Zobrazeno 1 - 6
of 6
pro vyhledávání: '"Andrea Bozzoli"'
Autor:
Steven M, Bromidge, Barbara, Bertani, Manuela, Borriello, Andrea, Bozzoli, Stefania, Faedo, Massimo, Gianotti, Laurie J, Gordon, Matthew, Hill, Valeria, Zucchelli, Jeannette M, Watson, Laura, Zonzini
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 19:2338-2342
8-[2-(4-Aryl-1-piperazinyl)ethyl]-2H-1,4-benzoxazin-3(4H)-ones have been identified as highly potent 5-HT(1A/B/D) receptor antagonists with and without additional SerT activity and a high degree of selectivity over hERG potassium channels. Modulation
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::95b8863b4add2e72b7ea182480d77a3a
https://doi.org/10.1016/j.bmcl.2009.02.056
https://doi.org/10.1016/j.bmcl.2009.02.056
Autor:
Andrea Bozzoli, Gordon J. Kennedy, Antonella Ursini, Marinella Antolini, Chiara Ghiron, Tino Rossi
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 9:1023-1028
A preliminary exploration of analogues of 4,5-bis(3,5-dichlorophenyl)-2-trifluoromethyl-1H-imidazole, 1, as novel antibacterial agents was carried out to determine the basic features of the structure responsible for the observed biological activity.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::10ddf0b3fa7ccb9cf89d8df3c19aa40f
https://doi.org/10.1016/s0960-894x(99)00112-2
https://doi.org/10.1016/s0960-894x(99)00112-2
Publikováno v:
Tetrahedron Letters. 34:3759-3762
Several 3-O-derivatives of (2S,3S)-5-(2-dimethylaminoethyl)-2,3-dihydro-3-hydroxy-2-(4-methoxyphenyl)-1,5-benzothiazepin-4(5H)-one, the parent compound of diltiazem, have been prepared and the M/P conformation ratios have been determined by 1H NMR sp
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::99da72e951828a04a25981f75f817dcf
https://doi.org/10.1016/s0040-4039(00)79221-5
https://doi.org/10.1016/s0040-4039(00)79221-5
Autor:
Gordon J. Kennedy, Tino Rossi, Andrea Bozzoli, Antonella Ursini, Marinella Antolini, Chiara Ghiron
Publikováno v:
ChemInform. 30
A preliminary exploration of analogues of 4,5-bis(3,5-dichlorophenyl)-2-trifluoromethyl-1H-imidazole, 1, as novel antibacterial agents was carried out to determine the basic features of the structure responsible for the observed biological activity.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::d522f2474c855d450f71bea4e4b332e8
https://doi.org/10.1002/chin.199932116
https://doi.org/10.1002/chin.199932116
Autor:
Alessandro Falchi, Barbara Bertani, Daniele Donati, Angelo Pecunioso, Colin Philip Leslie, Romano Di Fabio, Damiano Ghirlanda, Andrea Bozzoli, Manuela Borriello, Simone Spada, Giovanna Rumboldt, Riccardo Giovannini
Publikováno v:
Bioorganicmedicinal chemistry letters. 16(6)
The SAR of a new series of tetrahydrocarbazole derivatives is described: the appropriate decoration of this template led to the identification of a new class of NPY-1 antagonists showing good in vitro potency and a promising in vivo pharmacokinetic p
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b55050e414af1647a895f391267f0689
https://pubmed.ncbi.nlm.nih.gov/16364642
https://pubmed.ncbi.nlm.nih.gov/16364642
Autor:
Andrea Bozzoli, Angelo Pecunioso, Gordon J. Kennedy, Alessandra Pasquarello, Wieslaw M. Kazmierski
Publikováno v:
Bioorganicmedicinal chemistry letters. 10(24)
A library of 80 analogues of the antibacterial compound mureidomycin was prepared using solid-phase chemistry techniques.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::95de20ee35681c694ee79255b82a05a1
https://pubmed.ncbi.nlm.nih.gov/11133085
https://pubmed.ncbi.nlm.nih.gov/11133085