Zobrazeno 1 - 3
of 3
pro vyhledávání: '"Amélie Laversin"'
Autor:
Amélie Laversin, Robin Dufossez, Raphaël Bolteau, Romain Duroux, Séverine Ravez, Sergio Hernandez-Tapia, Martin Fossart, Mathilde Coevoet, Maxime Liberelle, Saïd Yous, Nicolas Lebègue, Patricia Melnyk
Publikováno v:
Molecules, Vol 29, Iss 16, p 3847 (2024)
The adenosine A2A receptor (A2AR) has been identified as a therapeutic target for treating neurodegenerative diseases and cancer. In recent years, we have highlighted the 2-aminoquinazoline heterocycle as an promising scaffold for designing new A2AR
Externí odkaz:
https://doaj.org/article/a703fdddfb0a4440a94b3374b1f753d3
Autor:
Raphaël, Bolteau, Romain, Duroux, Amélie, Laversin, Brandon, Vreulz, Anna, Shiriaeva, Benjamin, Stauch, Gye Won, Han, Vadim, Cherezov, Nicolas, Renault, Amélie, Barczyk, Séverine, Ravez, Mathilde, Coevoet, Patricia, Melnyk, Maxime, Liberelle, Saïd, Yous
Publikováno v:
European journal of medicinal chemistry. 241
The past fifty years have been marked by the surge of neurodegenerative diseases. Unfortunately, current treatments are only symptomatic. Hence, the search for new and innovative therapeutic targets for curative treatments becomes a major challenge.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid________::9dbcd2e0b44d5188113542cf70cf8484
https://pubmed.ncbi.nlm.nih.gov/35933788
https://pubmed.ncbi.nlm.nih.gov/35933788
Autor:
Maxime Liberelle, Philippe Delagrange, Amélie Laversin, Daniel Henri Caignard, Nicolas Lebegue, Mohamed Ettaoussi, Saïd Yous, Marouane Rami, Patricia Melnyk, Brandon Vreulz
Publikováno v:
ChemMedChem. 17(3)
In our constant search for new successors of agomelatine, we report herein a new series of compounds resulting from bioisosteric modulation of the naphthalene ring. The isoquinoline and tetrahydroisoquinoline derivatives were synthesized and pharmaco
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1f47969380e40559daea3163ab647855
https://pubmed.ncbi.nlm.nih.gov/34797951
https://pubmed.ncbi.nlm.nih.gov/34797951