Zobrazeno 1 - 10 of 10 pro vyhledávání: '"Alessio, Barilli"'
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Akademický článek
Identification of positive modulators of TRPM5 channel from a high-throughput screen using a fluorescent membrane potential assay
Autor: Caterina Virginio, Laura Aldegheri, Selena Nola, Daniela Brodbeck, Laurent Brault, Luca F. Raveglia, Alessio Barilli, Mark Sabat, Richard Myers
Publikováno v: SLAS Discovery, Vol 27, Iss 1, Pp 55-64 (2022)
Transient Receptor Potential Melastatin 5 (TRPM5) is an intracellular calcium-activated cation-selective ion channel expressed in a variety of cell types. Dysfunction of this channel has recently been implied in a range of disease states including di
Externí odkaz: https://doaj.org/article/4cf64e986b4845aa93cac6e858d386ee
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2
Tuft cell-derived acetylcholine regulates epithelial fluid secretion
Autor: Tyler E. Billipp, Connie Fung, Lily M. Webeck, Derek B. Sargent, Matthew B. Gologorsky, Margaret M. McDaniel, Darshan N. Kasal, John W. McGinty, Kaitlyn A. Barrow, Lucille M. Rich, Alessio Barilli, Mark Sabat, Jason S. Debley, Richard Myers, Michael R. Howitt, Jakob von Moltke
Publikováno v: bioRxiv
Tuft cells are solitary chemosensory epithelial cells that can sense lumenal stimuli at mucosal barriers and secrete effector molecules to regulate the physiology and immune state of their surrounding tissue. In the small intestine, tuft cells detect
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e7a5077dec2253525a95e08a19d5a318
https://doi.org/10.1101/2023.03.17.533208
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3
Identification of positive modulators of TRPM5 channel from a high-throughput screen using a fluorescent membrane potential assay
Autor: Raveglia Luca Francesco, Richard M. Myers, Caterina Virginio, Mark Sabat, Daniela Brodbeck, Laurent Brault, Selena Nola, Alessio Barilli, Laura Aldegheri
Publikováno v: SLAS Discovery. 27:55-64
Transient Receptor Potential Melastatin 5 (TRPM5) is an intracellular calcium-activated cation-selective ion channel expressed in a variety of cell types. Dysfunction of this channel has recently been implied in a range of disease states including di
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::feac2b5c5ecd8e0a04d427042b52264e
https://doi.org/10.1016/j.slasd.2021.10.004
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6
Enzyme assisted enantioselective synthesis of the alkaloid (+)-aloperine
Autor: Giordano Lesma, Bruno Danieli, Daniele Passarella, Alessandra Silvani, Alessio Barilli, Sergio Riva, Francesca Belinghieri
Publikováno v: Tetrahedron: Asymmetry. 15:2921-2925
The enantioselective synthesis of the lupinine alkaloid (+)-aloperine is described. The synthetic scheme presents three steps that are mediated by enzymes: kinetic resolution, oxidation of a primary alcohol to an aldehyde and oxidation of a secondary
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::62660db776d992f8b49a7b6cea94d970
https://doi.org/10.1016/j.tetasy.2004.06.056
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7
Remote Stereocenter Discrimination in the Enzymatic Resolution of Piperidine-2-ethanol. Short Enantioselective Synthesis of Sedamine and Allosedamine
Autor: Bruno Danieli, Sergio Riva, Giordano Lesma, Marco Angoli, and Alessandra Silvani, Daniele Passarella, Alessio Barilli
Publikováno v: The Journal of Organic Chemistry. 68:9525-9527
Kinetic resolution of N-Boc-piperidine-2-ethanol (2), a case of remote stereocenter discrimination, was accomplished by sequential transesterification mediated by two enzymes, Lipase PS and porcine pancreatic lipase, showing opposite enantioselectivi
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::cb4516f093c5e7923800d3c83a74a74b
https://doi.org/10.1021/jo035215g
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8
Nature-inspired indolyl-2-azabicyclo[2.2.2]oct-7-ene derivatives as promising agents for the attenuation of withdrawal symptoms: synthesis of 20-desethyl-20-hydroxymethyl-11-demethoxyibogaine
Autor: Elaine Elisabetsky, Mirna Bainy Leal, V. M. Linck, Deborah C. Mash, Marisa Martinelli, I. Peretto, Alessandra Silvani, Daniele Passarella, Alessio Barilli, Giordano Lesma, Simon M. N. Efange, Bruno Danieli
Publikováno v: Natural product research. 20(8)
Microwave assisted Diels-Alder cycloaddition of 5-Br-N-benzylpyridinone (2) with methyl acrylate is described to gain an easy access to 7-bromo-2-benzyl-3-oxo-2-aza-5 or 6-carbomethoxy bicyclo[2.2.2]oct-7-enes (3)-(6). The preparation of the ibogaine
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::79110961e704eba92c5a42089f3607c2
https://pubmed.ncbi.nlm.nih.gov/16753910
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10
Short Enantioselective Synthesis of Sedridines, Ethylnorlobelols and Coniine via Reagent-Based Differentiation
Autor: Francesca Belinghieri, Alessandra Silvani, Sergio Riva, Bruno Danieli, Paola Fassi, Daniele Passarella, Alessandro Sacchetti, Alessio Barilli
Publikováno v: 16 (2005): 2225–2229.
info:cnr-pdr/source/autori:Passarella D., Barilli A., Belinghieri F., Fassi P., Riva S., Sacchetti A., Silvani A., Danieli B./titolo:Short enantioselective synthesis of sedridines, ethylnorlobelols and coniine via reagent-based differentiation/doi:/rivista:/anno:2005/pagina_da:2225/pagina_a:2229/intervallo_pagine:2225–2229/volume:16
The preparation of collections of structurally diverse small molecules is a useful tool for studying biology and medicine with chemistry. Herein, we demonstrate the versatility of the pure enantiomers of 2-(2-oxo-ethyl)-piperidine-1-carboxylic acid t
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7ab61fcd0def3c5841456bf6e92fc70e
http://hdl.handle.net/2434/16193
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