Zobrazeno 1 - 7
of 7
pro vyhledávání: '"Alan, Futran"'
Autor:
Emily C. Cherney, Liping Zhang, Julian Lo, Tram Huynh, Donna Wei, Vijay Ahuja, Claude Quesnelle, Gary L. Schieven, Alan Futran, Gregory A. Locke, Zeyu Lin, Laura Monereau, Charu Chaudhry, Jordan Blum, Sha Li, Mark Fereshteh, Bifang Li-Wang, Sanjeev Gangwar, Chin Pan, Colin Chong, Xiao Zhu, Shana L. Posy, John S. Sack, Ping Zhang, Max Ruzanov, Mary Harner, Fahad Akhtar, Gretchen M. Schroeder, Gregory Vite, Brian Fink
Publikováno v:
Journal of Medicinal Chemistry. 65:3518-3538
Autor:
Shivam Rai, Jan Stetka, MARC Usart, Hui Hao-Shen, Young Park, Remie Houston, Anthony R. Martinez Benitez, Matthew Wereski, Emily Guzzardi, Sonali Persaud, Hailey Ramzan, Alan Futran, Charley Xu, Jeremy Greenwood, Sayan Mondal, Craig Masse, Ross L. Levine, Radek C. Skoda, Andrew Dunbar
Publikováno v:
Blood. 140:6722-6723
Autor:
John Morrison, Steven Sheriff, Mark D. Wittman, Gregory A. Locke, Bradley C. Pearce, Erika M. V. Araujo, Andrew P. Degnan, Christopher W. Allard, Dan You, Xin Li, Kurt Zimmermann, Anwar Murtaza, Benjamin M. Johnson, Caitlyn Stromko, Jinqi Liu, Gregory D. Vite, Godwin Kwame Kumi, Karen E. Parrish, Alan Futran, Johnson Walter Lewis
Publikováno v:
ACS Medicinal Chemistry Letters
While the discovery of immune checkpoint inhibitors has led to robust, durable responses in a range of cancers, many patients do not respond to currently available therapeutics. Therefore, an urgent need exists to identify alternative mechanisms to a
Autor:
Emily C, Cherney, Liping, Zhang, Julian, Lo, Tram, Huynh, Donna, Wei, Vijay, Ahuja, Claude, Quesnelle, Gary L, Schieven, Alan, Futran, Gregory A, Locke, Zeyu, Lin, Laura, Monereau, Charu, Chaudhry, Jordan, Blum, Sha, Li, Mark, Fereshteh, Bifang, Li-Wang, Sanjeev, Gangwar, Chin, Pan, Colin, Chong, Xiao, Zhu, Shana L, Posy, John S, Sack, Ping, Zhang, Max, Ruzanov, Mary, Harner, Fahad, Akhtar, Gretchen M, Schroeder, Gregory, Vite, Brian, Fink
Publikováno v:
Journal of medicinal chemistry. 65(4)
The identification of agonists of the stimulator of interferon genes (STING) pathway has been an area of intense research due to their potential to enhance innate immune response and tumor immunogenicity in the context of immuno-oncology therapy. Ini
Autor:
Joe Baldick, Jonathan Lippy, Peter Chase, Austin Crithary, Sha Li, Jing Chen, Alan Futran, Brian J. Arey, Alex Wolicki, Kylie Fogarty
Publikováno v:
SLAS discovery : advancing life sciences RD. 26(3)
We previously developed a panel of one-step real-time quantitative reverse transcription PCR (one-step qRT-PCR; hereafter referred to as qRT-PCR) assays to assess compound efficacy. However, these high-cost, conventional qRT-PCR manual assays are not
Autor:
Liping Fang, Takao Suzuki, Kristian Jensen, Mats A. Svensson, Robert Pelleltier, Jeffrey A. Bell, Zef Konst, Hamish Wright, Wayne Tang, Katherine Amberg-Johnson, Shuping Xu, Xianhai Huang, Karen Dingley, Yan Zhang, Heng Qian, Markus K. Dahlgren, Michael Trzoss, Alan Futran, Karen Akinsanya, Xiaoxiao Yang, Sarah Boyce, Saidi He, Li Xing, Jiayi Xu, Tao Guo, David Madge, Tao Lu, Heidi Koldsoe, Fang-Yu Lin, Zhaowu Xu, Jie Xu, Engin Yapici
Publikováno v:
Cancer Research. 81:1338-1338
Introduction: Ubiquitin-specific protease 7 (USP7) is a deubiquitinase that regulates several proteins involved in cell cycle, DNA repair, genomic stability, and epigenetics and has been implicated in cancer progression. A key substrate of USP7 is MD
Investigations of Pd-Catalyzed ArX Coupling Reactions Informed by Reaction Progress Kinetic Analysis
Autor:
Jinu S. Mathew, Donna G. Blackmond, Alan Futran, Martin Klussmann, Hiroshi Iwamura, Fernando E. Valera, Emma Anna Carolina Emanuelsson
Publikováno v:
ChemInform. 37
This Perspective highlights how the methodology of reaction progress kinetic analysis can provide a rapid and comprehensive kinetic profile of complex catalytic reaction networks under synthetically relevant conditions in a fraction of the number of