Zobrazeno 1 - 5
of 5
pro vyhledávání: '"Alessia Chelini"'
Autor:
Maurizio Anzini, Giulia Chemi, Alessia Chelini, Germano Giuliani, Angela Di Capua, Lorenzo Di Cesare Mannelli, Gianluca Giorgi, Concettina La Motta, Annalisa Reale, Massimo Valoti, Antonietta Rossi, Lidia Sautebin, Simona Pace, Marco Paolino, Elena Lucarini, Andrea Cappelli, Simone Brogi, Alessandro Grillo, Carla Ghelardini
A novel series of 1,5-diarylpyrrol-3-sulfur derivatives (10–12) was synthesized and characterized by NMR and mass spectroscopy and x-ray diffraction. The biological activity of these compounds was evaluated in in vitro and in vivo tests to assess t
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6820359b41e3db181ca2676dc960a721
http://hdl.handle.net/11588/766499
http://hdl.handle.net/11588/766499
Autor:
Gianluca Giorgi, Andrea Cappelli, Simone Brogi, Lorenzo Di Cesare Mannelli, Alessia Chelini, Laura Micheli, Maurizio Anzini, Carla Ghelardini, Mersedeh Farzad, Angela Di Capua, Marco Paolino
LDN-212320 (3) was found to be a potent EAAT2 activator at a translational level, restoring the normal clearance of glutamate and providing neuronal protection. Since the pharmacologic activation of EAAT2 represents a valuable strategy to relieve neu
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d9653c9ccf846aada94f9da593ef4306
http://hdl.handle.net/11365/1012781
http://hdl.handle.net/11365/1012781
Autor:
Lorenzo Ricci, Erminia Leonelli, Gianluca Giorgi, Alessandra Mancini, Angela Di Capua, Antonio Giordani, Alessia Chelini, Jacopo Magistretti, Maurizio Anzini, Germano Giuliani, Marco Paolino, Andrea Cappelli, Simone Brogi, Loretta Castelli, Maria Frosini
Publikováno v:
European journal of medicinal chemistry. 126
Neurodegenerative diseases are disorders related to the degeneration of central neurons that gradually lead to various, severe alterations of cognitive and/or motor functions. Currently, for no such diseases does any pharmacological treatment exist a
Autor:
Maurizio Anzini, Germano Giuliani, Gianfranco Caselli, Maria Cristina Menziani, Antonio Giordani, Andrea Cappelli, Chiara Sabatini, Marco Paolino, Alessia Chelini, Laura Mennuni, Chiara Nannicini, Francesco Makovec, Gianluca Giorgi, Salvatore Vomero
Two new fluorophenylindenone derivatives were designed as potential p38α MAPK modulators by preserving the key interactions of the vicinal pyridine/fluorophenyl pharmacophore with the enzyme protein. Interestingly, these two fluorophenylindenone iso
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::11b3d971c122757490d6f923b3acf13c
http://hdl.handle.net/11365/998341
http://hdl.handle.net/11365/998341
Autor:
Maurizio Anzini, Alessia Chelini, Alessandra Mancini, Andrea Cappelli, Maria Frosini, Lorenzo Ricci, Massimo Valoti, Jacopo Magistretti, Loretta Castelli, Antonio Giordani, Francesco Makovec, Salvatore Vomero
Publikováno v:
Journal of Medicinal Chemistry; Jan2010, Vol. 53 Issue 2, p734-744, 11p