Zobrazeno 1 - 3
of 3
pro vyhledávání: '"Adrian Fretland"'
Autor:
Terry, Podoll, Paul G, Pearson, Allard, Kaptein, Jerry, Evarts, Gerjan, de Bruin, Maaike, Emmelot-van Hoek, Anouk, de Jong, Bart, van Lith, Hao, Sun, Stephen, Byard, Adrian, Fretland, Niels, Hoogenboom, Tjeerd, Barf, J Greg, Slatter
Publikováno v:
Journal of Pharmacology and Experimental Therapeutics. 384:173-186
Acalabrutinib is a covalent Bruton tyrosine kinase (BTK) inhibitor approved for relapsed/refractory mantle cell lymphoma and chronic lymphocytic leukemia/small lymphocytic lymphoma. A major metabolite of acalabrutinib (M27, ACP-5862) was observed in
Autor:
Maayan Levy, Gino Ferraro, Li Li, Yongshuai Han, Lilian Varricchio, Sara Fournier, Xiuli An, Ronald Hoffman, Adrian Fretland, Anne Roulston, Yelena Ginzburg
Publikováno v:
Blood. 140:8194-8195
Autor:
Micaela B, Reddy, Alyson, Connor, Barbara J, Brennan, Peter N, Morcos, Amy, Zhou, Pamela, McLawhon, Adrian, Fretland, Philip, Evans, Patrick, Smith, Jonathan Q, Tran
Publikováno v:
Biopharmaceuticsdrug disposition. 32(5)
Danoprevir, a potent, selective inhibitor of HCV NS3/4A protease, has a short half-life in humans. Therefore, the feasibility of a controlled release (CR) formulation to allow less frequent dosing was investigated using experimental approaches and ph