Zobrazeno 1 - 10
of 18
pro vyhledávání: '"Adriana Ferreira Lopes Vilela"'
Autor:
Cintia Duarte de Freitas Milagre, Bruno Sergio do Amaral, João Marcos Batista Junior, Adriana Ferreira Lopes Vilela, Carmen Lúcia Cardoso, Humberto Marcio Santos Milagre
Publikováno v:
Eclética Química, Vol 47, Iss 2, Pp 17-35 (2022)
A chemoenzymatic approach for the synthesis of Alpha-N-heterocyclic ethyl- and phenylacetamides, levetiracetam analogs, is described. Eight nitrile substrates were prepared through the N-alkylation of heterocycles (2-pyrrolidinone, 2-piperidinone, 2-
Externí odkaz:
https://doaj.org/article/9e099bfe16f4408cb32a022310f9b528
Publikováno v:
Frontiers in Chemistry, Vol 9 (2021)
We have developed a dual enzymatic system assay involving liquid chromatography-mass spectrometry (LC–MS) to screen AChE and BACE1 ligands. A fused silica capillary (30 cm × 0.1 mm i.d. × 0.362 mm e.d.) was used as solid support. The co-immobiliz
Externí odkaz:
https://doaj.org/article/089edfc8aa5d4ecb9ebf3dde1c4d4078
Autor:
Vilma Menezes de Jesus Prado, Raphael Amancio de Jesus, Julio Manoel Andrade Oliveira, Arie Fitzgerald Blank, Daniel Pereira Bezerra, Milena Botelho Pereira Soares, Valdenizia Rodrigues Silva, Luciano de Souza Santos, Carmen Lúcia Cardoso, Adriana Ferreira Lopes Vilela, Paulo Cesar de Lima Nogueira, Valéria Regina de Souza Moraes
Publikováno v:
Repositório Institucional da USP (Biblioteca Digital da Produção Intelectual)
Universidade de São Paulo (USP)
instacron:USP
Universidade de São Paulo (USP)
instacron:USP
Publikováno v:
Frontiers in Chemistry, Vol 9 (2021)
Frontiers in Chemistry
Repositório Institucional da USP (Biblioteca Digital da Produção Intelectual)
Universidade de São Paulo (USP)
instacron:USP
Frontiers in Chemistry
Repositório Institucional da USP (Biblioteca Digital da Produção Intelectual)
Universidade de São Paulo (USP)
instacron:USP
We have developed a dual enzymatic system assay involving liquid chromatography-mass spectrometry (LC–MS) to screen AChE and BACE1 ligands. A fused silica capillary (30 cm × 0.1 mm i.d. × 0.362 mm e.d.) was used as solid support. The co-immobiliz
Autor:
Carmen Lúcia Cardoso, Claudia Seidl, Juliana Maria Lima, Gabriel Mazzi Leme, Adriana Ferreira Lopes Vilela
Publikováno v:
Analytica Chimica Acta. 1072:81-86
This work describes a new simultaneous on-flow dual parallel enzyme assay based on immobilized enzyme reactors (ICERs) with mass spectrometry detection. The novelty of this work relies on the fact that two different enzymes can be screened at the sam
Publikováno v:
Repositório Institucional da USP (Biblioteca Digital da Produção Intelectual)
Universidade de São Paulo (USP)
instacron:USP
Universidade de São Paulo (USP)
instacron:USP
This study presents a rapid and simple method to screen and detect new drugs to treat Alzheimer’s disease. The method uses a test system based on an immobilized acetylcholinesterase from Electrophorus electricus (AChE). The optimal AChE immobilized
Autor:
Maria C. M. Young, Alana E. Honório, Vanderlan da Silva Bolzani, Paulo Michel Pinheiro Ferreira, Regina Maria Barretto Cicarelli, Fernando Rogério Pavan, Juliana R. Gubiani, Vanessa Mara Chapla, Adriana Ferreira Lopes Vilela, Carmen Lúcia Cardoso, Angela Regina Araújo
Publikováno v:
Repositório Institucional da USP (Biblioteca Digital da Produção Intelectual)
Universidade de São Paulo (USP)
instacron:USP
Scopus
Repositório Institucional da UNESP
Universidade Estadual Paulista (UNESP)
instacron:UNESP
Universidade de São Paulo (USP)
instacron:USP
Scopus
Repositório Institucional da UNESP
Universidade Estadual Paulista (UNESP)
instacron:UNESP
Made available in DSpace on 2020-12-12T02:18:32Z (GMT). No. of bitstreams: 0 Previous issue date: 2020-10-01 Coordenação de Aperfeiçoamento de Pessoal de Nível Superior (CAPES) Three new oxygenated cyclohexanoids, namely, speciosin U (1), specios
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8bc956643b82a3a1d2cc7fa2cb75ce83
Autor:
Dulce Helena Siqueira Silva, Carmen Lúcia Cardoso, Angela Regina Araújo, Helori Vanni Domingos, Claudia Seidl, Raymond J. Andersen, João M. Batista, Adriana Ferreira Lopes Vilela, Letícia V. Costa-Lotufo, Rebeca Previate Medina
Publikováno v:
Scopus
Repositório Institucional da UNESP
Universidade Estadual Paulista (UNESP)
instacron:UNESP
Repositório Institucional da USP (Biblioteca Digital da Produção Intelectual)
Universidade de São Paulo (USP)
instacron:USP
Scientific Reports
Scientific Reports, Vol 9, Iss 1, Pp 1-11 (2019)
Repositório Institucional da UNESP
Universidade Estadual Paulista (UNESP)
instacron:UNESP
Repositório Institucional da USP (Biblioteca Digital da Produção Intelectual)
Universidade de São Paulo (USP)
instacron:USP
Scientific Reports
Scientific Reports, Vol 9, Iss 1, Pp 1-11 (2019)
A chemical study of the EtOAc extract of Nemania bipapillata (AT-05), an endophytic fungus isolated from the marine red alga Asparagopsis taxiformis - Falkenbergia stage, led to the isolation of five new botryane sesquiterpenes, including the diaster
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::bbf55d68e6d81a006592e51ca9b4c55b
Publikováno v:
Analytical Methods. 9:2189-2196
The enzyme β-secretase1 (BACE1) is an aspartyl protease that initiates the cleavage of the Aβ amyloid precursor protein (APP), to generate and aggregate β-amyloid (Aβ) peptides. Aggregates of Aβ peptides are implicated in the pathogenesis of Alz
Publikováno v:
Biblioteca Digital de Teses e Dissertações da USP
Universidade de São Paulo (USP)
instacron:USP
Universidade de São Paulo (USP)
instacron:USP
As enzimas, acetilcolinesterase (AChE) e ?-secretase1 (BACE1), são alvos validados para o tratamento da Doença de Alzheimer (DA) uma vez que atuam no sistema nervoso central contribuindo para o avanço da doença. Neste contexto, o interesse por in
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c7a1a6d62c7b64e7c8968e3867571720
https://doi.org/10.11606/t.59.2018.tde-06072018-110632
https://doi.org/10.11606/t.59.2018.tde-06072018-110632