Zobrazeno 1 - 10
of 18
pro vyhledávání: '"Andrea Czompa"'
Autor:
Andrea Czompa, Dóra Bogdán, Balázs Balogh, Eszter Erdei, Patrik Selymes, Attila Csomos, István M. Mándity
Publikováno v:
International Journal of Molecular Sciences, Vol 25, Iss 10, p 5523 (2024)
A new, eco-friendly process utilising the green solvent propylene carbonate (PC) has been developed to perform N-alkylation of N-, O- and/or S-containing heterocyclic compounds. PC in these reactions served as both the reagent and solvent. Importantl
Externí odkaz:
https://doaj.org/article/46f86c7c1f274298a6cac88d8805d37d
Autor:
Krisztina Kónya, Renáta Ferenczi, Andrea Czompa, Attila Kiss-Szikszai, Tibor Kurtán, Sándor Antus
Publikováno v:
ARKIVOC, Vol 2008, Iss 3, Pp 200-210 (2008)
Externí odkaz:
https://doaj.org/article/66409f57849140b9a80981b071e845b7
Autor:
Zoltán Varga, Andrea Czompa, Dóra Bogdán, István M. Mándity, Krisztina Ludányi, Zoltán Mucsi, Balázs László Pásztor, Jennifer Alizadeh Sahar
Publikováno v:
RSC Advances. 9:37818-37824
The Suzuki-Miyaura reaction is one of the most used transformations in drug research. Thus making this reaction more sustainable is of considerable current interest. Here we show that propylene carbonate (PC) can be used as a solvent for the Suzuki-M
Autor:
Miklós Poór, Andrea Czompa, Zsuzsanna Helyes, Violetta Mohos, Ádám Horváth, Dóra Bogdán, Eszter Fliszár-Nyúl, Diána Derdák, Csaba Hetényi, Ruth Deme, Péter Mátyus, Cecília P. Sár, Tamás Kálai, Balázs Zoltán Zsidó, Beáta Lemli, Zelma Faisal
Publikováno v:
Journal of Molecular Liquids. 333:115945
SZV 1287 is our novel multi-target analgesic, which seems to be a promising drug candidate for the treatment of neuropathic pain. Therefore, the drug development process has been started in 2016. Since the pharmacokinetic characterization of a drug c
Autor:
Éva Szőke, Andrea Czompa, Maja Payrits, Péter Mátyus, Zoltán Sándor, Zs. Helyes, Ruth Deme, R. Ludmerczki, Éva Sághy
Publikováno v:
Neuroscience. 324
Transient Receptor Potential Ankyrin 1 and Vanilloid 1 (TRPA1, TRPV1) ion channels expressed on nociceptive primary sensory neurons are important regulators of pain and inflammation. TRPA1 is activated by several inflammatory mediators including form
Autor:
Florin Dan Irimie, Laura Ancua Pop, Péter Mátyus, Csaba Paizs, Andrea Czompa, Elemér Vass, Monica Ioana Toşa
Publikováno v:
Synthesis. 2011:2921-2928
The lipase-catalyzed synthesis of both enantiomers of 3- chloro-1-(4-fluorophenyl)propan-1-ol, 3-chloro-1-(4-iodophe- nyl)propan-1-ol, and 3-chloro-1-phenylpropan-1-ol is described. The procedure is based on the enantiomer-selective acylation of the
Autor:
Valéria Tékus, Bálint Scheich, Attila Mócsai, Janka Zsófia Csepregi, Bálint Botz, Andrea Czompa, Péter Mátyus, Erika Pintér, Ádám Horváth, Zsuzsanna Helyes, János Szolcsányi, Robert Ludmerczki
Publikováno v:
Neuropeptides. 65:130
Autor:
Andrea Czompa, Péter Mátyus, Pál Tapolcsányi, Zsolt Juranyi, Istvan Gacsalyi, Laszlo G. Harsing
Publikováno v:
Current Medicinal Chemistry. 13:1017-1044
The ionotropic glutamate receptor NMDA is allosterically modulated by glycine, a coagonist, its presence is an absolute requirement for receptor activation. The transport of glycine in glutamatergic synapse is carried out by glycine transporter-1 (Gl
Autor:
Pál Tapolcsányi, Laszlo G. Harsing, Julia Timár, Katalin Nagy, Péter Mátyus, Marko Bernadett Martonne, Andrea Czompa, Szabolcs Udvari, Geza Szabo, Ákos Kocsis, Gabriella Zsilla
Publikováno v:
Current pharmaceutical design. 21(17)
We have synthesized a novel series of N-substituted sarcosines, analogues of NFPS ( N -[3-(biphenyl-4- yloxy)-3-(4-fluorophenyl)propyl]- N -methylglycine), as type-1 glycine transporter (GlyT-1) inhibitors. Several compounds incorporated a diazine ri
Publikováno v:
Journal of Heterocyclic Chemistry. 37:991-995
An effective kinetic resolution of hydroxymethylchromanes racemic 2a and 3a has been achieved by means of enantioselective transesterification with vinyl acetate in organic solvents. The alcohols (-)-R-2a and (-)-S-3a were obtained with high optical