Synthesis and evaluation of 2,4,5-trisubstitutedthiazoles as carbonic anhydrase-III inhibitors.

Autor: Al-Jaidi BA; Department of Pharmaceutical Sciences, Faculty of Pharmacy, Philadelphia University, Amman, Jordan.; Faculty of Pharmacy, Yarmouk University, Irbid, Jordan., Deb PK; Department of Pharmaceutical Sciences, Faculty of Pharmacy, Philadelphia University, Amman, Jordan., Telfah ST; Department of Pharmaceutical Sciences, Faculty of Pharmacy, Philadelphia University, Amman, Jordan., Dakkah AN; Department of Pharmaceutical Sciences, Faculty of Pharmacy, Philadelphia University, Amman, Jordan., Bataineh YA; Department of Pharmaceutical Sciences, Faculty of Pharmacy, Philadelphia University, Amman, Jordan., Khames Aga QAA; Department of Pharmaceutical Sciences, Faculty of Pharmacy, Philadelphia University, Amman, Jordan., Al-Dhoun MA; Department of Pharmaceutical Sciences, Faculty of Pharmacy, Philadelphia University, Amman, Jordan., Ahmad Al-Subeihi AA; Faculty of Pharmacy, Amman Arab University, Amman, Jordan., Odetallah HM; Department of Pharmaceutical Sciences, Faculty of Pharmacy, Philadelphia University, Amman, Jordan., Bardaweel SK; Department of Pharmaceutical Sciences, School of Pharmacy, University of Jordan, Amman, Jordan., Mailavaram R; Pharmaceutical Chemistry Division, Sri Vishnu College of Pharmacy, Bhimavaram, India., Venugopala KN; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa, Saudi Arabia.; Department of Biotechnology and Food Technology, Durban University of Technology, Durban, South Africa., Nair AB; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa, Saudi Arabia.

Publikováno v: Journal of enzyme inhibition and medicinal chemistry [J Enzyme Inhib Med Chem] 2020 Dec; Vol. 35 (1), pp. 1483-1490.

Cytotoxicity and Antimycobacterial Properties of Pyrrolo[1,2- a ]quinoline Derivatives: Molecular Target Identification and Molecular Docking Studies.

Autor: Venugopala KN; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia.; Department of Biotechnology and Food Technology, Durban University of Technology, Durban 4001, South Africa., Uppar V; Department of Chemistry, School of Basic Science, Rani Channamma University, Belagavi 591156, India., Chandrashekharappa S; Institute for Stem Cell Biology and Regenerative Medicine, National Center for Biological Sciences (NCBS), Tata Institute of Fundamental Research (TIFR), Gandhi Krishi Vignana Kendra (GKVK) Campus, Bangalore 560065, India., Abdallah HH; Chemistry Department, College of Education, Salahaddin University, Erbil 44001, Iraq., Pillay M; Department of Microbiology, National Health Laboratory Services, KZN Academic Complex, Inkosi Albert Luthuli Central Hospital, Durban 4001, South Africa., Deb PK; Faculty of Pharmacy, Philadelphia University, Amman 19392, Jordan., Morsy MA; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia.; Department of Pharmacology, Faculty of Medicine, Minia University, El-Minia 61511, Egypt., Aldhubiab BE; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia., Attimarad M; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia., Nair AB; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia., Sreeharsha N; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia., Tratrat C; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia., Yousef Jaber A; Faculty of Pharmacy, Philadelphia University, Amman 19392, Jordan., Venugopala R; Department of Public Health Medicine, University of KwaZulu-Natal, Howard College Campus, Durban 4001, South Africa., Mailavaram RP; Department of Pharmaceutical Chemistry, Shri Vishnu College of Pharmacy, Vishnupur, Bhimavaram 534 202, India., Al-Jaidi BA; Faculty of Pharmacy, Yarmouk University, Irbid 21163, Jordan., Kandeel M; Department of Biomedical Sciences, College of Veterinary Medicine, King Faisal University, Al-Ahsa 31982, Saudi Arabia.; Department of Pharmacology, Faculty of Veterinary Medicine, Kafrelsheikh University, Kafrelsheikh 33516, Egypt., Haroun M; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia., Padmashali B; Department of Chemistry, School of Basic Science, Rani Channamma University, Belagavi 591156, India.

Publikováno v: Antibiotics (Basel, Switzerland) [Antibiotics (Basel)] 2020 May 07; Vol. 9 (5). Date of Electronic Publication: 2020 May 07.