illness caused by the parasite Trypanosoma cruzi (T. cruzi). With around seven million people infected worldwide and over 50,000 deaths per year, CD is a major public health issue in Latin America. The main r
Externí odkaz:
https://doaj.org/article/3118ce227d5044f9bf37bf205896847d
Autor:
Ana Carina Cruz de Mello, Felipe Pereira da Silva, Everton Gripa, Andrea Medeiros Salgado, Fabiana Valéria da Fonseca
Publikováno v:
Water, Vol 15, Iss 21, p 3778 (2023)
Tyrosinase enzyme in a crude extract was immobilized in granular activated carbon (GAC) and activated chitosan beads (ACBs), two low-cost supports. It was possible to immobilize up to 70% of the enzymes in GAC under the conditions of 20 g/L support,
Externí odkaz:
https://doaj.org/article/a84a45ba381b42278b115496ca225fae
Publikováno v:
Em Questão, Vol 27, Iss 3, Pp 68-93 (2021)
A mediação cultural e a mediação da informação promovem a disseminação e a apropriação da informação que permeia a esfera social, além de favorecer o acesso à memória e, ao mesmo tempo, potencializar o reconhecimento dos sentimentos de
Externí odkaz:
https://doaj.org/article/1aa1e7d85fa9489eb301e9865007730c
Autor:
Andrea Medeiros, Diego Benítez, Ricarda S. Korn, Vinicius C. Ferreira, Exequiel Barrera, Federico Carrión, Otto Pritsch, Sergio Pantano, Conrad Kunick, Camila I. de Oliveira, Oliver C. F. Orban, Marcelo A. Comini
Publikováno v:
Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 35, Iss 1, Pp 1345-1358 (2020)
Trypanothione synthetase (TryS) produces N1,N8-bis(glutathionyl)spermidine (or trypanothione) at the expense of ATP. Trypanothione is a metabolite unique and essential for survival and drug-resistance of trypanosomatid parasites. In this study, we re
Externí odkaz:
https://doaj.org/article/c7e8b72ceda647528cd31f98709c09d0
Autor:
Olalla Barreiro-Costa, Cristina Quiroga Lozano, Erika Muñoz, Patricio Rojas-Silva, Andrea Medeiros, Marcelo A. Comini, Jorge Heredia-Moya
Publikováno v:
Biomedicines, Vol 10, Iss 8, p 1913 (2022)
Trypanosomiasis and leishmaniasis are neglected infections caused by trypanosomatid parasites. The first-line treatments have many adverse effects, high costs, and are prone to resistance development, hence the necessity for new chemotherapeutic opti
Externí odkaz:
https://doaj.org/article/64574da4e3bc4b7791f1ac40d481e673
Publikováno v:
Navus: Revista de Gestão e Tecnologia, Vol 6, Iss 1, Pp 47-59 (2016)
O presente artigo aborda o tema Gestão do Conhecimento e enfatiza a importância de suas práticas dentro de uma Instituição Escolar em Recife que utiliza a abordagem de ensino e aprendizagem socioconstrutivista. Por meio de estudo de caso, buscou
Externí odkaz:
https://doaj.org/article/6059c374c77f499c8cd5cc8b5455486a
Autor:
Diego Benítez, Andrea Medeiros, Lucía Fiestas, Esteban A Panozzo-Zenere, Franziska Maiwald, Kyriakos C Prousis, Marina Roussaki, Theodora Calogeropoulou, Anastasia Detsi, Timo Jaeger, Jonas Šarlauskas, Lucíja Peterlin Mašič, Conrad Kunick, Guillermo R Labadie, Leopold Flohé, Marcelo A Comini
Publikováno v:
PLoS Neglected Tropical Diseases, Vol 10, Iss 4, p e0004617 (2016)
BACKGROUND:The search for novel chemical entities targeting essential and parasite-specific pathways is considered a priority for neglected diseases such as trypanosomiasis and leishmaniasis. The thiol-dependent redox metabolism of trypanosomatids re
Externí odkaz:
https://doaj.org/article/437dd6f537b74d759f740c4c444491a2