Zobrazeno 1 - 10
of 13
pro vyhledávání: '"Akihisa Tokuda"'
Autor:
Hikari Yamamoto, Yasuyuki Nagumo, Yukiko Ishikawa, Yoko Irukayama-Tomobe, Yukiko Namekawa, Tsuyoshi Nemoto, Hiromu Tanaka, Genki Takahashi, Akihisa Tokuda, Tsuyoshi Saitoh, Hiroshi Nagase, Hiromasa Funato, Masashi Yanagisawa
Publikováno v:
PLoS ONE, Vol 17, Iss 7, p e0271901 (2022)
Acquired loss of hypothalamic orexin (hypocretin)-producing neurons causes the chronic sleep disorder narcolepsy-cataplexy. Orexin replacement therapy using orexin receptor agonists is expected as a mechanistic treatment for narcolepsy. Orexins act o
Externí odkaz:
https://doaj.org/article/eca4900ef18e47168c9b01a29a3ececa
Autor:
Kenta Maeda, Sayaka Ohrui, Akihisa Tokuda, Yasuyuki Nagumo, Naoshi Yamamoto, Ryuji Tanimura, Tsuyoshi Saitoh, Noriki Kutsumura, Hiroshi Nagase
Publikováno v:
Organic Letters. 25:3407-3411
Autor:
Keita Iio, Kao Hashimoto, Yasuyuki Nagumo, Mao Amezawa, Taisei Hasegawa, Naoshi Yamamoto, Noriki Kutsumura, Katsuhiko Takeuchi, Yukiko Ishikawa, Hikari Yamamoto, Akihisa Tokuda, Tetsu Sato, Yasuo Uchida, Asuka Inoue, Ryuji Tanimura, Masashi Yanagisawa, Hiroshi Nagase, Tsuyoshi Saitoh
Publikováno v:
Journal of Medicinal Chemistry. 66:5453-5464
Autor:
Noriki Kutsumura, Tsuyoshi Saitoh, Jumpei Horiuchi, Yukiko Ishikawa, Emi Hasegawa, Yasuyuki Nagumo, Masashi Yanagisawa, Takeshi Sakurai, Ryuji Tanimura, Hiroaki Gouda, Naoshi Yamamoto, Yasuhiro Ogawa, Akihisa Tokuda, Tetsu Sato, Yoko Irukayama-Tomobe, Mao Amezawa, Hiroshi Nagase, Ryuichiro Oshita, Yasuo Uchida
Structurally diverse small compounds are utilized to obtain hit compounds that have suitable pharmacophores in appropriate three-dimensional conformations for the target drug receptors. We have focused on the 1,3,5-trioxazatriquinane skeleton, which
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::f4079393b5fe25c5fc1566ec1c12834a
https://doi.org/10.33774/chemrxiv-2021-08md1
https://doi.org/10.33774/chemrxiv-2021-08md1
Autor:
Tsuyoshi Saitoh, Mao Amezawa, Jumpei Horiuchi, Yasuyuki Nagumo, Naoshi Yamamoto, Noriki Kutsumura, Ryuichiro Ohshita, Akihisa Tokuda, Yoko Irukayama-Tomobe, Yasuhiro Ogawa, Yukiko Ishikawa, Emi Hasegawa, Takeshi Sakurai, Yasuo Uchida, Tetsu Sato, Hiroaki Gouda, Ryuji Tanimura, Masashi Yanagisawa, Hiroshi Nagase
Structurally diverse small compounds are utilized to obtain hit compounds that have suitable pharmacophores in appropriate three-dimensional conformations for the target drug receptors. We have focused on the 1,3,5-trioxazatriquinane skeleton, which
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::dd0571529b5d14b8ad54e10a712a84a9
https://doi.org/10.26434/chemrxiv-2021-08md1
https://doi.org/10.26434/chemrxiv-2021-08md1
Autor:
Noriki Kutsumura, Tsuyoshi Saitoh, Akihisa Tokuda, Yasuyuki Nagumo, Ryoji Kise, Kao Hashimoto, Hirokazu Mizoguchi, Hiroshi Nagase, Asuka Inoue, Keita Iio, Naoshi Yamamoto
Publikováno v:
Bioorganicmedicinal chemistry letters. 56
Mas-related G protein-coupled receptor X2 (MRGPRX2) mediates the itch response in neurons and is involved in atopic dermatitis (AD)-associated inflammation and itch. Potent and MRGPRX2-selective ligands are essential to an understanding of the detail
Autor:
Vladimir Hutanu, Taka-hisa Arima, Motohiro Suzuki, Katsuya Inoue, Hiroyuki Ohsumi, Kazuki Ohishi, Naomi Kawamura, Kazuhisa Kakurai, Y. Miyamoto, Takayasu Hanashima, Javier Campo, T. Koyama, Yusuke Kousaka, J. Suzuki, A. Sera, Akiko Nakao, Akihisa Tokuda, Jun Akimitsu
Publikováno v:
Zaguán. Repositorio Digital de la Universidad de Zaragoza
instname
Digital.CSIC. Repositorio Institucional del CSIC
instname
Digital.CSIC. Repositorio Institucional del CSIC
This work was supported by JSPS KAKENHI Grants No. 25220803, No. 25390139, No. 26108719, No. 15H03680, No. 15H05885, No. 15H05886, No. 16KK0102, 17H02912, No. 17H02767, and No. 17H02815. K.K. acknowledges the support by the Helmholtz International Fe
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d38db0b5fd70037e04e640ac09fd873e
http://zaguan.unizar.es/record/75681
http://zaguan.unizar.es/record/75681
Autor:
Masaki Takata, Naomi Kawamura, Yusuke Kousaka, Hiroyuki Ohsumi, Taka-hisa Arima, Jun Akimitsu, Soshi Takeshita, Akihisa Tokuda, Motohiro Suzuki
Publikováno v:
Angewandte Chemie International Edition. 52:8718-8721
Autor:
Hideto Tsuji, Xiaoli Sun, Akihisa Tokuda, T. Nakatani, Isao Takahashi, Shouke Yan, Yusuke Oji, Yukihiro Ozaki
Publikováno v:
Macromolecules. 45:2485-2493
Blends of poly[(R)-3-hydroxybutyrate] (PHB) with poly(l-lactide acid) (PLLA) were prepared to study the crystallization behavior of PHB in the blends. To investigate the effect of molar mass of PLLA on the crystallization of PHB, two types of PLLA wi
Autor:
Akihisa Tokuda, Hidenori Takagi, Taka-hisa Arima, Kenya Ohgushi, Soshi Takeshita, Hiroyuki Ohsumi, Kunihisa Sugimoto, Jun-ichi Yamaura, Masaki Takata
Publikováno v:
Physical Review Letters. 110
We performed resonant x-ray diffraction experiments at the L absorption edges for the post-perovskite-type compound CaIrO(3) with a (t(2g))^{5} electronic configuration. By observing the magnetic signals, we could clearly see that the magnetic struct